EA202092514A1 - IZOINDOLINES AS HDAC INHIBITORS - Google Patents

IZOINDOLINES AS HDAC INHIBITORS

Info

Publication number
EA202092514A1
EA202092514A1 EA202092514A EA202092514A EA202092514A1 EA 202092514 A1 EA202092514 A1 EA 202092514A1 EA 202092514 A EA202092514 A EA 202092514A EA 202092514 A EA202092514 A EA 202092514A EA 202092514 A1 EA202092514 A1 EA 202092514A1
Authority
EA
Eurasian Patent Office
Prior art keywords
izoindolines
hdac inhibitors
hdac
inhibitors
formulas
Prior art date
Application number
EA202092514A
Other languages
Russian (ru)
Inventor
Сяочжан Чжэн
Мэттью В. Мартин
Пуи Йи Нг
Дженнифер Р. Томасон
Бинсун Хан
Александра Рудницкая
мл. Дэвид Р. Лансия
Original Assignee
Вейло Эрли Дискавери, Инк.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Вейло Эрли Дискавери, Инк. filed Critical Вейло Эрли Дискавери, Инк.
Priority claimed from PCT/US2019/028026 external-priority patent/WO2019204550A1/en
Publication of EA202092514A1 publication Critical patent/EA202092514A1/en

Links

Abstract

Данное описание относится к ингибиторам цинкзависимых гистондеацетилаз (HDAC), имеющим формулугде Z, X1, X2, Y1, Y2, Y3, L, Z и R описаны в данном документе.This disclosure relates to zinc dependent histone deacetylase (HDAC) inhibitors having the formulas Z, X1, X2, Y1, Y2, Y3, L, Z and R are described herein.

EA202092514A 2018-05-09 2019-04-18 IZOINDOLINES AS HDAC INHIBITORS EA202092514A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201862669286P 2018-05-09 2018-05-09
PCT/US2019/028026 WO2019204550A1 (en) 2018-04-20 2019-04-18 Isoindolines as hdac inhibitors

Publications (1)

Publication Number Publication Date
EA202092514A1 true EA202092514A1 (en) 2021-02-17

Family

ID=74855462

Family Applications (1)

Application Number Title Priority Date Filing Date
EA202092514A EA202092514A1 (en) 2018-05-09 2019-04-18 IZOINDOLINES AS HDAC INHIBITORS

Country Status (1)

Country Link
EA (1) EA202092514A1 (en)

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