EA202090644A1 - IMIDAZO DERIVATIVES [1,5-a] PYRASINE AS PI3K INHIBITORS - Google Patents

IMIDAZO DERIVATIVES [1,5-a] PYRASINE AS PI3K INHIBITORS

Info

Publication number
EA202090644A1
EA202090644A1 EA202090644A EA202090644A EA202090644A1 EA 202090644 A1 EA202090644 A1 EA 202090644A1 EA 202090644 A EA202090644 A EA 202090644A EA 202090644 A EA202090644 A EA 202090644A EA 202090644 A1 EA202090644 A1 EA 202090644A1
Authority
EA
Eurasian Patent Office
Prior art keywords
pyrasine
pi3k inhibitors
imidazo derivatives
present
imidazo
Prior art date
Application number
EA202090644A
Other languages
Russian (ru)
Inventor
Цзин Ли
Хайбо ЧЖАО
Чживэй Ван
Original Assignee
Бейджин, Лтд.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Бейджин, Лтд. filed Critical Бейджин, Лтд.
Priority claimed from PCT/CN2018/104559 external-priority patent/WO2019047915A1/en
Publication of EA202090644A1 publication Critical patent/EA202090644A1/en

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

В настоящем изобретении раскрыты соединение формулы (I) или его стереоизомер, или его фармацевтически приемлемая соль и фармацевтические композиции, содержащие его. В настоящем изобретении также раскрыт способ лечения заболеваний или расстройств, связанных с PI3K, с применением соединения по настоящему изобретению.The present invention discloses a compound of formula (I) or a stereoisomer thereof, or a pharmaceutically acceptable salt thereof, and pharmaceutical compositions containing it. The present invention also discloses a method for treating diseases or disorders associated with PI3K using a compound of the present invention.

EA202090644A 2018-05-11 2018-09-07 IMIDAZO DERIVATIVES [1,5-a] PYRASINE AS PI3K INHIBITORS EA202090644A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CN2018086555 2018-05-11
PCT/CN2018/104559 WO2019047915A1 (en) 2017-09-08 2018-09-07 IMIDAZO[1,5-A]PYRAZINE DERIVATIVES AS PI3Kdelta INHIBITORS

Publications (1)

Publication Number Publication Date
EA202090644A1 true EA202090644A1 (en) 2020-06-24

Family

ID=71138813

Family Applications (1)

Application Number Title Priority Date Filing Date
EA202090644A EA202090644A1 (en) 2018-05-11 2018-09-07 IMIDAZO DERIVATIVES [1,5-a] PYRASINE AS PI3K INHIBITORS

Country Status (1)

Country Link
EA (1) EA202090644A1 (en)

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