DOP2005000158A - SUBSTITUTED AMIDAS OF TIENOPIRROLCARBOXILICO ACID, AMIDAS OF THE PIRROLOTIAZOLCARBONOXILIO ACID, AND RELATED ANALOGS AS INHIBITORS OF CASEINA CINASA I - Google Patents

SUBSTITUTED AMIDAS OF TIENOPIRROLCARBOXILICO ACID, AMIDAS OF THE PIRROLOTIAZOLCARBONOXILIO ACID, AND RELATED ANALOGS AS INHIBITORS OF CASEINA CINASA I

Info

Publication number
DOP2005000158A
DOP2005000158A DO2005000158A DO2005000158A DOP2005000158A DO P2005000158 A DOP2005000158 A DO P2005000158A DO 2005000158 A DO2005000158 A DO 2005000158A DO 2005000158 A DO2005000158 A DO 2005000158A DO P2005000158 A DOP2005000158 A DO P2005000158A
Authority
DO
Dominican Republic
Prior art keywords
amidas
acid
formula
inhibitors
tienopirrolcarboxilico
Prior art date
Application number
DO2005000158A
Other languages
Spanish (es)
Inventor
David Marc Fink
Yulin Chiang
Nicola Dawn Collar
Original Assignee
Aventis Pharma Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma Inc filed Critical Aventis Pharma Inc
Priority to DO2005000158A priority Critical patent/DOP2005000158A/en
Publication of DOP2005000158A publication Critical patent/DOP2005000158A/en

Links

Landscapes

  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

La presentes invención describe y reivindica compuestos de fórmula (I) y fórmula como inhibidores de la caseína cinasa Is humana y m6todos para utilizar dichos compuestos para tratar enfermedades y trastornos del sistema nervioso central, incluyendo trastornos del ánimo y trastornos del sueho. También se describen y se reivindican composiciones farmacéuticas qua comprenden compuestos de fórmula (I) o fórmula (II) y un método de preparación de compuestos de fórmula (I) o fórmula (II).The present invention describes and claims compounds of formula (I) and formula as inhibitors of human casein kinase Is and methods for using said compounds to treat diseases and disorders of the central nervous system, including mood disorders and sleep disorders. Pharmaceutical compositions are also described and claimed which comprise compounds of formula (I) or formula (II) and a method of preparing compounds of formula (I) or formula (II).

DO2005000158A 2005-08-12 2005-08-12 SUBSTITUTED AMIDAS OF TIENOPIRROLCARBOXILICO ACID, AMIDAS OF THE PIRROLOTIAZOLCARBONOXILIO ACID, AND RELATED ANALOGS AS INHIBITORS OF CASEINA CINASA I DOP2005000158A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
DO2005000158A DOP2005000158A (en) 2005-08-12 2005-08-12 SUBSTITUTED AMIDAS OF TIENOPIRROLCARBOXILICO ACID, AMIDAS OF THE PIRROLOTIAZOLCARBONOXILIO ACID, AND RELATED ANALOGS AS INHIBITORS OF CASEINA CINASA I

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DO2005000158A DOP2005000158A (en) 2005-08-12 2005-08-12 SUBSTITUTED AMIDAS OF TIENOPIRROLCARBOXILICO ACID, AMIDAS OF THE PIRROLOTIAZOLCARBONOXILIO ACID, AND RELATED ANALOGS AS INHIBITORS OF CASEINA CINASA I

Publications (1)

Publication Number Publication Date
DOP2005000158A true DOP2005000158A (en) 2006-10-31

Family

ID=44340179

Family Applications (1)

Application Number Title Priority Date Filing Date
DO2005000158A DOP2005000158A (en) 2005-08-12 2005-08-12 SUBSTITUTED AMIDAS OF TIENOPIRROLCARBOXILICO ACID, AMIDAS OF THE PIRROLOTIAZOLCARBONOXILIO ACID, AND RELATED ANALOGS AS INHIBITORS OF CASEINA CINASA I

Country Status (1)

Country Link
DO (1) DOP2005000158A (en)

Similar Documents

Publication Publication Date Title
UY29077A1 (en) SUBSTITUTED AMIDES OF TIENOPIRROLCARBOXYL ACID, AMIDAS OF THE PYRROLOTIAZOLCARBOXYL ACID AND RELATED ANALOGS AS INHIBITORS OF CASEINE CINASE IE (EPSILON)
MX353461B (en) Processes for making compounds useful as inhibitors of atr kinase.
EA201190158A1 (en) Derivatives of benzofuranyl for use as glucose kinase inhibitors
NI200700296A (en) IMIDAZOQUINOLINAS AS INHIBITORS OF KINASE OF LIPIDO
BR112015028501B8 (en) BIPYRAZOLE DERIVATIVE COMPOUNDS, THEIR SALTS, COMPOSITION COMPRISING THE COMPOUND OR THE SALT, METHOD FOR IN VITRO INHIBITION OF A JAK1 ACTIVITY, AND PROCESS FOR PREPARING PHOSPHORIC ACID SALT
EA201992126A1 (en) JAK INHIBITORS CONTAINING 4-MEMBER HETEROCYCLIC AMIDE
EA201491592A1 (en) CONNECTIONS OF INDOLS AND INDAZOLS ACTIVATING AMPK
TN2009000128A1 (en) Dihydropyridine derivatives useful as protein kinase inhibitors
EA201500182A1 (en) 4-METHYL-2,3,5,9,9b-PENTAASACYCLOPENT [a] NAFTAIL
BR112013032720A2 (en) "azetidinyl phenyl, pyridyl or pyrazinyl carboxamide derivatives as jak inhibitors, composition and use of said derivatives"
EA201071057A1 (en) DERIVATIVES OF AZETIDINE AND CYCLUBUTAN AS JAK-KINAZ INHIBITORS
NO20083214L (en) Pyrimidinylarylurea derivatives which are converted to FGF inhibitors
EA201200373A1 (en) COMPOUNDS AND COMPOSITIONS AS PROTEINKINAZ INHIBITORS
BR112014004560A2 (en) compounds and compositions as c-kit kinase inhibitors
BR112015028452A2 (en) somastatin subtype 4 receptor agonists (sstr4)
MX2012013081A (en) Compounds useful as inhibitors of atr kinase.
EA201200952A1 (en) DERIVATIVES OF PYRAZINE AND THEIR APPLICATION FOR THE TREATMENT OF NEUROLOGICAL DISORDERS
CO6630193A2 (en) Inhibitors of selected tyrosine kinase protein activity
UY33889A (en) DIMALEATE OF 9- [4- (3-CHLORO-2-FLUORO-PHENYLAMINE) -7-METOXIQUINAZOLIN-6-ILOXI] -1,4-DIAZA-ESPIRO [5 .5] UNDECAN-5-ONA, ITS USE AS A MEDICINAL PRODUCT AND HIS PREPARATION
ES2333026T3 (en) DERIVED FROM CICLOHEXIL-1,4-DIAMINE SUBSTITUTED.
BR112021026531A2 (en) Compound, pharmaceutical composition, and method for preventing or treating a disease mediated by tyrosine kinase 2
CL2018000856A1 (en) Derivatives of pyrazolo cyclic ether [1,5-a] pyrimidin-3-carboxyamide.
PA8642901A1 (en) AMIDAS OF ACID 5 AND 6-AMINOALQUIL INDOL-2-CARBOXILICO 3-SUBSTITUTES AND RELATED ANALOGS AS INHIBITORS OF CASEINA CINASA I
EA201100422A1 (en) (PHENYL) AMIDA 7- (PIPERAZIN-1-ILMETHYL) -1H-INDOL-2-CARBIC ACID AND RELATED CONNECTIONS AS P38 MAR-KINASE INHIBITORS FOR THE TREATMENT OF DISEASES
DOP2005000158A (en) SUBSTITUTED AMIDAS OF TIENOPIRROLCARBOXILICO ACID, AMIDAS OF THE PIRROLOTIAZOLCARBONOXILIO ACID, AND RELATED ANALOGS AS INHIBITORS OF CASEINA CINASA I