ECSP003523A - N- CYCLOPENTIL MODULATORS OF THE RECEPTORY ACTIVITY OF BEMOQUINE - Google Patents

N- CYCLOPENTIL MODULATORS OF THE RECEPTORY ACTIVITY OF BEMOQUINE

Info

Publication number
ECSP003523A
ECSP003523A ECSP003523A ECSP003523A EC SP003523 A ECSP003523 A EC SP003523A EC SP003523 A ECSP003523 A EC SP003523A EC SP003523 A ECSP003523 A EC SP003523A
Authority
EC
Ecuador
Prior art keywords
modulators
activity
bemoquine
receptory
cyclopentil
Prior art date
Application number
Other languages
Spanish (es)
Inventor
Sander G Mills
Paul E Finke
Kerry A Hilfiker
Malcolm Maccoss
Kevin T Chapman
Jennifer L Loebach
Ravi N Guthikonda
Shrenik K Shah
Dooseop Kim
Dong-Ming Shen
Bryan Oates
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Priority to ECSP003523 priority Critical patent/ECSP003523A/en
Publication of ECSP003523A publication Critical patent/ECSP003523A/en

Links

Abstract

La presente invención está dirigida a los compuestos de la fórmula I (gráfico), (en que R1, R3, R4, R5, R6, R7, R8, X n, x y y se definen en este trabajo) que son útiles como moduladores de la actividad receptora de la quemoquina. En particular, estos compuestos son útiles como moduladores de los receptores CCR-5 y/o CCR-3 de la quemoquina.The present invention is directed to compounds of formula I (graph), (where R1, R3, R4, R5, R6, R7, R8, X n, x, and y are defined herein) which are useful as modulators of the chemokine receptor activity. In particular, these compounds are useful as modulators of chemokine CCR-5 and / or CCR-3 receptors.

ECSP003523 2000-06-09 2000-06-09 N- CYCLOPENTIL MODULATORS OF THE RECEPTORY ACTIVITY OF BEMOQUINE ECSP003523A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
ECSP003523 ECSP003523A (en) 2000-06-09 2000-06-09 N- CYCLOPENTIL MODULATORS OF THE RECEPTORY ACTIVITY OF BEMOQUINE

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ECSP003523 ECSP003523A (en) 2000-06-09 2000-06-09 N- CYCLOPENTIL MODULATORS OF THE RECEPTORY ACTIVITY OF BEMOQUINE

Publications (1)

Publication Number Publication Date
ECSP003523A true ECSP003523A (en) 2000-08-18

Family

ID=42041147

Family Applications (1)

Application Number Title Priority Date Filing Date
ECSP003523 ECSP003523A (en) 2000-06-09 2000-06-09 N- CYCLOPENTIL MODULATORS OF THE RECEPTORY ACTIVITY OF BEMOQUINE

Country Status (1)

Country Link
EC (1) ECSP003523A (en)

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