EA202092648A1 - SOLID FORMS OF FGFR INHIBITOR AND METHODS FOR THEIR PREPARATION - Google Patents
SOLID FORMS OF FGFR INHIBITOR AND METHODS FOR THEIR PREPARATIONInfo
- Publication number
- EA202092648A1 EA202092648A1 EA202092648A EA202092648A EA202092648A1 EA 202092648 A1 EA202092648 A1 EA 202092648A1 EA 202092648 A EA202092648 A EA 202092648A EA 202092648 A EA202092648 A EA 202092648A EA 202092648 A1 EA202092648 A1 EA 202092648A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- preparation
- solid forms
- methods
- fgfr inhibitor
- fgfr
- Prior art date
Links
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
Настоящее изобретение относится к 3-(2,6-дифтор-3,5-диметоксифенил)-1-этил-8-(морфолин-4-илметил)-1,3,4,7-тетрагидро-2H-пирроло[3',2':5,6]пиридо[4,3-d]пиримидин-2-ону, его твердым формам и полиморфам, способам их получения и промежуточным соединениям при их получении, которые применимы при лечении FGFR-ассоциированных или опосредованных заболеваний, таких как рак.The present invention relates to 3- (2,6-difluoro-3,5-dimethoxyphenyl) -1-ethyl-8- (morpholin-4-ylmethyl) -1,3,4,7-tetrahydro-2H-pyrrolo [3 ' , 2 ': 5,6] pyrido [4,3-d] pyrimidin-2-one, its solid forms and polymorphs, processes for their preparation and intermediates upon their preparation, which are useful in the treatment of FGFR-associated or mediated diseases such like cancer.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201962815539P | 2019-03-08 | 2019-03-08 | |
PCT/US2019/030633 WO2019213544A2 (en) | 2018-05-04 | 2019-05-03 | Solid forms of an fgfr inhibitor and processes for preparing the same |
Publications (1)
Publication Number | Publication Date |
---|---|
EA202092648A1 true EA202092648A1 (en) | 2021-03-24 |
Family
ID=75262214
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA202092648A EA202092648A1 (en) | 2019-03-08 | 2019-05-03 | SOLID FORMS OF FGFR INHIBITOR AND METHODS FOR THEIR PREPARATION |
Country Status (1)
Country | Link |
---|---|
EA (1) | EA202092648A1 (en) |
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2019
- 2019-05-03 EA EA202092648A patent/EA202092648A1/en unknown
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