EA202191250A1 - MIXTURES AND COMPOSITIONS INCLUDING 5-FLUORO-4-IMINO-3-METHYL-1-TOSIL-3,4-DIHYDROPYRIMIDIN-2-ON, AND METHODS FOR THEIR APPLICATION - Google Patents

MIXTURES AND COMPOSITIONS INCLUDING 5-FLUORO-4-IMINO-3-METHYL-1-TOSIL-3,4-DIHYDROPYRIMIDIN-2-ON, AND METHODS FOR THEIR APPLICATION

Info

Publication number
EA202191250A1
EA202191250A1 EA202191250A EA202191250A EA202191250A1 EA 202191250 A1 EA202191250 A1 EA 202191250A1 EA 202191250 A EA202191250 A EA 202191250A EA 202191250 A EA202191250 A EA 202191250A EA 202191250 A1 EA202191250 A1 EA 202191250A1
Authority
EA
Eurasian Patent Office
Prior art keywords
mixtures
methods
compositions
tosil
dihydropyrimidin
Prior art date
Application number
EA202191250A
Other languages
Russian (ru)
Inventor
Сами Шабтаи
Ноам Шеффер
Дженни Лернер Ярдени
Джеймс Слоан
Original Assignee
Адама Мактешим Лтд.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Адама Мактешим Лтд. filed Critical Адама Мактешим Лтд.
Publication of EA202191250A1 publication Critical patent/EA202191250A1/en

Links

Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N25/00—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests
    • A01N25/02—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests containing liquids as carriers, diluents or solvents
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N25/00—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests
    • A01N25/02—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests containing liquids as carriers, diluents or solvents
    • A01N25/04—Dispersions, emulsions, suspoemulsions, suspension concentrates or gels
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N25/00—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests
    • A01N25/12—Powders or granules
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N25/00—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests
    • A01N25/30—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests characterised by the surfactants
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01P—BIOCIDAL, PEST REPELLANT, PEST ATTRACTANT OR PLANT GROWTH REGULATORY ACTIVITY OF CHEMICAL COMPOUNDS OR PREPARATIONS
    • A01P3/00—Fungicides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Environmental Sciences (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Dentistry (AREA)
  • Agronomy & Crop Science (AREA)
  • Chemical & Material Sciences (AREA)
  • Toxicology (AREA)
  • Organic Chemistry (AREA)
  • Dispersion Chemistry (AREA)
  • Microbiology (AREA)
  • Mycology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

В настоящем изобретении предлагается стабильные жидкие композиции, включающие (a) эффективное с точки зрения фунгицидного действия количество соединения формулы I и (b) жидкий носитель. В настоящем изобретении также предлагаются смеси и композиции, включающие (a) эффективное с точки зрения фунгицидного действия количество соединения формулы I и (b) по меньшей мере одно вспомогательное вещество, выбранное из группы, состоящей из следующих соединений: (i) алкиловый эфир полиалкиленоксида; (ii) сополимер силоксана и полиалкиленоксида; (iii) эфиры жирной кислоты; (iv) винилпирролидоны и их производные; и (v) поверхностно-активные вещества на основе сахаров. В настоящем изобретении также предлагаются способы применения раскрытых в изобретении смесей и композиций и способы приготовления раскрытых в изобретении смесей и композиций.The present invention provides stable liquid compositions comprising (a) a fungicidal effective amount of a compound of Formula I and (b) a liquid carrier. The present invention also provides mixtures and compositions comprising (a) a fungicidal effective amount of a compound of formula I and (b) at least one excipient selected from the group consisting of the following compounds: (i) a polyalkylene oxide alkyl ether; (ii) a copolymer of siloxane and polyalkylene oxide; (iii) fatty acid esters; (iv) vinylpyrrolidones and their derivatives; and (v) sugar-based surfactants. The present invention also provides methods of using the mixtures and compositions disclosed in the invention and methods for preparing the mixtures and compositions disclosed in the invention.

EA202191250A 2018-11-05 2019-11-04 MIXTURES AND COMPOSITIONS INCLUDING 5-FLUORO-4-IMINO-3-METHYL-1-TOSIL-3,4-DIHYDROPYRIMIDIN-2-ON, AND METHODS FOR THEIR APPLICATION EA202191250A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201862755866P 2018-11-05 2018-11-05
PCT/IB2019/059456 WO2020095181A1 (en) 2018-11-05 2019-11-04 Mixtures and compositions comprising 5-fluoro-4-imino-3- methyl-1-tosyl-3,4-dihydropyrimidin-2-one, and methods of use thereof

Publications (1)

Publication Number Publication Date
EA202191250A1 true EA202191250A1 (en) 2021-08-20

Family

ID=68542683

Family Applications (1)

Application Number Title Priority Date Filing Date
EA202191250A EA202191250A1 (en) 2018-11-05 2019-11-04 MIXTURES AND COMPOSITIONS INCLUDING 5-FLUORO-4-IMINO-3-METHYL-1-TOSIL-3,4-DIHYDROPYRIMIDIN-2-ON, AND METHODS FOR THEIR APPLICATION

Country Status (23)

Country Link
US (1) US20210378235A1 (en)
EP (1) EP3876717A1 (en)
JP (1) JP2022507026A (en)
KR (1) KR20210136961A (en)
CN (1) CN113260255A (en)
AR (1) AR116996A1 (en)
AU (1) AU2019374510A1 (en)
BR (1) BR112021008755A2 (en)
CA (1) CA3118729A1 (en)
CL (2) CL2021001173A1 (en)
CO (1) CO2021007328A2 (en)
CR (1) CR20210270A (en)
DO (1) DOP2021000084A (en)
EA (1) EA202191250A1 (en)
EC (1) ECSP21039539A (en)
IL (1) IL282939B1 (en)
MA (1) MA54148A (en)
MX (1) MX2021005283A (en)
PE (1) PE20212103A1 (en)
PH (1) PH12021551040A1 (en)
TW (1) TW202031640A (en)
UY (1) UY38450A (en)
WO (1) WO2020095181A1 (en)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX2022013874A (en) * 2020-05-04 2022-11-30 Adama Makhteshim Ltd Mixtures and compositions comprising 5-fluoro-4-imino-3- methyl-1-tosyl-3,4-dihydropyrimidin-2-one, and methods of use thereof.
EP4284173A1 (en) * 2021-01-27 2023-12-06 Adama Makhteshim Ltd. 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2(1 h)-one for controlling plant diseases
TW202345695A (en) * 2022-03-07 2023-12-01 以色列商安道麥馬克西姆有限公司 Novel agrochemical suspension of sdhi and/or strobilurin fungicides
WO2024028812A1 (en) 2022-08-03 2024-02-08 Adama Makhteshim Ltd. 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2(1h)-one for fungicide-resistant fungus

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
LT2563129T (en) 2010-04-26 2016-10-25 Adama Makhteshim Ltd N3-substituted-n1-sulfonyl-5-fluoropyrimidinone derivatives
BR112016015158A2 (en) 2013-12-31 2017-08-08 Adama Makhteshim Ltd SYNERGISTIC FUNGICIDIAL MIXTURES FOR CONTROL OF FUNGI IN CEREALS
CA2935601C (en) 2013-12-31 2023-03-14 Adama Makhteshim Ltd. 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one and processes for their preparation
MA41272A (en) 2014-12-23 2017-10-31 Adama Makhteshim Ltd 5-FLUORO-4-IMINO-3- (ALKYL / ALKYL SUBSTITUTED) -1- (ARYLSULFONYL) -3,4-DIHYDROPYRIMIDIN-2 (1H) -ONE AS SEED TREATMENT
UY36964A (en) * 2015-10-27 2017-05-31 Bayer Cropscience Ag COMBINATIONS OF ACTIVE PRINCIPLES THAT INCLUDE A DERIVATIVE OF (UNCLE) CARBOXAMIDE AND A FUNGUITED COMPOUND
JP6922272B2 (en) * 2016-03-11 2021-08-18 住友化学株式会社 Plant disease control composition and plant disease control method
WO2019038583A1 (en) 2017-07-17 2019-02-28 Adama Makhteshim Ltd. Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one

Also Published As

Publication number Publication date
BR112021008755A2 (en) 2021-08-10
CL2023001663A1 (en) 2023-12-15
AU2019374510A1 (en) 2021-06-17
MA54148A (en) 2022-02-09
CL2021001173A1 (en) 2021-12-10
EP3876717A1 (en) 2021-09-15
TW202031640A (en) 2020-09-01
CA3118729A1 (en) 2020-05-14
JP2022507026A (en) 2022-01-18
PH12021551040A1 (en) 2022-01-03
ECSP21039539A (en) 2021-07-30
AR116996A1 (en) 2021-06-30
WO2020095181A1 (en) 2020-05-14
IL282939B1 (en) 2024-06-01
CO2021007328A2 (en) 2021-09-30
CR20210270A (en) 2021-07-20
KR20210136961A (en) 2021-11-17
IL282939A (en) 2021-06-30
US20210378235A1 (en) 2021-12-09
PE20212103A1 (en) 2021-11-04
UY38450A (en) 2020-05-29
MX2021005283A (en) 2021-06-18
CN113260255A (en) 2021-08-13
DOP2021000084A (en) 2021-08-15

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