EA202090087A3 - 1,2,4-OXADIAZOLE AND THIADIAZOLIC COMPOUNDS AS IMMUNOMODULATORS - Google Patents
1,2,4-OXADIAZOLE AND THIADIAZOLIC COMPOUNDS AS IMMUNOMODULATORSInfo
- Publication number
- EA202090087A3 EA202090087A3 EA202090087A EA202090087A EA202090087A3 EA 202090087 A3 EA202090087 A3 EA 202090087A3 EA 202090087 A EA202090087 A EA 202090087A EA 202090087 A EA202090087 A EA 202090087A EA 202090087 A3 EA202090087 A3 EA 202090087A3
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- oxadiazole
- compounds
- thiadiazolic
- immunomodulators
- inhibiting
- Prior art date
Links
Abstract
Настоящее изобретение относится к 1,2,4-оксадиазольным и тиадиазольным соединениям формулы (I) и их применению для ингибирования сигнального пути запрограммированной гибели клетки 1 (PD1) и/или для лечения нарушений путем ингибирования иммуносупрессивного сигнала, индицированного PD-1, PD-L1 или PD-L2.The present invention relates to 1,2,4-oxadiazole and thiadiazole compounds of formula (I) and their use for inhibiting the programmed cell death 1 (PD1) signaling pathway and / or for treating disorders by inhibiting the immunosuppressive signal indicated by PD-1, PD- L1 or PD-L2.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IN1180CH2015 | 2015-03-10 |
Publications (2)
Publication Number | Publication Date |
---|---|
EA202090087A2 EA202090087A2 (en) | 2020-11-30 |
EA202090087A3 true EA202090087A3 (en) | 2020-12-30 |
Family
ID=73649890
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA202090087A EA202090087A3 (en) | 2015-03-10 | 2016-03-07 | 1,2,4-OXADIAZOLE AND THIADIAZOLIC COMPOUNDS AS IMMUNOMODULATORS |
Country Status (1)
Country | Link |
---|---|
EA (1) | EA202090087A3 (en) |
-
2016
- 2016-03-07 EA EA202090087A patent/EA202090087A3/en unknown
Also Published As
Publication number | Publication date |
---|---|
EA202090087A2 (en) | 2020-11-30 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
PH12017501454A1 (en) | 1,2,4-oxadiazole and thiadiazole compounds as immunomodulators | |
EA201791629A1 (en) | 1,3,4-OXADIAZOL AND TIADIAZOLIC CONNECTIONS AS IMMUNOMODULATORS | |
EA201791634A1 (en) | 3-SUBSTITUTE 1,3,4-OXADIAZOLE AND TIADIAZOLE COMPOUNDS AS IMMUNOMODULATORS | |
PH12017501455A1 (en) | 3-substituted-1,2,4-oxadiazole and thiadiazole compounds as immunomodulators | |
PH12017501456A1 (en) | Therapeutic cyclic compounds as immunomodulators | |
EA201990997A1 (en) | VISTA DOUBLE INHIBITORS AND WAYS PD-1 | |
CY1122986T1 (en) | 1,2,4-OXADIAZOLE DERIVATIVES AS IMMUNE MODULATORS | |
EA201600234A1 (en) | 1,3,4-OXADIAZOLE AND 1,3,4-TIADIAZOLE DERIVATIVES AS AN IMMUNOMODULATOR | |
EA201600235A1 (en) | CYCLIC PEPTIDOMYMETIC COMPOUNDS AS IMMUNOMODULATORS | |
PH12015502611A1 (en) | Heterocyclic compounds as hedgehog signaling pathway inhibitors | |
PH12020550511A1 (en) | Dual inhibitors of tim-3 and pd-1 pathways | |
EA202090087A3 (en) | 1,2,4-OXADIAZOLE AND THIADIAZOLIC COMPOUNDS AS IMMUNOMODULATORS |