DOP2003000634A - TRIARIL-OXIARIL-ESPIRO-PYRIMIDINE-2,4,6-TRIONA METALOPROTEINASE INHIBITORS - Google Patents

TRIARIL-OXIARIL-ESPIRO-PYRIMIDINE-2,4,6-TRIONA METALOPROTEINASE INHIBITORS

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Publication number
DOP2003000634A
DOP2003000634A DO2003000634A DO2003000634A DOP2003000634A DO P2003000634 A DOP2003000634 A DO P2003000634A DO 2003000634 A DO2003000634 A DO 2003000634A DO 2003000634 A DO2003000634 A DO 2003000634A DO P2003000634 A DOP2003000634 A DO P2003000634A
Authority
DO
Dominican Republic
Prior art keywords
pyrimidine
triaril
oxiaril
triona
espiro
Prior art date
Application number
DO2003000634A
Other languages
Spanish (es)
Inventor
Kevin Daniel Freeman-Cook
Mark Carl Noe
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Priority to DO2003000634A priority Critical patent/DOP2003000634A/en
Publication of DOP2003000634A publication Critical patent/DOP2003000634A/en

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

La presente invención se refiere a inhibidores de metaloproteinasa de triaril-oxiaril-espiro-pirimidina-2, 4, 6-triona de formula en la que el anillo x es un anillo heterocíclido de 5-7 miembros, y donde a, y, b, g y w son tal y como se han definido en la memoria descriptiva; y a composiciones farmacéuticas y procedimientos de tratamiento de la inflamación, cánceres y otros trastornos.The present invention relates to triaryl-oxyaryl-spiro-pyrimidine-2, 4, 6-trione metalloproteinase inhibitors of the formula in which the x-ring is a 5-7 membered heterocyclic ring, and wherein a, y, b , gyw are as defined in the specification; and to pharmaceutical compositions and methods of treating inflammation, cancers and other disorders.

DO2003000634A 2003-04-24 2003-04-24 TRIARIL-OXIARIL-ESPIRO-PYRIMIDINE-2,4,6-TRIONA METALOPROTEINASE INHIBITORS DOP2003000634A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
DO2003000634A DOP2003000634A (en) 2003-04-24 2003-04-24 TRIARIL-OXIARIL-ESPIRO-PYRIMIDINE-2,4,6-TRIONA METALOPROTEINASE INHIBITORS

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DO2003000634A DOP2003000634A (en) 2003-04-24 2003-04-24 TRIARIL-OXIARIL-ESPIRO-PYRIMIDINE-2,4,6-TRIONA METALOPROTEINASE INHIBITORS

Publications (1)

Publication Number Publication Date
DOP2003000634A true DOP2003000634A (en) 2003-10-31

Family

ID=44261177

Family Applications (1)

Application Number Title Priority Date Filing Date
DO2003000634A DOP2003000634A (en) 2003-04-24 2003-04-24 TRIARIL-OXIARIL-ESPIRO-PYRIMIDINE-2,4,6-TRIONA METALOPROTEINASE INHIBITORS

Country Status (1)

Country Link
DO (1) DOP2003000634A (en)

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