EA202090982A1 - BENZIMIDAZOLE DERIVATIVES AND VARIANTS OF THEIR APPLICATION - Google Patents

BENZIMIDAZOLE DERIVATIVES AND VARIANTS OF THEIR APPLICATION

Info

Publication number
EA202090982A1
EA202090982A1 EA202090982A EA202090982A EA202090982A1 EA 202090982 A1 EA202090982 A1 EA 202090982A1 EA 202090982 A EA202090982 A EA 202090982A EA 202090982 A EA202090982 A EA 202090982A EA 202090982 A1 EA202090982 A1 EA 202090982A1
Authority
EA
Eurasian Patent Office
Prior art keywords
present
variants
application
benzimidazole derivatives
compound
Prior art date
Application number
EA202090982A
Other languages
Russian (ru)
Inventor
Майкл Д. Бартбергер
Нагасрее Чакка
Хуа Гао
Анхель Гусман-Перес
Дэниел Б. Хорн
Цзихао Хуа
Мадлен Киффер
Дэниэл С.Х. Лин
Бенджамин Чарльз Милграм
Джейн Пантелеев
Лори Шенкел
Джон Стеллваген
Мэттью Вайсс
Райан Д. Уайт
Вей Чжао
Original Assignee
Эмджен Инк.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Эмджен Инк. filed Critical Эмджен Инк.
Priority claimed from PCT/US2018/056484 external-priority patent/WO2019079578A1/en
Publication of EA202090982A1 publication Critical patent/EA202090982A1/en

Links

Abstract

Настоящее изобретение относится к ингибиторам активности белка канала 6 транзиторного рецепторного потенциала (TRPC6). В настоящем изобретении предусмотрены соединение формулы (I) или его фармацевтически приемлемая соль, фармацевтические композиции, содержащие соединение по настоящему изобретению, способ изготовления соединений по настоящему изобретению и варианты их терапевтического применения.The present invention relates to inhibitors of transient receptor potential channel 6 (TRPC6) protein activity. The present invention provides a compound of formula (I) or a pharmaceutically acceptable salt thereof, pharmaceutical compositions containing a compound of the present invention, a method for preparing the compounds of the present invention, and their therapeutic uses.

EA202090982A 2018-05-14 2018-10-18 BENZIMIDAZOLE DERIVATIVES AND VARIANTS OF THEIR APPLICATION EA202090982A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201862671090P 2018-05-14 2018-05-14
PCT/US2018/056484 WO2019079578A1 (en) 2017-10-19 2018-10-18 Benzimidazole derivatives and their uses

Publications (1)

Publication Number Publication Date
EA202090982A1 true EA202090982A1 (en) 2020-10-27

Family

ID=73129288

Family Applications (1)

Application Number Title Priority Date Filing Date
EA202090982A EA202090982A1 (en) 2018-05-14 2018-10-18 BENZIMIDAZOLE DERIVATIVES AND VARIANTS OF THEIR APPLICATION

Country Status (1)

Country Link
EA (1) EA202090982A1 (en)

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