EA201591218A1 - Способы и композиции для введения оксибутинина - Google Patents
Способы и композиции для введения оксибутининаInfo
- Publication number
- EA201591218A1 EA201591218A1 EA201591218A EA201591218A EA201591218A1 EA 201591218 A1 EA201591218 A1 EA 201591218A1 EA 201591218 A EA201591218 A EA 201591218A EA 201591218 A EA201591218 A EA 201591218A EA 201591218 A1 EA201591218 A1 EA 201591218A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- salt
- agents
- compositions
- methods
- oxybutynin
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/007—Pulmonary tract; Aromatherapy
- A61K9/0073—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy
- A61K9/0075—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy for inhalation via a dry powder inhaler [DPI], e.g. comprising micronized drug mixed with lactose carrier particles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
- A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
- A61K31/216—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acids having aromatic rings, e.g. benactizyne, clofibrate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Pulmonology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Epidemiology (AREA)
- Otolaryngology (AREA)
- Emergency Medicine (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Настоящее изобретение касается способов и композиций для лечения заболевания легких, включающих доставку непосредственно в легкие пациента терапевтически эффективного количества оксибутинина в комбинации с одним или более фармацевтически эффективными средствами. Оксибутинин может быть выбран из группы, состоящей, но не в порядке ограничения, из ксинафоатной соли, пальмитатной соли, соли памовой кислоты, резинатной соли, лауратной соли и других солей. Фармацевтически эффективные средства включают бронходилататоры, противовоспалительные средства, кортикостероиды, средство для реверсии действия кортикостероидов или средства альвеолярного роста или другие средства, выбираемые из ингибиторов протеиназы или протеазы.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US13/728,706 US9119777B2 (en) | 2008-05-30 | 2012-12-27 | Methods and compositions for administration of oxybutynin |
PCT/US2013/074759 WO2014105446A1 (en) | 2012-12-27 | 2013-12-12 | Methods and compositions for administration of oxybutynin |
Publications (1)
Publication Number | Publication Date |
---|---|
EA201591218A1 true EA201591218A1 (ru) | 2015-11-30 |
Family
ID=51021931
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA201591218A EA201591218A1 (ru) | 2012-12-27 | 2013-12-12 | Способы и композиции для введения оксибутинина |
Country Status (15)
Country | Link |
---|---|
EP (1) | EP2938329A4 (ru) |
JP (1) | JP2016504358A (ru) |
KR (1) | KR20150100902A (ru) |
CN (1) | CN104955444A (ru) |
AR (1) | AR094287A1 (ru) |
AU (1) | AU2013368298B2 (ru) |
BR (1) | BR112015015421A2 (ru) |
CA (1) | CA2895955A1 (ru) |
EA (1) | EA201591218A1 (ru) |
HK (2) | HK1215396A1 (ru) |
IL (1) | IL239623A0 (ru) |
MX (1) | MX2015008333A (ru) |
NZ (1) | NZ628479A (ru) |
UY (1) | UY35230A (ru) |
WO (1) | WO2014105446A1 (ru) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US20190046493A1 (en) * | 2016-02-25 | 2019-02-14 | Hisamitsu Pharmaceutical Co., Inc. | Liquid external preparation |
Family Cites Families (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP2003500354A (ja) * | 1999-05-20 | 2003-01-07 | セプラコール, インク. | S−オキシブチニンを用いる喘息の治療方法 |
US6339107B1 (en) * | 2000-08-02 | 2002-01-15 | Syntex (U.S.A.) Llc | Methods for treatment of Emphysema using 13-cis retinoic acid |
AU2003267796A1 (en) * | 2002-10-29 | 2004-05-25 | Pharmacia & Upjohn Company Llc | Quaternary ammonium compounds |
GB0410398D0 (en) * | 2004-05-10 | 2004-06-16 | Arakis Ltd | The treatment of respiratory disease |
EP1817034A1 (en) * | 2004-10-25 | 2007-08-15 | Schering Corporation | M1 and/or m3 receptor antagonists in combination with other actives for treating respiratory disorders |
US8415390B2 (en) * | 2008-05-30 | 2013-04-09 | Microdose Therapeutx, Inc. | Methods and compositions for administration of oxybutynin |
EP3311820A1 (en) * | 2008-02-26 | 2018-04-25 | Sunovion Respiratory Development Inc. | Method and system for the treatment of chronic obstructive pulmonary disease with nebulized anticholinergic administrations |
AU2010260513A1 (en) * | 2009-06-16 | 2012-02-02 | Wen Tan | Use of R-Bambuterol as inhaled medicament and combination therapies for treatment of respiratory disorders |
GB0918450D0 (en) * | 2009-10-21 | 2009-12-09 | Innovata Ltd | Composition |
CN102858326A (zh) * | 2010-04-01 | 2013-01-02 | 奇斯药制品公司 | 用于制备可吸入干粉所用的载体颗粒的方法 |
EP2621588A4 (en) * | 2010-09-27 | 2014-09-03 | Microdose Therapeutx Inc | METHODS AND COMPOSITIONS FOR TREATING DISEASE USING INHALATION |
-
2013
- 2013-12-12 AU AU2013368298A patent/AU2013368298B2/en not_active Ceased
- 2013-12-12 EA EA201591218A patent/EA201591218A1/ru unknown
- 2013-12-12 EP EP13867956.8A patent/EP2938329A4/en not_active Withdrawn
- 2013-12-12 CA CA2895955A patent/CA2895955A1/en not_active Abandoned
- 2013-12-12 CN CN201380068230.5A patent/CN104955444A/zh active Pending
- 2013-12-12 NZ NZ628479A patent/NZ628479A/en not_active IP Right Cessation
- 2013-12-12 JP JP2015550444A patent/JP2016504358A/ja active Pending
- 2013-12-12 KR KR1020157020335A patent/KR20150100902A/ko not_active Application Discontinuation
- 2013-12-12 BR BR112015015421A patent/BR112015015421A2/pt not_active IP Right Cessation
- 2013-12-12 MX MX2015008333A patent/MX2015008333A/es unknown
- 2013-12-12 WO PCT/US2013/074759 patent/WO2014105446A1/en active Application Filing
- 2013-12-20 UY UY0001035230A patent/UY35230A/es not_active Application Discontinuation
- 2013-12-27 AR ARP130105037A patent/AR094287A1/es unknown
-
2015
- 2015-06-24 IL IL239623A patent/IL239623A0/en unknown
-
2016
- 2016-03-23 HK HK16103431.3A patent/HK1215396A1/zh unknown
- 2016-04-25 HK HK16104715.8A patent/HK1216843A1/zh unknown
Also Published As
Publication number | Publication date |
---|---|
CN104955444A (zh) | 2015-09-30 |
AU2013368298B2 (en) | 2016-08-11 |
IL239623A0 (en) | 2015-08-31 |
CA2895955A1 (en) | 2014-07-03 |
BR112015015421A2 (pt) | 2017-07-11 |
NZ628479A (en) | 2016-06-24 |
MX2015008333A (es) | 2015-11-09 |
EP2938329A4 (en) | 2016-08-10 |
JP2016504358A (ja) | 2016-02-12 |
HK1216843A1 (zh) | 2016-12-09 |
EP2938329A1 (en) | 2015-11-04 |
KR20150100902A (ko) | 2015-09-02 |
AU2013368298A1 (en) | 2015-07-02 |
UY35230A (es) | 2015-01-30 |
WO2014105446A1 (en) | 2014-07-03 |
HK1215396A1 (zh) | 2016-08-26 |
AR094287A1 (es) | 2015-07-22 |
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