EA202192822A1 - Naphthyridine Compounds as Jak Kinase Inhibitors - Google Patents

Naphthyridine Compounds as Jak Kinase Inhibitors

Info

Publication number
EA202192822A1
EA202192822A1 EA202192822A EA202192822A EA202192822A1 EA 202192822 A1 EA202192822 A1 EA 202192822A1 EA 202192822 A EA202192822 A EA 202192822A EA 202192822 A EA202192822 A EA 202192822A EA 202192822 A1 EA202192822 A1 EA 202192822A1
Authority
EA
Eurasian Patent Office
Prior art keywords
compounds
kinase inhibitors
jak kinase
naphthyridine compounds
methods
Prior art date
Application number
EA202192822A
Other languages
Russian (ru)
Inventor
Райан Хадсон
Дженнифер Козак
Пол Р. Фазери
Данте Д. Подесто
Гари И.л. Брандт
Мелисса Флери
Анн-Мари Босолей
Сяоцзюнь Хуан
Венкат Р. Таллади
Original Assignee
ТЕРЕВАНС БАЙОФАРМА Ар энд Ди АйПи, ЭлЭлСи
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by ТЕРЕВАНС БАЙОФАРМА Ар энд Ди АйПи, ЭлЭлСи filed Critical ТЕРЕВАНС БАЙОФАРМА Ар энд Ди АйПи, ЭлЭлСи
Publication of EA202192822A1 publication Critical patent/EA202192822A1/en

Links

Abstract

Изобретение обеспечивает соединения формулы (I)где переменные определены в описании изобретения, или их фармацевтически приемлемые соли, которые являются ингибиторами JAK киназ. Изобретение также обеспечивает фармацевтические композиции, включающие такие соединения, способы применения таких соединений для лечения воспалительных заболеваний кишечника и способы и промежуточные соединения для получения таких соединений.The invention provides compounds of formula (I) wherein the variables are defined in the specification, or pharmaceutically acceptable salts thereof, which are inhibitors of JAK kinases. The invention also provides pharmaceutical compositions comprising such compounds, methods of using such compounds to treat inflammatory bowel diseases, and methods and intermediates for preparing such compounds.

EA202192822A 2016-03-23 2016-05-26 Naphthyridine Compounds as Jak Kinase Inhibitors EA202192822A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201662312273P 2016-03-23 2016-03-23

Publications (1)

Publication Number Publication Date
EA202192822A1 true EA202192822A1 (en) 2022-02-03

Family

ID=67734920

Family Applications (2)

Application Number Title Priority Date Filing Date
EA201990686A EA201990686A1 (en) 2016-03-23 2016-05-26 NAPHTHIRIDINE COMPOUNDS AS JAK KINASE INHIBITORS
EA202192822A EA202192822A1 (en) 2016-03-23 2016-05-26 Naphthyridine Compounds as Jak Kinase Inhibitors

Family Applications Before (1)

Application Number Title Priority Date Filing Date
EA201990686A EA201990686A1 (en) 2016-03-23 2016-05-26 NAPHTHIRIDINE COMPOUNDS AS JAK KINASE INHIBITORS

Country Status (1)

Country Link
EA (2) EA201990686A1 (en)

Also Published As

Publication number Publication date
EA201990686A1 (en) 2019-08-30

Similar Documents

Publication Publication Date Title
EA201792619A1 (en) NAPHTHYRIDINE CONNECTIONS AS JAK KINASE INHIBITORS
CO2018011408A2 (en) Pyrimidine compounds as inhibitors of jak kinase
EA201992128A1 (en) JAK CONDENSED IMIDAZOPIPERIDINE INHIBITORS
EA202090413A1 (en) Pyrazole and triazobicyclic compounds as inhibitors of JAK kinases
EA201691302A1 (en) NEW HETEROCYCLIC COMPOUNDS
MY195427A (en) Jak Kinase Inhibitor Compounds for Treatment of Respiratory Disease
EA201592199A1 (en) BIPYRAZOL DERIVATIVES AS JAK INHIBITORS
MD4800B1 (en) Aminopyrimidinyl compounds as JAK inhibitors
EA201790395A1 (en) AMINOTRIAZIN DERIVATIVES SUITABLE FOR USING AS TANK-BINDING KINASE INHIBITORS
MX2016015565A (en) Certain protein kinase inhibitors.
EA201790246A1 (en) HETEROCYCLIC CARBONIC ACIDS AS ACTIVATORS OF SOLUBLE GUANYLATZYCLIC
EA201990678A1 (en) Heteroarylcarboxamide Compounds as Ripk2 Inhibitors
EA201692260A1 (en) 1,3,4-TIADIAZOLE COMPOUNDS AND THEIR APPLICATION IN CANCER TREATMENT
PH12017500595A1 (en) Aldosterone synthase inhibitors
EA201790253A1 (en) ALDOSTERONSYNTASE INHIBITORS
EA201600002A1 (en) DERIVATIVES OF SUBSTITUTED TRIAZOLOPIRIDINES
EA201891319A1 (en) COMPOUNDS OF ALKYDYDYDROCHINOLINSULPHONAMIDE
EA202192822A1 (en) Naphthyridine Compounds as Jak Kinase Inhibitors
MY192305A (en) Bipyrazole derivatives as jak inhibitors