EA202090066A1 - THERAPEUTIC FOR THE TREATMENT OF ASPIRATED PNEUMONIA, PULMONARY FORCING OR LUNG ABCESS - Google Patents

THERAPEUTIC FOR THE TREATMENT OF ASPIRATED PNEUMONIA, PULMONARY FORCING OR LUNG ABCESS

Info

Publication number
EA202090066A1
EA202090066A1 EA202090066A EA202090066A EA202090066A1 EA 202090066 A1 EA202090066 A1 EA 202090066A1 EA 202090066 A EA202090066 A EA 202090066A EA 202090066 A EA202090066 A EA 202090066A EA 202090066 A1 EA202090066 A1 EA 202090066A1
Authority
EA
Eurasian Patent Office
Prior art keywords
treatment
pulmonary
pneumonia
aspirated
forcing
Prior art date
Application number
EA202090066A
Other languages
Russian (ru)
Inventor
Масааки Одадзима
Саёко Таниока
Такааки Суноути
Асако Табути
Original Assignee
Керин Фармасьютикал Ко., Лтд.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Керин Фармасьютикал Ко., Лтд. filed Critical Керин Фармасьютикал Ко., Лтд.
Publication of EA202090066A1 publication Critical patent/EA202090066A1/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4375Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a six-membered ring having nitrogen as a ring heteroatom, e.g. quinolizines, naphthyridines, berberine, vincamine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/4709Non-condensed quinolines and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/007Pulmonary tract; Aromatherapy
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Pulmonology (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Настоящее изобретение относится к безопасному и более эффективному терапевтическому средству для лечения инфекций дыхательных путей. Решение: терапевтическое средство для лечения аспирационной пневмонии, легочного нагноения или абсцесса легких, включающее в качестве активного ингредиента 7-[(3S,4S)-3-{(циклопропиламино)метил}-4-фторпирролидин-1-ил]-6-фтор-1-(2-фторэтил)-8-метокси-4-оксо-1,4-дигидрохинолин-3-карбоновую кислоту или ее фармацевтически приемлемую соль.The present invention relates to a safer and more effective therapeutic agent for the treatment of respiratory tract infections. Solution: A therapeutic agent for the treatment of aspiration pneumonia, pulmonary suppuration or lung abscess, containing as an active ingredient 7-[(3S,4S)-3-{(cyclopropylamino)methyl}-4-fluoropyrrolidin-1-yl]-6-fluoro -1-(2-fluoroethyl)-8-methoxy-4-oxo-1,4-dihydroquinoline-3-carboxylic acid or a pharmaceutically acceptable salt thereof.

EA202090066A 2018-03-30 2018-06-15 THERAPEUTIC FOR THE TREATMENT OF ASPIRATED PNEUMONIA, PULMONARY FORCING OR LUNG ABCESS EA202090066A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2018068159 2018-03-30
PCT/JP2018/022846 WO2018230686A1 (en) 2017-06-16 2018-06-15 Therapeutic agent for aspiration pneumonia, lung suppuration, or lung abscess

Publications (1)

Publication Number Publication Date
EA202090066A1 true EA202090066A1 (en) 2020-04-15

Family

ID=64660738

Family Applications (1)

Application Number Title Priority Date Filing Date
EA202090066A EA202090066A1 (en) 2018-03-30 2018-06-15 THERAPEUTIC FOR THE TREATMENT OF ASPIRATED PNEUMONIA, PULMONARY FORCING OR LUNG ABCESS

Country Status (3)

Country Link
CN (1) CN116549446A (en)
EA (1) EA202090066A1 (en)
WO (1) WO2018230686A1 (en)

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT1666477E (en) 2003-09-10 2013-08-28 Kyorin Seiyaku Kk 7-(4-substituted 3- cyclopropylaminomethyl-1- pyrrolidinyl) q uinolonecarboxylic acid derivative
SA112330992B1 (en) 2011-11-10 2015-09-13 كيورين فارماسوتيكال كو.، ليمتد Crystalline form of the 7-{(3S,4S)-3 [(cyclopropylamino)methyl]-4- fluoropyrrolidine-1-YL}-6-fluoro-1-(2-fluoroethyl)-8-methoxy-4-OXO- 1,4-dihydroquinoline-3-carboxylic acid
US20180042918A1 (en) * 2015-03-13 2018-02-15 Kyorin Pharmaceutical Co., Ltd. Respiratory infection treating agent
CA2987879A1 (en) 2015-06-02 2016-12-08 Kyorin Pharmaceutical Co., Ltd. Aqueous drug

Also Published As

Publication number Publication date
CN116549446A (en) 2023-08-08
WO2018230686A1 (en) 2018-12-20

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