ECSP003787A - A PIRAZOLOTRIAZINE REPLACED AS SELECTIVE INVESTED AGONISTS FOR THE GABA-A ALFA5 RECEPTOR SUBTIPE - Google Patents

A PIRAZOLOTRIAZINE REPLACED AS SELECTIVE INVESTED AGONISTS FOR THE GABA-A ALFA5 RECEPTOR SUBTIPE

Info

Publication number
ECSP003787A
ECSP003787A ECSP003787A ECSP003787A EC SP003787 A ECSP003787 A EC SP003787A EC SP003787 A ECSP003787 A EC SP003787A EC SP003787 A ECSP003787 A EC SP003787A
Authority
EC
Ecuador
Prior art keywords
subtipe
pirazolotriazine
alfa5
invested
gaba
Prior art date
Application number
Other languages
Spanish (es)
Inventor
William Robert Carling
Original Assignee
Merck Sharp & Dohme
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Sharp & Dohme filed Critical Merck Sharp & Dohme
Publication of ECSP003787A publication Critical patent/ECSP003787A/en

Links

Abstract

Se describen 3-tere-butil-7-(5-metilisoxazol-3-il)-2-(2-metil-2H-[1.2.4]triazol-3-ilmetoxi)pirazolo [1,5-d] [1.2.4]triazina, composiciones farmacéuticas que los comprenden, se usa para estimular la cognición y en procedimientos de tratamiento de sujetos que sufren cognición reducida.3-Tere-butyl-7- (5-methylisoxazol-3-yl) -2- (2-methyl-2H- [1.2.4] triazol-3-ylmethoxy) pyrazolo [1,5-d] [1.2 are described .4] triazine, pharmaceutical compositions that comprise them, is used to stimulate cognition and in treatment procedures for subjects suffering from reduced cognition.

ECSP003787 1999-11-25 2000-11-24 A PIRAZOLOTRIAZINE REPLACED AS SELECTIVE INVESTED AGONISTS FOR THE GABA-A ALFA5 RECEPTOR SUBTIPE ECSP003787A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB9927874.9A GB9927874D0 (en) 1999-11-25 1999-11-25 Therapeutic agents

Publications (1)

Publication Number Publication Date
ECSP003787A true ECSP003787A (en) 2002-05-23

Family

ID=10865128

Family Applications (1)

Application Number Title Priority Date Filing Date
ECSP003787 ECSP003787A (en) 1999-11-25 2000-11-24 A PIRAZOLOTRIAZINE REPLACED AS SELECTIVE INVESTED AGONISTS FOR THE GABA-A ALFA5 RECEPTOR SUBTIPE

Country Status (2)

Country Link
EC (1) ECSP003787A (en)
GB (1) GB9927874D0 (en)

Also Published As

Publication number Publication date
GB9927874D0 (en) 2000-01-26

Similar Documents

Publication Publication Date Title
NZ515705A (en) Substituted phenylpropionic acid derivatives as agonists to human peroxisome proliferator-activated receptor (PPAR) alpha
CO5011096A1 (en) MEDICINES CONTAINING ANTAGONISTS OF THE 5-HT3 RECEPTOR FOR THE TREATMENT OF IBS
ES2132223T3 (en) INDOL DERIVATIVES CONDENSED AS ANTAGONISTS OF THE 5-HT4 RECEPTOR.
EA200101156A1 (en) DRUG COMPOSITIONS OF A NEW TYPE ON THE BASIS OF POSSESSING HOLYNTHERGIC ACTION OF COMPOUNDS AND β-MIMETIC
EA199901107A1 (en) SYSTEMS AND DEVICES FOR THE TREATMENT OF BONE FRACTURES OR BONE PATIENTS WITH THE HELP OF EXPANDABLE BODIES (OPTIONS), STERILE SET OF TOOLS FOR INTRODUCTION IN BONE (OPTIONS)
CU23208A3 (en) OXAZOLIDINONAS REPLACED AND ITS USE IN THE FIELD OF THE SANGUINEA COAGULATION
ES2186015T3 (en) DERIVATIVES OF 2- (PURIN-9-IL) -TETRAHIDROFURAN-3,4-DIOL.
SV2005002148A (en) "MODULATING COMPOUNDS OF THE C-KIT ACTIVITY AND USES OF THE SAME"
AR007961A1 (en) CYCLOALKYL DERIVATIVES AS INHIBITORS OF BONE RESORPTION AND VITRONECTIN RECEPTOR ANTAGONISTS, PROCEDURE FOR THEIR PREPARATION AND PHARMACEUTICAL PREPARATION.
AR025960A1 (en) SUBSTANCES LIBRARY CONTAINING BICYCLE IMIDAZO-5-IL-AMINES AND / OR BICYCLIC 3-IL-AMINAS IMMEDITION, PROCEDURE FOR THE PREPARATION OF SUBSTANTIAL LIBRARY, AND USE OF SUBSTANCES OF THIS LIBRARY FOR THE PREPARATION OF DRUG PREPARATION
CL2008003939A1 (en) Use of escitalopram or a pharmaceutically acceptable salt thereof to prepare a drug useful in the treatment of social anxiety (divisional application 1799-00).
BR0011856A (en) N-pyrazole a2a receptor agonists
AR008991A1 (en) DIMETHYL- (3-ARYL-BUT-3-ENYL) -AMINE COMPOUNDS, PROCEDURES FOR THEIR PREPARATION AND APPLICATION OF THEM
DE69932510D1 (en) VASKULARISIERUNGSINHIBITOREN
BR0113291A (en) aporphine esters and their use in therapy
BR0107628A (en) 1,2-diarylbenzimidazoles for treating diseases that are associated with microglial activation
CR6398A (en) 5HT1 ANTAGONISTS FOR ANTIDEPRESSIVE THERAPY
DK122191D0 (en) BENZIMIDAZOLE DERIVATIVES AND PHYSIOLOGICALLY ACCEPTABLE SALTS AND PROCEDURES FOR THE PREPARATION OF SAME
ES2124861T3 (en) AMINO ACID DERIVATIVES AND THEIR USE AS ENCEPHALINASE INHIBITORS.
CO5011066A1 (en) TRIAZINE COMPOUNDS
ECSP003787A (en) A PIRAZOLOTRIAZINE REPLACED AS SELECTIVE INVESTED AGONISTS FOR THE GABA-A ALFA5 RECEPTOR SUBTIPE
DE69933671D1 (en) ADENOSINE A1 ANTAGONISTS AGAINST MALE STERILITY
AR037496A1 (en) NOVEDOUS USE OF 2- [5- (4-FLUOROPHENYL) -3-PIRIDILMETILAMINOMETIL] -CROMANO AND ITS PHYSIOLOGICALLY ACCEPTABLE SALTS
AR026475A1 (en) A PIRAZOLOTRIAZINA REPLACED AS A SELECTIVE INVESTED AGONIST APRA THE GABA-A ALFA RECEIVER SUBTIPE 5
ES2191908T3 (en) 4-AMINOPIRROL (3,2-D) PYRIMIDINS AS ANTAGONISTS OF THE NEUROPEPTIDE RECEPTOR.