EA201991730A1 - N - {[2- (PIPERIDIN-1-IL) Phenyl] (Phenyl) Methyl} -2- (3-OXO-3,4-DIHYDRO-2H-1,4-Benzoxazazin-7-IL) ACETAMIDE DERIVATIVES AND RELATED COMPOUNDS AS ROR-GAMMA MODULATORS FOR TREATMENT OF AUTOIMMUNE DISEASES - Google Patents

N - {[2- (PIPERIDIN-1-IL) Phenyl] (Phenyl) Methyl} -2- (3-OXO-3,4-DIHYDRO-2H-1,4-Benzoxazazin-7-IL) ACETAMIDE DERIVATIVES AND RELATED COMPOUNDS AS ROR-GAMMA MODULATORS FOR TREATMENT OF AUTOIMMUNE DISEASES

Info

Publication number
EA201991730A1
EA201991730A1 EA201991730A EA201991730A EA201991730A1 EA 201991730 A1 EA201991730 A1 EA 201991730A1 EA 201991730 A EA201991730 A EA 201991730A EA 201991730 A EA201991730 A EA 201991730A EA 201991730 A1 EA201991730 A1 EA 201991730A1
Authority
EA
Eurasian Patent Office
Prior art keywords
phenyl
ror
piperidin
dihydro
oxo
Prior art date
Application number
EA201991730A
Other languages
Russian (ru)
Inventor
Жан-Франсуа Деломель
Энрико Перспикас
Заухер Майд
Пэгги Паррош
Роберт Вальчак
Original Assignee
Женфит
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Женфит filed Critical Женфит
Priority claimed from PCT/EP2018/052172 external-priority patent/WO2018138362A1/en
Publication of EA201991730A1 publication Critical patent/EA201991730A1/en

Links

Landscapes

  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Изобретение предоставляет, например, N-{[2-(пиперидин-1-ил)фенил](фенил)метил}-2-(3-оксо-3,4-дигидро-2H-1,4-бензоксазин-7-ил)ацетамидные производные и родственные соединения в качестве модуляторов ROR-гамма для лечения аутоиммунных заболеваний, аутоиммунно-ассоциированных заболеваний, воспалительных заболеваний, нарушений обмена веществ, фиброзных заболеваний или холестатических заболеваний, таких как артрит и астма.The invention provides, for example, N - {[2- (piperidin-1-yl) phenyl] (phenyl) methyl} -2- (3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl ) acetamide derivatives and related compounds as ROR-gamma modulators for the treatment of autoimmune diseases, autoimmune-associated diseases, inflammatory diseases, metabolic disorders, fibrotic diseases or cholestatic diseases such as arthritis and asthma.

EA201991730A 2017-06-29 2018-01-29 N - {[2- (PIPERIDIN-1-IL) Phenyl] (Phenyl) Methyl} -2- (3-OXO-3,4-DIHYDRO-2H-1,4-Benzoxazazin-7-IL) ACETAMIDE DERIVATIVES AND RELATED COMPOUNDS AS ROR-GAMMA MODULATORS FOR TREATMENT OF AUTOIMMUNE DISEASES EA201991730A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP17178888 2017-06-29
PCT/EP2018/052172 WO2018138362A1 (en) 2017-01-27 2018-01-29 N-{[2-(piperidin-1-yl)phenyl](phenyl)methyl}-2-(3-oxo-3,4-dihydro-2h-1,4-benzoxa zin-7-yl)acetamide derivatives and related compounds as ror-gamma modulators for treating autoimmune diseases

Publications (1)

Publication Number Publication Date
EA201991730A1 true EA201991730A1 (en) 2019-12-30

Family

ID=59258142

Family Applications (1)

Application Number Title Priority Date Filing Date
EA201991730A EA201991730A1 (en) 2017-06-29 2018-01-29 N - {[2- (PIPERIDIN-1-IL) Phenyl] (Phenyl) Methyl} -2- (3-OXO-3,4-DIHYDRO-2H-1,4-Benzoxazazin-7-IL) ACETAMIDE DERIVATIVES AND RELATED COMPOUNDS AS ROR-GAMMA MODULATORS FOR TREATMENT OF AUTOIMMUNE DISEASES

Country Status (1)

Country Link
EA (1) EA201991730A1 (en)

Similar Documents

Publication Publication Date Title
PH12019501684A1 (en) N-[2-(piperidin-1-yl)phenyl](phenyl)methyl-2-(3-oxo-3,4-dihydro-2h-1,4-benzoxa zin-7-yl)acetamide derivatives and related compounds as ror-gamma modulators for treating autoimmune diseases
EA201890325A1 (en) PEPTIDE INHIBITORS OF INTERLEUKIN-23 RECEPTOR AND THEIR APPLICATION FOR THE TREATMENT OF INFLAMMATORY DISEASES
EA201891201A1 (en) COMPOSITIONS CONTAINING BACTERIAL STRAINS
EA202091479A1 (en) ARYL- AND HETEROARYL-SUBSTITUTED INDOL COMPOUNDS
EA201890049A1 (en) COMPOSITIONS CONTAINING BACTERIAL STRAINS
GEP20227369B (en) Antibodies specific for hyperphosphorylated tau and methods of use thereof
EA201890256A1 (en) 2-AMINO-3-Fluoro-3- (Fluoromethyl) -6-Methyl-6-phenyl-3,4,5,6-TETRAHYDROPYRIDINE AS BACE1 INHIBITORS
CY1120846T1 (en) 2-AMINO-6- (DIFTHOROMETHYL) -5,5-DIFFORRO-6-PHENYL-3,4,5,6-TETRAHYDROPYRIDINE AS INHIBITORS BACE1
DK3681500T3 (en) USE OF PILOCARPINE HYDROCHLORIDE FOR THE TREATMENT OF PRESBYOPIA
PE20181074A1 (en) HETEROAROMATIC COMPOUNDS AS BTK INHIBITORS
DK3609529T3 (en) RNA FOR THE TREATMENT OF AUTOIMMUNE DISEASES
EA201790892A1 (en) CRYSTAL FORMS OF 5-CHLOR-N4- [2- (DIMETHYLPHOSPHORIL) PHENYL] -N2- {2-METHOXY-4- [4- (4-METHILPIPERAZIN-1-IL) PIPERIDIN-1-IL]} PYRIMIDIN-1-IL -DIAMINE
EA201792604A1 (en) AUTOTAXIN INHIBITORS AND THEIR APPLICATIONS
EA200970818A1 (en) HETEROCYCLIC COMPOUNDS CONTAINING THEIR COMPOSITIONS AND METHODS OF THEIR APPLICATION
EA201790600A1 (en) MODULATING P2X7 N-ACYL TRIAZOLOPIRASINS
EA201691367A1 (en) CRYSTAL SHAPES OF DIMALEATE AFATINIB
EA201790206A1 (en) NEW 2,5-SUBSTITUTED PYRIMIDINES AS PDE4 INHIBITORS
EA201791367A1 (en) 2,3,4,5-TETRAHYDROPYRIDIN-6-AMINE AND 3,4-DIHYDRO-2H-PIRROL-5-AMIN COMPOUNDS - BETA SECRETASE INHIBITORS
PH12016501941A1 (en) Use of heterocyclic compounds for controlling nematodes
EA201890208A1 (en) HERBICID-ACTIVE DERIVATIVES N- (1,3,4-OXADIAZOL-2-IL) ARILKARBOXAMID
EA202091337A1 (en) MYST FAMILY HISTONACETYLTRANSFERASE INHIBITORS
DK3473337T3 (en) PROCEDURE FOR MANUFACTURE OF SUPPORTED PLATINUM PARTICLES
EA201790209A1 (en) NEW 2.5-SUBSTITUTED PYRIMIDINES AS PDE INHIBITORS
DK3724173T3 (en) Compounds for the treatment of neuromuscular disorders
DK3658547T3 (en) PROCESS FOR THE PREPARATION OF N-(5-(4-(4-FORMYL-3-PHENYL-1H-PYRAZOL-1-YL)PYRIMIDIN-2-YLAMINO)-4-METHOXY-2-MORPHOLINOPHENYL)ACRYLAMIDE