EA202190527A1 - SUBSTITUTED THIOHYDANTHOIN DERIVATIVES AS ANTAGONISTS OF THE ANDROGENIC RECEPTOR - Google Patents

SUBSTITUTED THIOHYDANTHOIN DERIVATIVES AS ANTAGONISTS OF THE ANDROGENIC RECEPTOR

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Publication number
EA202190527A1
EA202190527A1 EA202190527A EA202190527A EA202190527A1 EA 202190527 A1 EA202190527 A1 EA 202190527A1 EA 202190527 A EA202190527 A EA 202190527A EA 202190527 A EA202190527 A EA 202190527A EA 202190527 A1 EA202190527 A1 EA 202190527A1
Authority
EA
Eurasian Patent Office
Prior art keywords
thiohydanthoin
antagonists
derivatives
substituted
androgenic receptor
Prior art date
Application number
EA202190527A
Other languages
Russian (ru)
Inventor
Питер Дж. Коннолли
Иан Хиксон
Ливен Мерпул
Винет Панде
Чжумин ЧЖАН
Джонатан Брэнч
Кристиан Рокебой
Луис Б. Трабалон Эсколар
Жилль Биньян
Original Assignee
Янссен Фармацевтика Нв
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Янссен Фармацевтика Нв filed Critical Янссен Фармацевтика Нв
Publication of EA202190527A1 publication Critical patent/EA202190527A1/en

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  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Описаны соединения, композиции и способы лечения расстройств, которые зависят от антагонизма одного или более типов андрогенных рецепторов. Такие соединения представлены следующей формулой (I):где R1 и G определены в настоящем документе.Described are compounds, compositions and methods of treating disorders that depend on the antagonism of one or more types of androgen receptors. Such compounds are represented by the following formula (I): where R1 and G are defined herein.

EA202190527A 2016-07-18 2017-01-10 SUBSTITUTED THIOHYDANTHOIN DERIVATIVES AS ANTAGONISTS OF THE ANDROGENIC RECEPTOR EA202190527A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201662363534P 2016-07-18 2016-07-18

Publications (1)

Publication Number Publication Date
EA202190527A1 true EA202190527A1 (en) 2021-09-30

Family

ID=77912704

Family Applications (1)

Application Number Title Priority Date Filing Date
EA202190527A EA202190527A1 (en) 2016-07-18 2017-01-10 SUBSTITUTED THIOHYDANTHOIN DERIVATIVES AS ANTAGONISTS OF THE ANDROGENIC RECEPTOR

Country Status (1)

Country Link
EA (1) EA202190527A1 (en)

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