EA200701741A1 - Композиция, содержащая окаперидон - Google Patents
Композиция, содержащая окаперидонInfo
- Publication number
- EA200701741A1 EA200701741A1 EA200701741A EA200701741A EA200701741A1 EA 200701741 A1 EA200701741 A1 EA 200701741A1 EA 200701741 A EA200701741 A EA 200701741A EA 200701741 A EA200701741 A EA 200701741A EA 200701741 A1 EA200701741 A1 EA 200701741A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- okaperidone
- relates
- present
- okaperidon
- composition containing
- Prior art date
Links
- 239000000203 mixture Substances 0.000 title abstract 4
- 230000001225 therapeutic effect Effects 0.000 abstract 2
- ZZQNEJILGNNOEP-UHFFFAOYSA-N Ocaperidone Chemical compound FC1=CC=C2C(C3CCN(CC3)CCC3=C(C)N=C4N(C3=O)C=CC=C4C)=NOC2=C1 ZZQNEJILGNNOEP-UHFFFAOYSA-N 0.000 abstract 1
- 239000013543 active substance Substances 0.000 abstract 1
- 230000000561 anti-psychotic effect Effects 0.000 abstract 1
- 239000012736 aqueous medium Substances 0.000 abstract 1
- 239000002552 dosage form Substances 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 229940079593 drug Drugs 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 229950010634 ocaperidone Drugs 0.000 abstract 1
- 229920000642 polymer Polymers 0.000 abstract 1
- 238000002360 preparation method Methods 0.000 abstract 1
- 230000007928 solubilization Effects 0.000 abstract 1
- 238000005063 solubilization Methods 0.000 abstract 1
- 229920003169 water-soluble polymer Polymers 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0002—Galenical forms characterised by the drug release technique; Application systems commanded by energy
- A61K9/0004—Osmotic delivery systems; Sustained release driven by osmosis, thermal energy or gas
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
- A61K9/209—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat containing drug in at least two layers or in the core and in at least one outer layer
Landscapes
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Epidemiology (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Psychology (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Настоящее изобретение относится к композиции, содержащей окаперидон (как активное вещество) и водорастворимые полимеры в количестве, эффективном для повышения растворимости окаперидона. Кроме того, настоящее изобретение относится к терапевтической системе окаперидона, содержащей компартмент для лекарственной формы, содержащей указанную композицию, а также к процессу ее приготовления и к терапевтическому использованию указанной композиции в качестве антипсихотического лекарства. Настоящее изобретение также относится к солюбилизации окаперидона в водной среде с помощью водорастворимых набухающих полимеров.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP05290332A EP1690540A1 (en) | 2005-02-15 | 2005-02-15 | Composition comprising ocaperidone |
PCT/IB2006/000758 WO2006087639A1 (en) | 2005-02-15 | 2006-02-15 | Composition comprising ocaperidone |
Publications (2)
Publication Number | Publication Date |
---|---|
EA200701741A1 true EA200701741A1 (ru) | 2007-12-28 |
EA013596B1 EA013596B1 (ru) | 2010-06-30 |
Family
ID=34981863
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA200701741A EA013596B1 (ru) | 2005-02-15 | 2006-02-15 | Фармацевтическая система доставки, содержащая окаперидон |
Country Status (12)
Country | Link |
---|---|
US (2) | US20080103159A1 (ru) |
EP (2) | EP1690540A1 (ru) |
JP (1) | JP2008530080A (ru) |
KR (1) | KR20070102557A (ru) |
CN (1) | CN101128203A (ru) |
AU (1) | AU2006215309B2 (ru) |
BR (1) | BRPI0608083A2 (ru) |
CA (1) | CA2595269A1 (ru) |
EA (1) | EA013596B1 (ru) |
MX (1) | MX2007009916A (ru) |
NZ (1) | NZ556626A (ru) |
WO (1) | WO2006087639A1 (ru) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2011067296A1 (en) | 2009-12-01 | 2011-06-09 | Integragen | A combination of eight risk alleles associated with autism |
WO2014042657A1 (en) | 2012-09-17 | 2014-03-20 | Halliburton Energy Services, Inc. | Well tools with semi-permeable barrier for water-swellable material |
Family Cites Families (16)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3845770A (en) | 1972-06-05 | 1974-11-05 | Alza Corp | Osmatic dispensing device for releasing beneficial agent |
US3916899A (en) * | 1973-04-25 | 1975-11-04 | Alza Corp | Osmotic dispensing device with maximum and minimum sizes for the passageway |
US3977404A (en) * | 1975-09-08 | 1976-08-31 | Alza Corporation | Osmotic device having microporous reservoir |
US4111202A (en) * | 1976-11-22 | 1978-09-05 | Alza Corporation | Osmotic system for the controlled and delivery of agent over time |
US4327725A (en) * | 1980-11-25 | 1982-05-04 | Alza Corporation | Osmotic device with hydrogel driving member |
CH668187A5 (de) * | 1986-08-07 | 1988-12-15 | Ciba Geigy Ag | Therapeutisches system mit systemischer wirkung. |
DE3868077D1 (de) * | 1987-01-14 | 1992-03-12 | Ciba Geigy Ag | Therapeutisches system fuer schwerloesliche wirkstoffe. |
IT210468Z2 (it) | 1987-01-21 | 1988-12-30 | Iveco Fiat | Attuatore lineare elettromeccanico per il ribaltamento della cabina di guida di un veicolo industriale |
GB9008850D0 (en) * | 1990-04-19 | 1990-06-13 | Janssen Pharmaceutica Nv | Novel 2,9-disubstituted-4h-pyridol(1,2-a)pyrimidin-4-ones |
US7767708B2 (en) * | 1998-11-04 | 2010-08-03 | Schering-Plough Animal Health Corp. | Growth stimulant compositions |
AU5060499A (en) * | 1999-08-04 | 2001-03-05 | Ranbaxy Laboratories Limited | Hydrodynamically balanced oral drug delivery system |
US6599532B2 (en) * | 2000-01-13 | 2003-07-29 | Osmotica Corp. | Osmotic device containing alprazolam and an antipsychotic agent |
IN190699B (ru) * | 2001-02-02 | 2003-08-16 | Sun Pharmaceutical Ind Ltd | |
US6713479B2 (en) * | 2001-03-02 | 2004-03-30 | Sepracor Inc. | Piperidine-piperazine ligands for neurotransmitter receptors |
EP1411901B1 (en) * | 2001-07-04 | 2010-08-18 | Sun Pharma Advanced Research Company Ltd | Gastric retention controlled drug delivery system |
CA2409552A1 (en) * | 2001-10-25 | 2003-04-25 | Depomed, Inc. | Gastric retentive oral dosage form with restricted drug release in the lower gastrointestinal tract |
-
2005
- 2005-02-15 EP EP05290332A patent/EP1690540A1/en not_active Withdrawn
-
2006
- 2006-02-15 CN CNA2006800048733A patent/CN101128203A/zh active Pending
- 2006-02-15 KR KR1020077018864A patent/KR20070102557A/ko not_active Application Discontinuation
- 2006-02-15 WO PCT/IB2006/000758 patent/WO2006087639A1/en active Application Filing
- 2006-02-15 BR BRPI0608083-9A patent/BRPI0608083A2/pt not_active IP Right Cessation
- 2006-02-15 EP EP06710611A patent/EP1861103A1/en not_active Withdrawn
- 2006-02-15 MX MX2007009916A patent/MX2007009916A/es unknown
- 2006-02-15 NZ NZ556626A patent/NZ556626A/en not_active IP Right Cessation
- 2006-02-15 CA CA002595269A patent/CA2595269A1/en not_active Abandoned
- 2006-02-15 US US11/884,296 patent/US20080103159A1/en not_active Abandoned
- 2006-02-15 JP JP2007554679A patent/JP2008530080A/ja active Pending
- 2006-02-15 EA EA200701741A patent/EA013596B1/ru not_active IP Right Cessation
- 2006-02-15 AU AU2006215309A patent/AU2006215309B2/en not_active Ceased
-
2011
- 2011-09-21 US US13/238,577 patent/US20120009266A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
AU2006215309B2 (en) | 2011-03-24 |
AU2006215309A1 (en) | 2006-08-24 |
BRPI0608083A2 (pt) | 2009-11-10 |
KR20070102557A (ko) | 2007-10-18 |
US20080103159A1 (en) | 2008-05-01 |
CA2595269A1 (en) | 2006-08-24 |
JP2008530080A (ja) | 2008-08-07 |
EP1690540A1 (en) | 2006-08-16 |
EA013596B1 (ru) | 2010-06-30 |
US20120009266A1 (en) | 2012-01-12 |
WO2006087639A1 (en) | 2006-08-24 |
NZ556626A (en) | 2009-09-25 |
EP1861103A1 (en) | 2007-12-05 |
MX2007009916A (es) | 2007-09-25 |
CN101128203A (zh) | 2008-02-20 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
MM4A | Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s) |
Designated state(s): AM AZ BY KZ KG MD TJ TM RU |