ECSP003448A - SUBSTITUTED AZOLS - Google Patents
SUBSTITUTED AZOLSInfo
- Publication number
- ECSP003448A ECSP003448A ECSP003448A ECSP003448A EC SP003448 A ECSP003448 A EC SP003448A EC SP003448 A ECSP003448 A EC SP003448A EC SP003448 A ECSP003448 A EC SP003448A
- Authority
- EC
- Ecuador
- Prior art keywords
- azols
- substituted
- diseases
- tnf
- graph
- Prior art date
Links
- 201000010099 disease Diseases 0.000 abstract 2
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 2
- 108010002352 Interleukin-1 Proteins 0.000 abstract 1
- 208000001132 Osteoporosis Diseases 0.000 abstract 1
- 230000004097 bone metabolism Effects 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 230000001404 mediated effect Effects 0.000 abstract 1
- 239000002829 mitogen activated protein kinase inhibitor Substances 0.000 abstract 1
- 206010039073 rheumatoid arthritis Diseases 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Los compuestos de la fórmula I (gráfico), en donde los simbolos tienen los significados definidos en la presente, son inhibidores de cinasa MAP p38, y son útiles farmacéuticamente para el tratamiento de enfermedades mediadas por TNF e IL-1, tales como artritis reumatoide, y enfermedades del metabolismo óseo, por ejemplo osteoporosis.The compounds of formula I (graph), where the symbols have the meanings defined herein, are MAP kinase inhibitors p38, and are pharmaceutically useful for the treatment of diseases mediated by TNF and IL-1, such as rheumatoid arthritis , and diseases of bone metabolism, for example osteoporosis.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP003448 ECSP003448A (en) | 2000-04-27 | 2000-04-27 | SUBSTITUTED AZOLS |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP003448 ECSP003448A (en) | 2000-04-27 | 2000-04-27 | SUBSTITUTED AZOLS |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP003448A true ECSP003448A (en) | 2000-05-25 |
Family
ID=42041076
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSP003448 ECSP003448A (en) | 2000-04-27 | 2000-04-27 | SUBSTITUTED AZOLS |
Country Status (1)
| Country | Link |
|---|---|
| EC (1) | ECSP003448A (en) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US9029409B2 (en) | 2011-04-30 | 2015-05-12 | Abbvie Inc. | Isoxazolines as therapeutic agents |
-
2000
- 2000-04-27 EC ECSP003448 patent/ECSP003448A/en unknown
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US9029409B2 (en) | 2011-04-30 | 2015-05-12 | Abbvie Inc. | Isoxazolines as therapeutic agents |
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