DOP2001000184A - ACAT CARBOXIALQUILETER-INHIBITOR COMBINATIONS - Google Patents
ACAT CARBOXIALQUILETER-INHIBITOR COMBINATIONSInfo
- Publication number
- DOP2001000184A DOP2001000184A DO2001000184A DO2001000184A DOP2001000184A DO P2001000184 A DOP2001000184 A DO P2001000184A DO 2001000184 A DO2001000184 A DO 2001000184A DO 2001000184 A DO2001000184 A DO 2001000184A DO P2001000184 A DOP2001000184 A DO P2001000184A
- Authority
- DO
- Dominican Republic
- Prior art keywords
- acat
- carboxialquileter
- formula
- inhibitor combinations
- dyslipidemia
- Prior art date
Links
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
La invención es una composicion farmaceutica que comprende un carboxialquileter que reduce trigliceridos y LDL y eleva el HDL y un inhibidor de ACAT que mejora la dislipidemia en mamiferos, dicha composicion es util para tratar la dislipidemia y sindromes isquemicos y para prevenir o retardar el comienzo de ataques cardiacos. Los carboxialquieteres tienen la formula en donde Y1 e Y2 incluyen COOH, R1, R2, R3 y R4 pueden ser alquilo, y n y m son numeros enteros de 2 a 9; y los inhibidores de ACAT tienen la formula en donde R es hidrogeno, X es 0, R1 y R2 son fenilo sustituido, e Y es alquileno.The invention is a pharmaceutical composition comprising a carboxyalkylether that reduces triglycerides and LDL and elevates HDL and an ACAT inhibitor that improves dyslipidemia in mammals, said composition is useful for treating dyslipidemia and ischemic syndromes and for preventing or delaying the onset of heart attacks. The carboxyalkieters have the formula wherein Y1 and Y2 include COOH, R1, R2, R3 and R4 can be alkyl, and n and m are whole numbers from 2 to 9; and ACAT inhibitors have the formula wherein R is hydrogen, X is 0, R1 and R2 are substituted phenyl, and Y is alkylene.
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DO2001000184A DOP2001000184A (en) | 2001-06-05 | 2001-06-05 | ACAT CARBOXIALQUILETER-INHIBITOR COMBINATIONS |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DO2001000184A DOP2001000184A (en) | 2001-06-05 | 2001-06-05 | ACAT CARBOXIALQUILETER-INHIBITOR COMBINATIONS |
Publications (1)
Publication Number | Publication Date |
---|---|
DOP2001000184A true DOP2001000184A (en) | 2002-06-15 |
Family
ID=44261007
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DO2001000184A DOP2001000184A (en) | 2001-06-05 | 2001-06-05 | ACAT CARBOXIALQUILETER-INHIBITOR COMBINATIONS |
Country Status (1)
Country | Link |
---|---|
DO (1) | DOP2001000184A (en) |
-
2001
- 2001-06-05 DO DO2001000184A patent/DOP2001000184A/en unknown
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