DOP2004000966A - 6 MEMBER HETEROARILE COMPOUNDS FOR THE TREATMENT OF NEURODEGENERATIVE DISORDERS - Google Patents
6 MEMBER HETEROARILE COMPOUNDS FOR THE TREATMENT OF NEURODEGENERATIVE DISORDERSInfo
- Publication number
- DOP2004000966A DOP2004000966A DO2004000966A DO2004000966A DOP2004000966A DO P2004000966 A DOP2004000966 A DO P2004000966A DO 2004000966 A DO2004000966 A DO 2004000966A DO 2004000966 A DO2004000966 A DO 2004000966A DO P2004000966 A DOP2004000966 A DO P2004000966A
- Authority
- DO
- Dominican Republic
- Prior art keywords
- compounds
- heteroarile
- treatment
- neurodegenerative disorders
- formula
- Prior art date
Links
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- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
Abstract
La presente invencion se refiere a compuestos de la Formula en donde R1, R1a, R1b, R2, R3, R4, R5, R6, R7, R8, R9, R10, R11, R12, X, Y, W, U, Z, m y n son como se los define. Compuestos de la Formula I presentan actividad inhibidora de la produccion de peptido Ap. Esta invencion se refiere ademàs a composiciones farmaceuticas y metodos para tratar enfermedades, por ejemplo, enfermedades neurodegenerativas, i.e. enfermedad de Alzheimer, en un mamifero, que comprenden compuestos de la Formula I.The present invention relates to compounds of the Formula wherein R1, R1a, R1b, R2, R3, R4, R5, R6, R7, R8, R9, R10, R11, R12, X, Y, W, U, Z, Myn are as defined. Compounds of Formula I exhibit inhibitory activity of peptide production Ap. This invention also relates to pharmaceutical compositions and methods for treating diseases, for example, neurodegenerative diseases, i.e. Alzheimer's disease, in a mammal, comprising compounds of Formula I.
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DO2004000966A DOP2004000966A (en) | 2004-08-02 | 2004-08-02 | 6 MEMBER HETEROARILE COMPOUNDS FOR THE TREATMENT OF NEURODEGENERATIVE DISORDERS |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DO2004000966A DOP2004000966A (en) | 2004-08-02 | 2004-08-02 | 6 MEMBER HETEROARILE COMPOUNDS FOR THE TREATMENT OF NEURODEGENERATIVE DISORDERS |
Publications (1)
Publication Number | Publication Date |
---|---|
DOP2004000966A true DOP2004000966A (en) | 2005-02-15 |
Family
ID=44261387
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DO2004000966A DOP2004000966A (en) | 2004-08-02 | 2004-08-02 | 6 MEMBER HETEROARILE COMPOUNDS FOR THE TREATMENT OF NEURODEGENERATIVE DISORDERS |
Country Status (1)
Country | Link |
---|---|
DO (1) | DOP2004000966A (en) |
-
2004
- 2004-08-02 DO DO2004000966A patent/DOP2004000966A/en unknown
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