EA202090329A1 - PEPTIDE AMIDE COMPOUNDS, METHOD FOR PRODUCING AND MEDICAL USE - Google Patents

PEPTIDE AMIDE COMPOUNDS, METHOD FOR PRODUCING AND MEDICAL USE

Info

Publication number
EA202090329A1
EA202090329A1 EA202090329A EA202090329A EA202090329A1 EA 202090329 A1 EA202090329 A1 EA 202090329A1 EA 202090329 A EA202090329 A EA 202090329A EA 202090329 A EA202090329 A EA 202090329A EA 202090329 A1 EA202090329 A1 EA 202090329A1
Authority
EA
Eurasian Patent Office
Prior art keywords
medical use
producing
peptide amide
amide compounds
improved
Prior art date
Application number
EA202090329A
Other languages
Russian (ru)
Inventor
Чэнь ЧЖАН
Аньбан Хуан
Фей Йе
Лунбинь Хуан
Чжэнган Хуан
Цзяньминь Ван
Юнган Вэй
Панкэ Янь
Вэй Чжэн
Original Assignee
Сычуань Хайско Фармасьютикал Ко., Лтд.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Сычуань Хайско Фармасьютикал Ко., Лтд. filed Critical Сычуань Хайско Фармасьютикал Ко., Лтд.
Priority claimed from PCT/CN2018/096271 external-priority patent/WO2019015644A1/en
Publication of EA202090329A1 publication Critical patent/EA202090329A1/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/07Tetrapeptides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Immunology (AREA)
  • Neurosurgery (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)

Abstract

В изобретении предложено пептидное амидное соединение, представленное общей формулой (I), способ его получения и его медицинское применение. Соединение имеет новую структуру, обладает улучшенной биологической активностью и улучшенным обезболивающим действием.The invention provides a peptide amide compound represented by the general formula (I), a method for its preparation and its medical use. The compound has a new structure, has improved biological activity and an improved analgesic effect.

EA202090329A 2018-01-11 2018-07-19 PEPTIDE AMIDE COMPOUNDS, METHOD FOR PRODUCING AND MEDICAL USE EA202090329A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CN201810014939 2018-01-11
PCT/CN2018/096271 WO2019015644A1 (en) 2017-07-21 2018-07-19 Peptide amide compound and preparation method and medical use thereof

Publications (1)

Publication Number Publication Date
EA202090329A1 true EA202090329A1 (en) 2020-05-25

Family

ID=70847664

Family Applications (1)

Application Number Title Priority Date Filing Date
EA202090329A EA202090329A1 (en) 2018-01-11 2018-07-19 PEPTIDE AMIDE COMPOUNDS, METHOD FOR PRODUCING AND MEDICAL USE

Country Status (1)

Country Link
EA (1) EA202090329A1 (en)

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