EA201990074A1 - HETEROCYCLIC COMPOUNDS AS IMMUNOMODULATORS - Google Patents

HETEROCYCLIC COMPOUNDS AS IMMUNOMODULATORS

Info

Publication number
EA201990074A1
EA201990074A1 EA201990074A EA201990074A EA201990074A1 EA 201990074 A1 EA201990074 A1 EA 201990074A1 EA 201990074 A EA201990074 A EA 201990074A EA 201990074 A EA201990074 A EA 201990074A EA 201990074 A1 EA201990074 A1 EA 201990074A1
Authority
EA
Eurasian Patent Office
Prior art keywords
immunomodulators
compounds
heterocyclic compounds
alleviation
infections
Prior art date
Application number
EA201990074A
Other languages
Russian (ru)
Inventor
Кайцзюн Сяо
Фэнлэй Чжан
Лянсин У
Вэньцин Яо
Original Assignee
Инсайт Корпорейшн
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Инсайт Корпорейшн filed Critical Инсайт Корпорейшн
Priority claimed from PCT/US2017/038120 external-priority patent/WO2017222976A1/en
Publication of EA201990074A1 publication Critical patent/EA201990074A1/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D515/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen, oxygen, and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D515/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen, oxygen, and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D515/04Ortho-condensed systems

Abstract

Описаны соединения формулы (I), способы применения указанных соединений в качестве иммуномодуляторов, а также фармацевтические композиции, содержащие такие соединения. Указанные соединения пригодны при лечении, предупреждении или облегчении заболеваний или расстройств, таких как рак или инфекции.Compounds of formula (I) are described, methods of using said compounds as immunomodulators, as well as pharmaceutical compositions containing such compounds. These compounds are useful in the treatment, prevention, or alleviation of diseases or disorders, such as cancer or infections.

EA201990074A 2016-09-19 2017-06-19 HETEROCYCLIC COMPOUNDS AS IMMUNOMODULATORS EA201990074A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201662396353P 2016-09-19 2016-09-19
PCT/US2017/038120 WO2017222976A1 (en) 2016-06-20 2017-06-19 Heterocyclic compounds as immunomodulators

Publications (1)

Publication Number Publication Date
EA201990074A1 true EA201990074A1 (en) 2019-07-31

Family

ID=67399620

Family Applications (1)

Application Number Title Priority Date Filing Date
EA201990074A EA201990074A1 (en) 2016-09-19 2017-06-19 HETEROCYCLIC COMPOUNDS AS IMMUNOMODULATORS

Country Status (1)

Country Link
EA (1) EA201990074A1 (en)

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