EA202190393A1 - COMPOUNDS OF PYRAZOLO [3,4-b] PYRIDINE AS INHIBITORS OF TAM- AND MET-KINASES - Google Patents
COMPOUNDS OF PYRAZOLO [3,4-b] PYRIDINE AS INHIBITORS OF TAM- AND MET-KINASESInfo
- Publication number
- EA202190393A1 EA202190393A1 EA202190393A EA202190393A EA202190393A1 EA 202190393 A1 EA202190393 A1 EA 202190393A1 EA 202190393 A EA202190393 A EA 202190393A EA 202190393 A EA202190393 A EA 202190393A EA 202190393 A1 EA202190393 A1 EA 202190393A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- kinases
- tam
- met
- inhibitors
- compounds
- Prior art date
Links
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
В данном документе предусмотрены соединения формулы Iи их стереоизомеры, таутомеры и фармацевтически приемлемые соли, в которых R1, R2, R9, X1 и G являются такими, как определяется в данном документе, которые представляют собой ингибиторы одной или нескольких TAM-киназ и/или c-Met-киназы, и являются приемлемыми в лечении и предупреждении заболеваний, которые могут лечиться ингибитором TAM-киназы и/или ингибитором c-Met киназы.Provided herein are compounds of Formula I and their stereoisomers, tautomers and pharmaceutically acceptable salts, in which R1, R2, R9, X1 and G are as defined herein, which are inhibitors of one or more TAM kinases and / or c Α-Met kinases, and are useful in the treatment and prevention of diseases that can be treated with a TAM kinase inhibitor and / or a c-Met kinase inhibitor.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201962858686P | 2019-06-07 | 2019-06-07 | |
| PCT/US2019/048701 WO2020047184A1 (en) | 2018-08-30 | 2019-08-29 | PYRAZOLO[3,4-b]PYRIDINE COMPOUNDS AS INHIBITORS OF TAM AND MET KINASES |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| EA202190393A1 true EA202190393A1 (en) | 2021-10-25 |
Family
ID=78572574
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| EA202190393A EA202190393A1 (en) | 2019-06-07 | 2019-08-29 | COMPOUNDS OF PYRAZOLO [3,4-b] PYRIDINE AS INHIBITORS OF TAM- AND MET-KINASES |
Country Status (1)
| Country | Link |
|---|---|
| EA (1) | EA202190393A1 (en) |
-
2019
- 2019-08-29 EA EA202190393A patent/EA202190393A1/en unknown
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