DOP2005000158A -
SUBSTITUTED AMIDAS OF TIENOPIRROLCARBOXILICO ACID, AMIDAS OF THE PIRROLOTIAZOLCARBONOXILIO ACID, AND RELATED ANALOGS AS INHIBITORS OF CASEINA CINASA I
- Google Patents
SUBSTITUTED AMIDAS OF TIENOPIRROLCARBOXILICO ACID, AMIDAS OF THE PIRROLOTIAZOLCARBONOXILIO ACID, AND RELATED ANALOGS AS INHIBITORS OF CASEINA CINASA I
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Priority to DO2005000158ApriorityCriticalpatent/DOP2005000158A/en
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Pharmaceuticals Containing Other Organic And Inorganic Compounds
(AREA)
Abstract
La presentes invención describe y reivindica compuestos de fórmula (I) y fórmula como inhibidores de la caseína cinasa Is humana y m6todos para utilizar dichos compuestos para tratar enfermedades y trastornos del sistema nervioso central, incluyendo trastornos del ánimo y trastornos del sueho. También se describen y se reivindican composiciones farmacéuticas qua comprenden compuestos de fórmula (I) o fórmula (II) y un método de preparación de compuestos de fórmula (I) o fórmula (II).The present invention describes and claims compounds of formula (I) and formula as inhibitors of human casein kinase Is and methods for using said compounds to treat diseases and disorders of the central nervous system, including mood disorders and sleep disorders. Pharmaceutical compositions are also described and claimed which comprise compounds of formula (I) or formula (II) and a method of preparing compounds of formula (I) or formula (II).
DO2005000158A2005-08-122005-08-12
SUBSTITUTED AMIDAS OF TIENOPIRROLCARBOXILICO ACID, AMIDAS OF THE PIRROLOTIAZOLCARBONOXILIO ACID, AND RELATED ANALOGS AS INHIBITORS OF CASEINA CINASA I
DOP2005000158A
(en)
SUBSTITUTED AMIDES OF TIENOPIRROLCARBOXYL ACID, AMIDAS OF THE PYRROLOTIAZOLCARBOXYL ACID AND RELATED ANALOGS AS INHIBITORS OF CASEINE CINASE IE (EPSILON)
BIPYRAZOLE DERIVATIVE COMPOUNDS, THEIR SALTS, COMPOSITION COMPRISING THE COMPOUND OR THE SALT, METHOD FOR IN VITRO INHIBITION OF A JAK1 ACTIVITY, AND PROCESS FOR PREPARING PHOSPHORIC ACID SALT
DIMALEATE OF 9- [4- (3-CHLORO-2-FLUORO-PHENYLAMINE) -7-METOXIQUINAZOLIN-6-ILOXI] -1,4-DIAZA-ESPIRO [5 .5] UNDECAN-5-ONA, ITS USE AS A MEDICINAL PRODUCT AND HIS PREPARATION