EA201791448A1 - ANESTHETIC BASED ON TETRAKAINE - Google Patents
ANESTHETIC BASED ON TETRAKAINEInfo
- Publication number
- EA201791448A1 EA201791448A1 EA201791448A EA201791448A EA201791448A1 EA 201791448 A1 EA201791448 A1 EA 201791448A1 EA 201791448 A EA201791448 A EA 201791448A EA 201791448 A EA201791448 A EA 201791448A EA 201791448 A1 EA201791448 A1 EA 201791448A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- tetrakaine
- molars
- tetracaine
- methods
- present
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
- A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
- A61K31/235—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids having an aromatic ring attached to a carboxyl group
- A61K31/24—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids having an aromatic ring attached to a carboxyl group having an amino or nitro group
- A61K31/245—Amino benzoic acid types, e.g. procaine, novocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4174—Arylalkylimidazoles, e.g. oxymetazolin, naphazoline, miconazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0043—Nose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61M—DEVICES FOR INTRODUCING MEDIA INTO, OR ONTO, THE BODY; DEVICES FOR TRANSDUCING BODY MEDIA OR FOR TAKING MEDIA FROM THE BODY; DEVICES FOR PRODUCING OR ENDING SLEEP OR STUPOR
- A61M11/00—Sprayers or atomisers specially adapted for therapeutic purposes
- A61M11/006—Sprayers or atomisers specially adapted for therapeutic purposes operated by applying mechanical pressure to the liquid to be sprayed or atomised
- A61M11/007—Syringe-type or piston-type sprayers or atomisers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61M—DEVICES FOR INTRODUCING MEDIA INTO, OR ONTO, THE BODY; DEVICES FOR TRANSDUCING BODY MEDIA OR FOR TAKING MEDIA FROM THE BODY; DEVICES FOR PRODUCING OR ENDING SLEEP OR STUPOR
- A61M19/00—Local anaesthesia; Hypothermia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P23/00—Anaesthetics
- A61P23/02—Local anaesthetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61M—DEVICES FOR INTRODUCING MEDIA INTO, OR ONTO, THE BODY; DEVICES FOR TRANSDUCING BODY MEDIA OR FOR TAKING MEDIA FROM THE BODY; DEVICES FOR PRODUCING OR ENDING SLEEP OR STUPOR
- A61M11/00—Sprayers or atomisers specially adapted for therapeutic purposes
- A61M11/006—Sprayers or atomisers specially adapted for therapeutic purposes operated by applying mechanical pressure to the liquid to be sprayed or atomised
- A61M11/008—Sprayers or atomisers specially adapted for therapeutic purposes operated by applying mechanical pressure to the liquid to be sprayed or atomised by squeezing, e.g. using a flexible bottle or a bulb
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61M—DEVICES FOR INTRODUCING MEDIA INTO, OR ONTO, THE BODY; DEVICES FOR TRANSDUCING BODY MEDIA OR FOR TAKING MEDIA FROM THE BODY; DEVICES FOR PRODUCING OR ENDING SLEEP OR STUPOR
- A61M2202/00—Special media to be introduced, removed or treated
- A61M2202/0007—Special media to be introduced, removed or treated introduced into the body
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61M—DEVICES FOR INTRODUCING MEDIA INTO, OR ONTO, THE BODY; DEVICES FOR TRANSDUCING BODY MEDIA OR FOR TAKING MEDIA FROM THE BODY; DEVICES FOR PRODUCING OR ENDING SLEEP OR STUPOR
- A61M2202/00—Special media to be introduced, removed or treated
- A61M2202/04—Liquids
- A61M2202/0468—Liquids non-physiological
- A61M2202/048—Anaesthetics
Abstract
Настоящее изобретение связано с анестезирующими составами на основе тетракаина и со способами их применения. Настоящее изобретение также связано со стоматологическими анестезирующими составами на основе тетракаина и со способами обезболивания верхних задних моляров верхнечелюстной зубной дуги и тканей вокруг верхнечелюстных задних моляров, включая дистальную половину первого моляра, второго и третьего моляров с применением этих составов.The present invention relates to tetracaine based anesthetic formulations and methods for their use. The present invention is also associated with tetracaine-based dental anesthetics and methods of anesthetizing the upper posterior molars of the maxillary dental arch and the tissues around the maxillary posterior molars, including the distal half of the first molar, second and third molars using these compositions.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201462096287P | 2014-12-23 | 2014-12-23 | |
PCT/US2015/000209 WO2016105482A1 (en) | 2014-12-23 | 2015-12-23 | Tetracaine-based anesthetic |
Publications (1)
Publication Number | Publication Date |
---|---|
EA201791448A1 true EA201791448A1 (en) | 2017-11-30 |
Family
ID=55237886
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA201791448A EA201791448A1 (en) | 2014-12-23 | 2015-12-23 | ANESTHETIC BASED ON TETRAKAINE |
Country Status (11)
Country | Link |
---|---|
EP (1) | EP3236941A1 (en) |
JP (1) | JP2017538777A (en) |
KR (1) | KR20170102892A (en) |
CN (1) | CN107249568A (en) |
AU (1) | AU2015371291A1 (en) |
BR (1) | BR112017013373A2 (en) |
CA (1) | CA2971156A1 (en) |
EA (1) | EA201791448A1 (en) |
IL (1) | IL253125A0 (en) |
MX (1) | MX2017008516A (en) |
WO (1) | WO2016105482A1 (en) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2019191200A1 (en) | 2018-03-27 | 2019-10-03 | American Genomics, Llc | Method and formulation for producing anesthesia of internal aspect of eye wall by topical application |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US8580282B2 (en) * | 2009-04-03 | 2013-11-12 | St. Renatus, Llc | Dental anesthetic comprising tetracaine and a vasoconstrictor for intranasal administration |
-
2015
- 2015-12-23 AU AU2015371291A patent/AU2015371291A1/en not_active Abandoned
- 2015-12-23 WO PCT/US2015/000209 patent/WO2016105482A1/en active Application Filing
- 2015-12-23 MX MX2017008516A patent/MX2017008516A/en unknown
- 2015-12-23 EA EA201791448A patent/EA201791448A1/en unknown
- 2015-12-23 BR BR112017013373A patent/BR112017013373A2/en not_active Application Discontinuation
- 2015-12-23 KR KR1020177019688A patent/KR20170102892A/en unknown
- 2015-12-23 JP JP2017533578A patent/JP2017538777A/en active Pending
- 2015-12-23 CA CA2971156A patent/CA2971156A1/en not_active Abandoned
- 2015-12-23 CN CN201580075138.0A patent/CN107249568A/en active Pending
- 2015-12-23 EP EP15828784.7A patent/EP3236941A1/en not_active Withdrawn
-
2017
- 2017-06-22 IL IL253125A patent/IL253125A0/en unknown
Also Published As
Publication number | Publication date |
---|---|
EP3236941A1 (en) | 2017-11-01 |
WO2016105482A9 (en) | 2017-08-03 |
BR112017013373A2 (en) | 2018-01-02 |
KR20170102892A (en) | 2017-09-12 |
IL253125A0 (en) | 2017-08-31 |
MX2017008516A (en) | 2017-09-19 |
JP2017538777A (en) | 2017-12-28 |
CN107249568A (en) | 2017-10-13 |
CA2971156A1 (en) | 2016-06-30 |
AU2015371291A9 (en) | 2017-08-24 |
AU2015371291A1 (en) | 2017-08-03 |
WO2016105482A1 (en) | 2016-06-30 |
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