EA201791835A3 - PROTEAS INHIBITORS - Google Patents

PROTEAS INHIBITORS

Info

Publication number
EA201791835A3
EA201791835A3 EA201791835A EA201791835A EA201791835A3 EA 201791835 A3 EA201791835 A3 EA 201791835A3 EA 201791835 A EA201791835 A EA 201791835A EA 201791835 A EA201791835 A EA 201791835A EA 201791835 A3 EA201791835 A3 EA 201791835A3
Authority
EA
Eurasian Patent Office
Prior art keywords
present
inhibitors
proteas
proteas inhibitors
methods
Prior art date
Application number
EA201791835A
Other languages
Russian (ru)
Other versions
EA034601B1 (en
EA201791835A2 (en
Inventor
Эдвард Дж. Олхава
Михаела Д. Данка
Original Assignee
Милленниум Фармасьютикалз, Инк.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Милленниум Фармасьютикалз, Инк. filed Critical Милленниум Фармасьютикалз, Инк.
Priority to EA201791835A priority Critical patent/EA034601B1/en
Publication of EA201791835A2 publication Critical patent/EA201791835A2/en
Publication of EA201791835A3 publication Critical patent/EA201791835A3/en
Publication of EA034601B1 publication Critical patent/EA034601B1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic System
    • C07F5/02—Boron compounds

Abstract

В настоящем изобретении предложены новые соединения, подходящие для применения в качестве ингибиторов протеасом. В настоящем изобретении также предложены фармацевтические композиции, содержащие соединения согласно настоящему изобретению, и способы применения указанных композиций для лечения различных заболеваний.In the present invention proposed new compounds suitable for use as proteasome inhibitors. The present invention also provides pharmaceutical compositions containing the compounds of the present invention, and methods of using the compositions for treating various diseases.

EA201791835A 2007-08-06 2007-08-06 Process for producing boronic acids EA034601B1 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
EA201791835A EA034601B1 (en) 2007-08-06 2007-08-06 Process for producing boronic acids

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EA201791835A EA034601B1 (en) 2007-08-06 2007-08-06 Process for producing boronic acids

Publications (3)

Publication Number Publication Date
EA201791835A2 EA201791835A2 (en) 2018-05-31
EA201791835A3 true EA201791835A3 (en) 2018-09-28
EA034601B1 EA034601B1 (en) 2020-02-25

Family

ID=62217545

Family Applications (1)

Application Number Title Priority Date Filing Date
EA201791835A EA034601B1 (en) 2007-08-06 2007-08-06 Process for producing boronic acids

Country Status (1)

Country Link
EA (1) EA034601B1 (en)

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6083903A (en) * 1994-10-28 2000-07-04 Leukosite, Inc. Boronic ester and acid compounds, synthesis and uses
JP4162491B2 (en) * 2001-01-25 2008-10-08 アメリカ合衆国 Boronic acid compound preparation
US7576206B2 (en) * 2003-08-14 2009-08-18 Cephalon, Inc. Proteasome inhibitors and methods of using the same
UA90108C2 (en) * 2004-03-30 2010-04-12 Мілленніум Фармасьютікалз, Інк. Synthesis of boronic ester and acid compounds

Also Published As

Publication number Publication date
EA034601B1 (en) 2020-02-25
EA201791835A2 (en) 2018-05-31

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Legal Events

Date Code Title Description
MM4A Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s)

Designated state(s): AM AZ KG MD TJ TM