EA202192639A1 - METHOD FOR PRODUCING SIPONIMOD AND ITS INTERMEDIATE - Google Patents

METHOD FOR PRODUCING SIPONIMOD AND ITS INTERMEDIATE

Info

Publication number
EA202192639A1
EA202192639A1 EA202192639A EA202192639A EA202192639A1 EA 202192639 A1 EA202192639 A1 EA 202192639A1 EA 202192639 A EA202192639 A EA 202192639A EA 202192639 A EA202192639 A EA 202192639A EA 202192639 A1 EA202192639 A1 EA 202192639A1
Authority
EA
Eurasian Patent Office
Prior art keywords
siponimod
producing
relates
intermediates
siponimoda
Prior art date
Application number
EA202192639A
Other languages
Russian (ru)
Inventor
Ролф Келтьенс
Ондрей Гилсе
Иржи Партл
Original Assignee
Синтон Б.В.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Синтон Б.В. filed Critical Синтон Б.В.
Priority claimed from PCT/EP2020/058884 external-priority patent/WO2020201172A1/en
Publication of EA202192639A1 publication Critical patent/EA202192639A1/en

Links

Landscapes

  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Изобретение относится к способу для получения соединения формулы (I) или его соли или его сольвата, т.е. сипонимодаИзобретение также относится к промежуточным соединениям, используемым в способе, и к твердым формам этих промежуточных соединений.The invention relates to a process for the preparation of a compound of formula (I) or a salt or solvate thereof, i.e. siponimoda The invention also relates to intermediates used in the process and to solid forms of these intermediates.

EA202192639A 2019-12-16 2020-03-29 METHOD FOR PRODUCING SIPONIMOD AND ITS INTERMEDIATE EA202192639A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP19216424 2019-12-16
PCT/EP2020/058884 WO2020201172A1 (en) 2019-03-29 2020-03-29 Process for making siponimod and intermediate thereof

Publications (1)

Publication Number Publication Date
EA202192639A1 true EA202192639A1 (en) 2021-12-10

Family

ID=68917532

Family Applications (1)

Application Number Title Priority Date Filing Date
EA202192639A EA202192639A1 (en) 2019-12-16 2020-03-29 METHOD FOR PRODUCING SIPONIMOD AND ITS INTERMEDIATE

Country Status (1)

Country Link
EA (1) EA202192639A1 (en)

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