EA201071119A1 - APPLICATION OF HETEROCYCLIC BENZO DERIVATIVES OF SULFAMIDE FOR THE TREATMENT OF ANXIETY DISORDERS - Google Patents

APPLICATION OF HETEROCYCLIC BENZO DERIVATIVES OF SULFAMIDE FOR THE TREATMENT OF ANXIETY DISORDERS

Info

Publication number
EA201071119A1
EA201071119A1 EA201071119A EA201071119A EA201071119A1 EA 201071119 A1 EA201071119 A1 EA 201071119A1 EA 201071119 A EA201071119 A EA 201071119A EA 201071119 A EA201071119 A EA 201071119A EA 201071119 A1 EA201071119 A1 EA 201071119A1
Authority
EA
Eurasian Patent Office
Prior art keywords
sulfamide
treatment
application
anxiety disorders
benzo derivatives
Prior art date
Application number
EA201071119A
Other languages
Russian (ru)
Other versions
EA019544B1 (en
Inventor
Вирджиния Л. Смит-Свинтоски
Original Assignee
Янссен Фармацевтика Н.В.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Янссен Фармацевтика Н.В. filed Critical Янссен Фармацевтика Н.В.
Publication of EA201071119A1 publication Critical patent/EA201071119A1/en
Publication of EA019544B1 publication Critical patent/EA019544B1/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/352Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline 
    • A61K31/3533,4-Dihydrobenzopyrans, e.g. chroman, catechin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/357Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having two or more oxygen atoms in the same ring, e.g. crown ethers, guanadrel
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics

Abstract

Изобретение представляет собой способ лечения тревожного расстройства и родственных патологических расстройств, включающий введение нуждающемуся в этом субъекту терапевтически эффективных количеств одного или более новых гетероциклических бензопроизводных сульфамида формулы (I) и формулы (II), как определяется настоящим документом. Настоящее изобретение направлено на создание способа лечения тревожного расстройства и родственных патологических расстройств, который включает введение монотерапии и в качестве варианта комбинированной терапии по крайней мере одним анксиолитиком.The invention is a method of treating anxiety disorder and related pathological disorders, comprising administering to a subject in need thereof a therapeutically effective amount of one or more new heterocyclic benzene derivatives of sulfamide of formula (I) and formula (II) as defined herein. The present invention is directed to a method for the treatment of anxiety disorder and related pathological disorders, which includes the introduction of monotherapy and as a combination therapy with at least one anxiolytic.

EA201071119A 2008-03-26 2008-03-26 Use of benzo-fused heterocycle sulfamide derivatives for the treatment of anxiety EA019544B1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/US2008/058210 WO2009120189A1 (en) 2008-03-26 2008-03-26 Use of benzo-fused heterocycle sulfamide derivatives for the treatment of anxiety

Publications (2)

Publication Number Publication Date
EA201071119A1 true EA201071119A1 (en) 2011-06-30
EA019544B1 EA019544B1 (en) 2014-04-30

Family

ID=39926425

Family Applications (1)

Application Number Title Priority Date Filing Date
EA201071119A EA019544B1 (en) 2008-03-26 2008-03-26 Use of benzo-fused heterocycle sulfamide derivatives for the treatment of anxiety

Country Status (8)

Country Link
EP (1) EP2276481B1 (en)
KR (1) KR101511574B1 (en)
AU (1) AU2008353489B2 (en)
BR (1) BRPI0822385A2 (en)
EA (1) EA019544B1 (en)
ES (1) ES2517598T3 (en)
UA (1) UA100552C2 (en)
WO (1) WO2009120189A1 (en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8609849B1 (en) 2010-11-30 2013-12-17 Fox Chase Chemical Diversity Center, Inc. Hydroxylated sulfamides exhibiting neuroprotective action and their method of use

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7662271B2 (en) * 2005-12-21 2010-02-16 Chevron U.S.A. Inc. Lubricating oil with high oxidation stability
US20070155824A1 (en) * 2005-12-19 2007-07-05 Smith-Swintosky Virginia L Use of benzo-fused heterocycle sulfamide derivatives for disease modification / epileptogenesis
US8691867B2 (en) * 2005-12-19 2014-04-08 Janssen Pharmaceutica Nv Use of benzo-fused heterocycle sulfamide derivatives for the treatment of substance abuse and addiction
US20070155827A1 (en) * 2005-12-19 2007-07-05 Smith-Swintosky Virginia L Use of benzo-fused heterocycle sulfamide derivatives for the treatment of depression

Also Published As

Publication number Publication date
EP2276481B1 (en) 2014-07-30
ES2517598T3 (en) 2014-11-03
EP2276481A1 (en) 2011-01-26
AU2008353489B2 (en) 2014-11-27
WO2009120189A1 (en) 2009-10-01
EA019544B1 (en) 2014-04-30
AU2008353489A1 (en) 2009-10-01
KR101511574B1 (en) 2015-04-15
UA100552C2 (en) 2013-01-10
KR20100134052A (en) 2010-12-22
BRPI0822385A2 (en) 2019-09-24

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Legal Events

Date Code Title Description
MM4A Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s)

Designated state(s): AM AZ BY KZ KG MD TJ TM RU