DOP2004000972A - 6- (2,2,2-TRIFLUOROETHYLAMINE) -7-CHLORINE-2,3,4,5-TETRAHYDR 1H-BENZO [D] AZEPIN AS A 5-HT2C RECEPTOR AGONIST - Google Patents

6- (2,2,2-TRIFLUOROETHYLAMINE) -7-CHLORINE-2,3,4,5-TETRAHYDR 1H-BENZO [D] AZEPIN AS A 5-HT2C RECEPTOR AGONIST

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Publication number
DOP2004000972A
DOP2004000972A DO2004000972A DO2004000972A DOP2004000972A DO P2004000972 A DOP2004000972 A DO P2004000972A DO 2004000972 A DO2004000972 A DO 2004000972A DO 2004000972 A DO2004000972 A DO 2004000972A DO P2004000972 A DOP2004000972 A DO P2004000972A
Authority
DO
Dominican Republic
Prior art keywords
benzo
tetrahydr
trifluoroethylamine
azepin
chlorine
Prior art date
Application number
DO2004000972A
Other languages
Spanish (es)
Inventor
Christopher Stanley Galka
Michael John Rodriguez
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Priority to DO2004000972A priority Critical patent/DOP2004000972A/en
Publication of DOP2004000972A publication Critical patent/DOP2004000972A/en

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Abstract

La presente invencion proporciona un 7-cloro-6-(2,2,2-trifluoretilamino)2,3,4,5-tetrahidro-1H-benzo[d]azepina de formula I: o una sal del mismo farmacéuticamente aceptable, y su use como agonista selectivo de 5-HT2c para el tratamiento de trastornos asociados con los receptores 5-HT2c, incluyendo obesidad, trastorno obsesivo/compulsivo, ansiedad y depresion.The present invention provides a 7-chloro-6- (2,2,2-trifluoroethylamino) 2,3,4,5-tetrahydro-1H-benzo [d] azepine of formula I: or a pharmaceutically acceptable salt thereof, and its use as a selective 5-HT2c agonist for the treatment of disorders associated with 5-HT2c receptors, including obesity, obsessive / compulsive disorder, anxiety and depression.

DO2004000972A 2004-08-09 2004-08-09 6- (2,2,2-TRIFLUOROETHYLAMINE) -7-CHLORINE-2,3,4,5-TETRAHYDR 1H-BENZO [D] AZEPIN AS A 5-HT2C RECEPTOR AGONIST DOP2004000972A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
DO2004000972A DOP2004000972A (en) 2004-08-09 2004-08-09 6- (2,2,2-TRIFLUOROETHYLAMINE) -7-CHLORINE-2,3,4,5-TETRAHYDR 1H-BENZO [D] AZEPIN AS A 5-HT2C RECEPTOR AGONIST

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DO2004000972A DOP2004000972A (en) 2004-08-09 2004-08-09 6- (2,2,2-TRIFLUOROETHYLAMINE) -7-CHLORINE-2,3,4,5-TETRAHYDR 1H-BENZO [D] AZEPIN AS A 5-HT2C RECEPTOR AGONIST

Publications (1)

Publication Number Publication Date
DOP2004000972A true DOP2004000972A (en) 2005-02-28

Family

ID=44261392

Family Applications (1)

Application Number Title Priority Date Filing Date
DO2004000972A DOP2004000972A (en) 2004-08-09 2004-08-09 6- (2,2,2-TRIFLUOROETHYLAMINE) -7-CHLORINE-2,3,4,5-TETRAHYDR 1H-BENZO [D] AZEPIN AS A 5-HT2C RECEPTOR AGONIST

Country Status (1)

Country Link
DO (1) DOP2004000972A (en)

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