DOP2005000235A - DERIVATIVES OF 3-PHENYL-PIRAZOL AS MODULATORS OF THE 5-HT2A SEROTONINE RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED TO THIS - Google Patents
DERIVATIVES OF 3-PHENYL-PIRAZOL AS MODULATORS OF THE 5-HT2A SEROTONINE RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED TO THISInfo
- Publication number
- DOP2005000235A DOP2005000235A DO2005000235A DO2005000235A DOP2005000235A DO P2005000235 A DOP2005000235 A DO P2005000235A DO 2005000235 A DO2005000235 A DO 2005000235A DO 2005000235 A DO2005000235 A DO 2005000235A DO P2005000235 A DOP2005000235 A DO P2005000235A
- Authority
- DO
- Dominican Republic
- Prior art keywords
- disorders
- psychosis
- treatment
- phenyl
- schizophrenia
- Prior art date
Links
Abstract
La presente invención está relacionada con ciertos derivados de 3-fenil-pirazol de fórmula (Ia) y sus composiciones farmacéuticas que modulan la actividad del receptor 5-HT,,, de la serotonina. Los compuestos y sus composiciones farmacéuticas están dirigidos hacia métodos d útiles en el tratamiento de la agregación plaquetaria, arteriopatía coronaria, infarto de miocardio, accidente isquémico transitorio, angina, accidente cerebrovascular, fibrilacion auricular, reducción del riesgo de formación de coagulos sanguineos, asma o sus sintomas, agitaci6n o un sintoma, trastomos de la coánducta, psicósis farmacógena, psicósis excitativa, síndrome de Gilles de la Tourette, trastomo maníaco, psicosis orgánica o sin especificación, trastorno psicótico, psicósis, esquizofrenia aguda, esquizofrenia crónica, esquizofrenia sin especificación y trastomos relacionados, y trastomos del sueño, trastomos relacionados con la diabetes, leucoencefalopatía multifocal progresiva y semejantes. La presente invención también está relacionada con los métodos para el tratamiento de trastomos originados por el receptor 5-HTz, de la serotonina en combinación con otros agentes fannacéuticos administrados juntos o por separado.The present invention is related to certain 3-phenyl-pyrazole derivatives of formula (Ia) and their pharmaceutical compositions that modulate the activity of the 5-HT receptor, serotonin. The compounds and their pharmaceutical compositions are directed towards useful methods in the treatment of platelet aggregation, coronary artery disease, myocardial infarction, transient ischemic accident, angina, stroke, atrial fibrillation, reduction of the risk of blood clot formation, asthma or its symptoms, agitation or a symptom, disorders of the coctact, pharmacogenic psychosis, excitatory psychosis, Gilles de la Tourette syndrome, manic disorder, organic or unspecified psychosis, psychotic disorder, psychosis, acute schizophrenia, chronic schizophrenia, unspecified schizophrenia and related disorders, and sleep disorders, diabetes-related disorders, progressive multifocal leukoencephalopathy and the like. The present invention is also related to methods for the treatment of disorders caused by the 5-HTz receptor, serotonin in combination with other fan agents administered together or separately.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DO2005000235A DOP2005000235A (en) | 2005-11-16 | 2005-11-16 | DERIVATIVES OF 3-PHENYL-PIRAZOL AS MODULATORS OF THE 5-HT2A SEROTONINE RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED TO THIS |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DO2005000235A DOP2005000235A (en) | 2005-11-16 | 2005-11-16 | DERIVATIVES OF 3-PHENYL-PIRAZOL AS MODULATORS OF THE 5-HT2A SEROTONINE RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED TO THIS |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DOP2005000235A true DOP2005000235A (en) | 2008-10-15 |
Family
ID=44676011
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DO2005000235A DOP2005000235A (en) | 2005-11-16 | 2005-11-16 | DERIVATIVES OF 3-PHENYL-PIRAZOL AS MODULATORS OF THE 5-HT2A SEROTONINE RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED TO THIS |
Country Status (1)
| Country | Link |
|---|---|
| DO (1) | DOP2005000235A (en) |
-
2005
- 2005-11-16 DO DO2005000235A patent/DOP2005000235A/en unknown
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