DOP2009000087A - DERIVATIVES OF 2- [1-PHENYL-5-HYDROXI-4ALFA-METHYL-HEXAHYDROCOCLOPENTA [F] INDAZOL-5-IL] ETHYL PHENYLL AS GLUCOCORTICOID RECEIVER LIGANDS - Google Patents

DERIVATIVES OF 2- [1-PHENYL-5-HYDROXI-4ALFA-METHYL-HEXAHYDROCOCLOPENTA [F] INDAZOL-5-IL] ETHYL PHENYLL AS GLUCOCORTICOID RECEIVER LIGANDS

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Publication number
DOP2009000087A
DOP2009000087A DO2009000087A DO2009000087A DOP2009000087A DO P2009000087 A DOP2009000087 A DO P2009000087A DO 2009000087 A DO2009000087 A DO 2009000087A DO 2009000087 A DO2009000087 A DO 2009000087A DO P2009000087 A DOP2009000087 A DO P2009000087A
Authority
DO
Dominican Republic
Prior art keywords
phenyl
indazol
derivatives
methyl
ethyl
Prior art date
Application number
DO2009000087A
Other languages
Spanish (es)
Inventor
James J Perkins
Christopher J Bungard
Jesse J Manikowski
Robert Meissner
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Priority to DO2009000087A priority Critical patent/DOP2009000087A/en
Publication of DOP2009000087A publication Critical patent/DOP2009000087A/en

Links

Abstract

La presente invención se refiere a derivados de 2-[1-fenil-5-hidroxi-4alfa-metil-hexahidrociclopenta[f)indazol-5-il)etil fenilo como ligandos al receptor glucocorticoide utiles para el tratamiento de una variedad de enfermedades o afecciones autoinmunes e inflamatorias. Tambien se incluyen composiciones farmacéuticas y procedimientos de uso.The present invention relates to derivatives of 2- [1-phenyl-5-hydroxy-4alpha-methyl-hexahydrocyclopenta [f) indazol-5-yl) ethyl phenyl as glucocorticoid receptor ligands useful for the treatment of a variety of diseases or autoimmune and inflammatory conditions. Also included are pharmaceutical compositions and methods of use.

DO2009000087A 2009-04-22 2009-04-22 DERIVATIVES OF 2- [1-PHENYL-5-HYDROXI-4ALFA-METHYL-HEXAHYDROCOCLOPENTA [F] INDAZOL-5-IL] ETHYL PHENYLL AS GLUCOCORTICOID RECEIVER LIGANDS DOP2009000087A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
DO2009000087A DOP2009000087A (en) 2009-04-22 2009-04-22 DERIVATIVES OF 2- [1-PHENYL-5-HYDROXI-4ALFA-METHYL-HEXAHYDROCOCLOPENTA [F] INDAZOL-5-IL] ETHYL PHENYLL AS GLUCOCORTICOID RECEIVER LIGANDS

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DO2009000087A DOP2009000087A (en) 2009-04-22 2009-04-22 DERIVATIVES OF 2- [1-PHENYL-5-HYDROXI-4ALFA-METHYL-HEXAHYDROCOCLOPENTA [F] INDAZOL-5-IL] ETHYL PHENYLL AS GLUCOCORTICOID RECEIVER LIGANDS

Publications (1)

Publication Number Publication Date
DOP2009000087A true DOP2009000087A (en) 2009-06-30

Family

ID=44680872

Family Applications (1)

Application Number Title Priority Date Filing Date
DO2009000087A DOP2009000087A (en) 2009-04-22 2009-04-22 DERIVATIVES OF 2- [1-PHENYL-5-HYDROXI-4ALFA-METHYL-HEXAHYDROCOCLOPENTA [F] INDAZOL-5-IL] ETHYL PHENYLL AS GLUCOCORTICOID RECEIVER LIGANDS

Country Status (1)

Country Link
DO (1) DOP2009000087A (en)

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