EA202190150A1 - AMINOPYRIMIDONYL DERIVATIVES, METHOD FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM - Google Patents

AMINOPYRIMIDONYL DERIVATIVES, METHOD FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

Info

Publication number
EA202190150A1
EA202190150A1 EA202190150A EA202190150A EA202190150A1 EA 202190150 A1 EA202190150 A1 EA 202190150A1 EA 202190150 A EA202190150 A EA 202190150A EA 202190150 A EA202190150 A EA 202190150A EA 202190150 A1 EA202190150 A1 EA 202190150A1
Authority
EA
Eurasian Patent Office
Prior art keywords
aminopyrimidonyl
derivatives
preparation
pharmaceutical compositions
compositions containing
Prior art date
Application number
EA202190150A
Other languages
Russian (ru)
Inventor
Чаба Вебер
Андраш Кочи
Аттила Вашаш
Арпад Кишш
Балаж Мольнар
Альба Масьяс
Андреа Фиумана
Николас Дэвис
Джеймс Брук Мюррей
Эмили Селлье
Дидье Демарль
Лиза Иваншитц
Оливье Женест
Original Assignee
Ле Лаборатуар Сервье
Верналис (Р&Д) Лимитед
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ле Лаборатуар Сервье, Верналис (Р&Д) Лимитед filed Critical Ле Лаборатуар Сервье
Priority claimed from PCT/EP2019/068050 external-priority patent/WO2020008013A1/en
Publication of EA202190150A1 publication Critical patent/EA202190150A1/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/14Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Соединения формулы (I)где R1, R2, R3, R4, R5, R6, J и n являются такими, как определено в описании. Лекарственные средства.Compounds of formula (I) wherein R1, R2, R3, R4, R5, R6, J and n are as defined herein. Medicines.

EA202190150A 2019-05-27 2019-07-04 AMINOPYRIMIDONYL DERIVATIVES, METHOD FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM EA202190150A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP19305667 2019-05-27
PCT/EP2019/068050 WO2020008013A1 (en) 2018-07-05 2019-07-04 Amino-pyrimidonyl derivatives, a process for their preparation and pharmaceutical compositions containing them

Publications (1)

Publication Number Publication Date
EA202190150A1 true EA202190150A1 (en) 2021-05-24

Family

ID=67003348

Family Applications (1)

Application Number Title Priority Date Filing Date
EA202190150A EA202190150A1 (en) 2019-05-27 2019-07-04 AMINOPYRIMIDONYL DERIVATIVES, METHOD FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

Country Status (1)

Country Link
EA (1) EA202190150A1 (en)

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