EA200970292A1 - Производные 5-тиоксилопиранозы и их применение в терапии - Google Patents

Производные 5-тиоксилопиранозы и их применение в терапии

Info

Publication number
EA200970292A1
EA200970292A1 EA200970292A EA200970292A EA200970292A1 EA 200970292 A1 EA200970292 A1 EA 200970292A1 EA 200970292 A EA200970292 A EA 200970292A EA 200970292 A EA200970292 A EA 200970292A EA 200970292 A1 EA200970292 A1 EA 200970292A1
Authority
EA
Eurasian Patent Office
Prior art keywords
derivatives
thyoxyl
pyranose
therapy
application
Prior art date
Application number
EA200970292A
Other languages
English (en)
Other versions
EA015067B1 (ru
Inventor
Вероник Барберусс
Дидье Тома
Мишель Бонду
Original Assignee
Лабораториз Фурнье С.А.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Лабораториз Фурнье С.А. filed Critical Лабораториз Фурнье С.А.
Publication of EA200970292A1 publication Critical patent/EA200970292A1/ru
Publication of EA015067B1 publication Critical patent/EA015067B1/ru

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/02—Heterocyclic radicals containing only nitrogen as ring hetero atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Cardiology (AREA)
  • Public Health (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Данное изобретение относится к новым производным 5-тиоксилозы, предпочтительно к производным 5-тиоксилопиранозы, к способу их получения и к применению указанных соединений в качестве активного ингредиента в лекарствах, предназначенных главным образом для лечения или предупреждения тромбоза, или сердечной недостаточности, или тромбоэмболических заболеваний.
EA200970292A 2006-09-27 2007-09-26 Производные 5-тиоксилопиранозы и их применение в терапии EA015067B1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0653961A FR2906248B1 (fr) 2006-09-27 2006-09-27 Nouveaux derives de 5-thioxylopyranose
PCT/FR2007/052005 WO2008037922A1 (fr) 2006-09-27 2007-09-26 Derives de 5 - thioxylopyranose et leur utilisation en therapeutique

Publications (2)

Publication Number Publication Date
EA200970292A1 true EA200970292A1 (ru) 2009-10-30
EA015067B1 EA015067B1 (ru) 2011-04-29

Family

ID=38042600

Family Applications (1)

Application Number Title Priority Date Filing Date
EA200970292A EA015067B1 (ru) 2006-09-27 2007-09-26 Производные 5-тиоксилопиранозы и их применение в терапии

Country Status (15)

Country Link
US (1) US8093394B2 (ru)
EP (1) EP2066683B1 (ru)
JP (1) JP5242574B2 (ru)
CN (1) CN101535329B (ru)
AT (1) ATE486881T1 (ru)
AU (1) AU2007301837B2 (ru)
CA (1) CA2665907A1 (ru)
DE (1) DE602007010326D1 (ru)
EA (1) EA015067B1 (ru)
ES (1) ES2355802T3 (ru)
FR (1) FR2906248B1 (ru)
HK (1) HK1131990A1 (ru)
MX (1) MX2009003253A (ru)
PL (1) PL2066683T3 (ru)
WO (1) WO2008037922A1 (ru)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2010232729A1 (en) 2009-03-31 2011-10-20 Arqule, Inc. Substituted indolo-pyridinone compounds

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2492830A1 (fr) 1980-10-29 1982-04-30 Sori Soc Rech Ind Nouveaux composes appartenant a la famille des benzoyl- et a-hydroxybenzyl-phenyl-osides, leur procede de preparation et leur application en therapeutique
FR2614893B1 (fr) * 1987-05-04 1989-12-22 Fournier Innovation Synergie Nouveaux b-d-phenyl-thioxylosides, leur procede de preparation et leur application en therapeutique
IE63544B1 (en) 1988-10-18 1995-05-17 Fournier Ind & Sante Novel Beta-d-phenylthioxylosides their method of preparation and their use in therapy
FR2637913B1 (fr) 1988-10-19 1994-06-03 Rhone Poulenc Chimie Procede de production de polysaccharides par fermentation d'une source hydrocarbonee a l'aide de microorganismes
DK0421829T3 (da) 1989-09-22 1995-01-16 Fournier Ind & Sante Nye benzopyranon-beta-D-thioxylosider, fremgangsmåde til deres fremstilling og deres terapeutiske anvendelse
FR2824559B1 (fr) * 2001-05-11 2004-02-13 Fournier Lab Sa Nouveaux derives 5-thio-beta-xylopyronasides, procede de preparation, compositions pharmaceutiques les contenant et leur utilisation en therapeutique
EP1609799A4 (en) * 2003-04-01 2008-10-29 Taisho Pharmaceutical Co Ltd HETEROARYL-5-THIO-BETA-D-GLUCOPYRANOSIDE DERIVATIVES AND AGENTS AGAINST DIABETES THEREOF
FR2860234B1 (fr) * 2003-09-25 2005-12-23 Fournier Lab Sa Nouveaux derives 666 du thioxylose
FR2883561B1 (fr) * 2005-03-25 2009-03-20 Fournier S A Sa Lab Nouveaux composes derives du 5-thioxylose et leur utilisation therapeutique

Also Published As

Publication number Publication date
US20090182013A1 (en) 2009-07-16
AU2007301837A1 (en) 2008-04-03
JP2010504947A (ja) 2010-02-18
MX2009003253A (es) 2009-04-08
ATE486881T1 (de) 2010-11-15
HK1131990A1 (en) 2010-02-12
AU2007301837B2 (en) 2012-09-27
WO2008037922A1 (fr) 2008-04-03
DE602007010326D1 (de) 2010-12-16
US8093394B2 (en) 2012-01-10
CN101535329B (zh) 2012-11-21
FR2906248B1 (fr) 2008-12-26
PL2066683T3 (pl) 2011-04-29
ES2355802T3 (es) 2011-03-31
CN101535329A (zh) 2009-09-16
EP2066683A1 (fr) 2009-06-10
EP2066683B1 (fr) 2010-11-03
FR2906248A1 (fr) 2008-03-28
CA2665907A1 (fr) 2008-04-03
JP5242574B2 (ja) 2013-07-24
EA015067B1 (ru) 2011-04-29

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Legal Events

Date Code Title Description
MM4A Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s)

Designated state(s): AM AZ BY KZ KG MD TJ TM

MM4A Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s)

Designated state(s): RU