ECSP034663A - PIRAZOL COMPOUNDS USED AS PROTEIN QUINASA INHIBITORS - Google Patents
PIRAZOL COMPOUNDS USED AS PROTEIN QUINASA INHIBITORSInfo
- Publication number
- ECSP034663A ECSP034663A ECSP034663A ECSP034663A EC SP034663 A ECSP034663 A EC SP034663A EC SP034663 A ECSP034663 A EC SP034663A EC SP034663 A ECSP034663 A EC SP034663A
- Authority
- EC
- Ecuador
- Prior art keywords
- compounds used
- inhibitors
- protein
- compounds
- pirazol
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title abstract 4
- 239000003112 inhibitor Substances 0.000 title abstract 2
- 102000004169 proteins and genes Human genes 0.000 title 1
- 108090000623 proteins and genes Proteins 0.000 title 1
- 108090000461 Aurora Kinase A Proteins 0.000 abstract 2
- 201000010099 disease Diseases 0.000 abstract 2
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 2
- 102000004000 Aurora Kinase A Human genes 0.000 abstract 1
- 102100032311 Aurora kinase A Human genes 0.000 abstract 1
- 206010028980 Neoplasm Diseases 0.000 abstract 1
- 102000001253 Protein Kinase Human genes 0.000 abstract 1
- 229940045988 antineoplastic drug protein kinase inhibitors Drugs 0.000 abstract 1
- 201000011510 cancer Diseases 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 108060006633 protein kinase Proteins 0.000 abstract 1
- 239000003909 protein kinase inhibitor Substances 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
La presente invención se refiere a la química medicinal y a los compuestos que son inhibidores protein quinasas, composiciones que contienen dichos compuestos y métodos de uso. Más particularmente, esta invención se refiere a compuestos que son inhibidores de Aurora -2 protein quinasas. La invención además se refiere a métodos para tratar enfermedades asociadas con protein quinasas, especialmente enfermedades asociadas con Aurora-2, tal como el cáncerThe present invention relates to medicinal chemistry and compounds that are protein kinase inhibitors, compositions containing said compounds and methods of use. More particularly, this invention relates to compounds that are inhibitors of Aurora -2 protein kinases. The invention further relates to methods for treating diseases associated with protein kinases, especially diseases associated with Aurora-2, such as cancer.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US25788700P | 2000-12-21 | 2000-12-21 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP034663A true ECSP034663A (en) | 2003-07-25 |
Family
ID=34078813
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSP034662 ECSP034662A (en) | 2000-12-21 | 2003-06-20 | PIRAZOL COMPOUNDS USED AS PROTEIN QUINASA INHIBITORS |
| ECSP034663 ECSP034663A (en) | 2000-12-21 | 2003-06-20 | PIRAZOL COMPOUNDS USED AS PROTEIN QUINASA INHIBITORS |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSP034662 ECSP034662A (en) | 2000-12-21 | 2003-06-20 | PIRAZOL COMPOUNDS USED AS PROTEIN QUINASA INHIBITORS |
Country Status (2)
| Country | Link |
|---|---|
| EC (2) | ECSP034662A (en) |
| ZA (8) | ZA200304472B (en) |
-
2003
- 2003-06-09 ZA ZA200304472A patent/ZA200304472B/en unknown
- 2003-06-09 ZA ZA200304471A patent/ZA200304471B/en unknown
- 2003-06-09 ZA ZA200304470A patent/ZA200304470B/en unknown
- 2003-06-09 ZA ZA200304469A patent/ZA200304469B/en unknown
- 2003-06-09 ZA ZA200304468A patent/ZA200304468B/en unknown
- 2003-06-09 ZA ZA200304474A patent/ZA200304474B/en unknown
- 2003-06-09 ZA ZA200304475A patent/ZA200304475B/en unknown
- 2003-06-09 ZA ZA200304473A patent/ZA200304473B/en unknown
- 2003-06-20 EC ECSP034662 patent/ECSP034662A/en unknown
- 2003-06-20 EC ECSP034663 patent/ECSP034663A/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| ZA200304472B (en) | 2004-06-25 |
| ZA200304469B (en) | 2004-06-24 |
| ZA200304468B (en) | 2004-06-24 |
| ECSP034662A (en) | 2003-07-25 |
| ZA200304474B (en) | 2004-06-25 |
| ZA200304471B (en) | 2004-06-24 |
| ZA200304470B (en) | 2004-06-24 |
| ZA200304473B (en) | 2004-06-24 |
| ZA200304475B (en) | 2004-06-24 |
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