ECSP18019949A - CYCLIC DINUCLEOTIDE COMPOUNDS AS STING AGONISTS - Google Patents
CYCLIC DINUCLEOTIDE COMPOUNDS AS STING AGONISTSInfo
- Publication number
- ECSP18019949A ECSP18019949A ECIEPI201819949A ECPI201819949A ECSP18019949A EC SP18019949 A ECSP18019949 A EC SP18019949A EC IEPI201819949 A ECIEPI201819949 A EC IEPI201819949A EC PI201819949 A ECPI201819949 A EC PI201819949A EC SP18019949 A ECSP18019949 A EC SP18019949A
- Authority
- EC
- Ecuador
- Prior art keywords
- cyclic dinucleotide
- sting agonists
- compounds
- dinucleotide compounds
- general formula
- Prior art date
Links
Abstract
Se proporciona una clase de compuestos policíclicos de fórmula general (I), de fórmula general (I'), o de fórmula general (II''), en las que Base1 , Base2 , Y, Ya , Xa , Xa1, Xb , Xb1, Xc , Xc1 , X d , Xd1, R1 , R1a, R2 , R2a, R3 , R4 , R4a, R5 , R6 , R6a, R7 , R7a, R8 y R8a se definen en el presente documento, que pueden ser útiles como inductores de la producción de interferones de tipo I, específicamente como agentes activos de STING. También se proporcionan procesos de síntesis y de uso de compuestos.A class of polycyclic compounds of general formula (I), general formula (I '), or general formula (II' ') is provided, wherein Base1, Base2, Y, Ya, Xa, Xa1, Xb, Xb1 , Xc, Xc1, X d, Xd1, R1, R1a, R2, R2a, R3, R4, R4a, R5, R6, R6a, R7, R7a, R8 and R8a are defined herein, which may be useful as inducers of the production of type I interferons, specifically as active agents of STING. Processes for synthesis and use of compounds are also provided.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201562204677P | 2015-08-13 | 2015-08-13 |
Publications (1)
Publication Number | Publication Date |
---|---|
ECSP18019949A true ECSP18019949A (en) | 2018-07-31 |
Family
ID=60451227
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ECIEPI201819949A ECSP18019949A (en) | 2015-08-13 | 2018-03-13 | CYCLIC DINUCLEOTIDE COMPOUNDS AS STING AGONISTS |
Country Status (2)
Country | Link |
---|---|
AR (1) | AR105683A1 (en) |
EC (1) | ECSP18019949A (en) |
-
2016
- 2016-08-11 AR ARP160102472A patent/AR105683A1/en unknown
-
2018
- 2018-03-13 EC ECIEPI201819949A patent/ECSP18019949A/en unknown
Also Published As
Publication number | Publication date |
---|---|
AR105683A1 (en) | 2017-11-01 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
DOP2018000046A (en) | CYCLIC DINUCLEOTIDE COMPOUNDS AS STING AGONISTS | |
NI201900029A (en) | BENZO [b] THIOPHENE COMPOUNDS AS STING AGONISTS | |
CR20150183A (en) | DERIVATIVES OF 5-FENOXI-3H-PIRIMIDIN-4-ONA AND ITS USE AS INHIBITORS OF HIV REVERSE TRANSCRIPT | |
CO2019010023A2 (en) | Modified cyclic dinucleotide compounds | |
NI201800023A (en) | BETA-AMINO ACID ESTER PHOSPHODIAMIDE ANTIVIRAL COMPOUNDS | |
PE20161073A1 (en) | AMINO-HETEROARYL-BENZAMIDES AS KINASE INHIBITORS | |
PE20160524A1 (en) | THERAPEUTICALLY ACTIVE COMPOUNDS AND THEIR METHODS OF USE | |
CL2016001509A1 (en) | Crystal forms of antiviral sofosbuvir analogs | |
CO2017010894A2 (en) | Innovative mixed body of iron compound and graphene oxide | |
CO6541645A2 (en) | INDOL COMPOUNDS AND THEIR PHARMACEUTICAL USE | |
AR076810A1 (en) | ANTI-BANERIGEN COMPOUNDS OF AMINO PYRIMIDINE | |
AR072016A1 (en) | ISOXAZOL DERIVATIVES THAT WORK AS POTENTIALS OF GLUTAMATE RECEIVERS | |
CL2018000786A1 (en) | Compuestos derivados de pirrolo[2,3-d]pirimidina, inhibidores de dyrk1a; proceso de preparacion; composicion farmaceutica; combinacion farmaceutica; uso para tratar el cancer, trastornos neurodegenerativos, o trastornos metabolicos. | |
PE20181346A1 (en) | IMIDAZO [4,5-C] QUINOLIN-2-ONA COMPOUNDS AND THEIR USE IN THE TREATMENT OF CANCER | |
NI201200146A (en) | NON-NUCLEOSIDIC INHIBITORS OF REVERSE TRANSCRIPTASE | |
CL2017001001A1 (en) | Carbazaol derivatives | |
PA8797701A1 (en) | DERIVATIVES OF QUINAZOLINADIONA, ITS PREPARATION AND ITS THERAPEUTIC APPLICATIONS | |
CR20160454A (en) | CHROMENE AND 1.1 a, 2.7b — TETRAHYDROCICLOPROPA [C] CHROME PIRIDOPIRAZINADIONAS NOVEDOSAS | |
PE20180116A1 (en) | HETEROCICLYLMETIL-THENURACILO AS AGONISTS OF THE ADENOSINE A2b RECEPTOR | |
CO6150181A2 (en) | COMPOUND 6- (BENCILO REPLACED WITH HETEROCICLE) -4-OXOQUINOLINE AND ITS USE AS AN INTEGRASA HIV INHIBITOR | |
UY33993A (en) | MACROCYCLIC ANALOG OF SANGLIFERINA AND ITS PRODUCTION METHOD | |
DOP2019000100A (en) | DERIVATIVES OF NAFTIRIDINONE AND ITS USE IN THE TREATMENT OF ARRITMIA | |
CR20180615A (en) | NEW DERIVATIVES OF [1,2,3] TRIAZOL [4,5-D] PYRIMIDINE | |
CL2020003248A1 (en) | N-substituted tetrahydrothienopyridine derivatives and their uses | |
ECSP18019949A (en) | CYCLIC DINUCLEOTIDE COMPOUNDS AS STING AGONISTS |