EA202090969A1 - TERTIARY ALCOHOLS AS PI3K INHIBITORS - Google Patents

TERTIARY ALCOHOLS AS PI3K INHIBITORS

Info

Publication number
EA202090969A1
EA202090969A1 EA202090969A EA202090969A EA202090969A1 EA 202090969 A1 EA202090969 A1 EA 202090969A1 EA 202090969 A EA202090969 A EA 202090969A EA 202090969 A EA202090969 A EA 202090969A EA 202090969 A1 EA202090969 A1 EA 202090969A1
Authority
EA
Eurasian Patent Office
Prior art keywords
tertiary alcohols
pi3k inhibitors
diseases
pi3k
disorders
Prior art date
Application number
EA202090969A
Other languages
Russian (ru)
Inventor
Брент Даути
Эндрю У. Бьюскинг
Дэвид М. Бернс
Эндрю П. Комбс
Нику Фалахатпишех
Рави Кумар Джаллури
Дэниел Леви
Падмаджа Полам
Лисинь Шао
Стейси Шепард
Артем Шварцбарт
Ричард Б. Спаркс
Эдди В. Юэ
Original Assignee
Инсайт Корпорейшн
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Инсайт Корпорейшн filed Critical Инсайт Корпорейшн
Priority claimed from PCT/US2018/056311 external-priority patent/WO2019079469A1/en
Publication of EA202090969A1 publication Critical patent/EA202090969A1/en

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Данная заявка относится к соединениям формулы (I)или его фармацевтически приемлемым солям, которые являются ингибиторами PI3K-, пригодным для лечения расстройств, таких как аутоиммунные заболевания, рак, сердечно-сосудистые заболевания и нейродегенеративные заболевания.This application relates to compounds of formula (I), or pharmaceutically acceptable salts thereof, which are PI3K-inhibitors useful in the treatment of disorders such as autoimmune diseases, cancer, cardiovascular diseases and neurodegenerative diseases.

EA202090969A 2018-09-05 2018-10-17 TERTIARY ALCOHOLS AS PI3K INHIBITORS EA202090969A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201862727316P 2018-09-05 2018-09-05
PCT/US2018/056311 WO2019079469A1 (en) 2017-10-18 2018-10-17 Condensed imidazole derivatives substituted by tertiary hydroxy groups as pi3k-gamma inhibitors

Publications (1)

Publication Number Publication Date
EA202090969A1 true EA202090969A1 (en) 2020-09-29

Family

ID=72615984

Family Applications (1)

Application Number Title Priority Date Filing Date
EA202090969A EA202090969A1 (en) 2018-09-05 2018-10-17 TERTIARY ALCOHOLS AS PI3K INHIBITORS

Country Status (1)

Country Link
EA (1) EA202090969A1 (en)

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