EA202091472A1 - TRIAZOL-AZINES OF CYCLOHEXYLIC ACID AS LPA ANTAGONISTS - Google Patents

TRIAZOL-AZINES OF CYCLOHEXYLIC ACID AS LPA ANTAGONISTS

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Publication number
EA202091472A1
EA202091472A1 EA202091472A EA202091472A EA202091472A1 EA 202091472 A1 EA202091472 A1 EA 202091472A1 EA 202091472 A EA202091472 A EA 202091472A EA 202091472 A EA202091472 A EA 202091472A EA 202091472 A1 EA202091472 A1 EA 202091472A1
Authority
EA
Eurasian Patent Office
Prior art keywords
azines
triazol
cyclohexylic acid
lpa antagonists
lpa
Prior art date
Application number
EA202091472A
Other languages
Russian (ru)
Inventor
Янь Ши
Ин Ван
Питер Тай Вах Чэн
Цзюнь ШИ
Шивэй Тао
Джеймс Р. Корте
Тианан Фан
Цзюнь Ли
Лоуренс Дж. Кеннеди
Роберт Ф. Кальтенбах III
Сутьяно Юсуф
Original Assignee
Бристол-Маерс Сквибб Компани
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Бристол-Маерс Сквибб Компани filed Critical Бристол-Маерс Сквибб Компани
Priority claimed from PCT/US2018/066121 external-priority patent/WO2019126093A1/en
Publication of EA202091472A1 publication Critical patent/EA202091472A1/en

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Abstract

Настоящее изобретение относится к соединениям формулы (I)или их стереоизомеру, таутомеру или их фармацевтически приемлемой соли или сольвату, где все переменные являются такими, как определено в настоящем документе. Данные соединения являются селективными ингибиторами рецепторов LPA.The present invention relates to compounds of formula (I), or a stereoisomer, tautomer, or a pharmaceutically acceptable salt or solvate thereof, where all variables are as defined herein. These compounds are selective inhibitors of LPA receptors.

EA202091472A 2018-11-26 2018-12-18 TRIAZOL-AZINES OF CYCLOHEXYLIC ACID AS LPA ANTAGONISTS EA202091472A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201862771214P 2018-11-26 2018-11-26
PCT/US2018/066121 WO2019126093A1 (en) 2017-12-19 2018-12-18 Cyclohexyl acid triazole azines as lpa antagonists

Publications (1)

Publication Number Publication Date
EA202091472A1 true EA202091472A1 (en) 2020-09-29

Family

ID=72616035

Family Applications (1)

Application Number Title Priority Date Filing Date
EA202091472A EA202091472A1 (en) 2018-11-26 2018-12-18 TRIAZOL-AZINES OF CYCLOHEXYLIC ACID AS LPA ANTAGONISTS

Country Status (1)

Country Link
EA (1) EA202091472A1 (en)

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