EA201991315A1 - CYCLIC DINUCLEOTIDES AS STING AGONISTS (INTERFERON GENE STIMULATOR) - Google Patents
CYCLIC DINUCLEOTIDES AS STING AGONISTS (INTERFERON GENE STIMULATOR)Info
- Publication number
- EA201991315A1 EA201991315A1 EA201991315A EA201991315A EA201991315A1 EA 201991315 A1 EA201991315 A1 EA 201991315A1 EA 201991315 A EA201991315 A EA 201991315A EA 201991315 A EA201991315 A EA 201991315A EA 201991315 A1 EA201991315 A1 EA 201991315A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- interferon gene
- sting agonists
- cyclic dinucleotides
- gene stimulator
- sting
- Prior art date
Links
Abstract
В данном описании предложено соединение, обладающее агонистической активностью STING, которое, как можно ожидать, будет пригодным в качестве средства для профилактики или лечения заболеваний, связанных со STING. Данное изобретение относится к соединению, представленному формулой (I)где каждый символ является таким, как определено в описании, или его солью.In this description, a compound is provided having a STING agonist activity, which can be expected to be useful as an agent for the prophylaxis or treatment of diseases associated with STING. This invention relates to a compound represented by formula (I) wherein each symbol is as defined herein, or a salt thereof.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201762589300P | 2017-11-21 | 2017-11-21 | |
PCT/IB2017/057588 WO2018100558A2 (en) | 2016-12-01 | 2017-12-01 | Cyclic dinucleotide |
Publications (2)
Publication Number | Publication Date |
---|---|
EA201991315A1 true EA201991315A1 (en) | 2019-12-30 |
EA038805B1 EA038805B1 (en) | 2021-10-21 |
Family
ID=69061877
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA201991315A EA038805B1 (en) | 2017-11-21 | 2017-12-01 | Cyclic dinucleotides as sting (stimulator of interferon genes) agonists |
Country Status (1)
Country | Link |
---|---|
EA (1) | EA038805B1 (en) |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2014179335A1 (en) * | 2013-04-29 | 2014-11-06 | Memorial Sloan Kettering Cancer Center | Compositions and methods for altering second messenger signaling |
ES2754269T3 (en) * | 2013-05-18 | 2020-04-16 | Aduro Biotech Inc | Compositions and Activation Methods of "Interferon Gene Stimulator-dependent" Signaling |
EP3546473A1 (en) * | 2014-12-16 | 2019-10-02 | Kayla Therapeutics | Cyclic [(2',5')p(3',5')p]-dinucleotides for cytokine induction |
WO2017027645A1 (en) * | 2015-08-13 | 2017-02-16 | Merck Sharp & Dohme Corp. | Cyclic di-nucleotide compounds as sting agonists |
WO2017161349A1 (en) * | 2016-03-18 | 2017-09-21 | Immune Sensor, Llc | Cyclic di-nucleotide compounds and methods of use |
-
2017
- 2017-12-01 EA EA201991315A patent/EA038805B1/en unknown
Also Published As
Publication number | Publication date |
---|---|
EA038805B1 (en) | 2021-10-21 |
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