DK630686A - 2'-SUBSTITUTED 4-DEOXYTIAZOLO (5,4-C) RIFAMYCIN SV DERIVATIVES AND MEDICINAL CONTAINING SUCH DERIVATIVES - Google Patents

2'-SUBSTITUTED 4-DEOXYTIAZOLO (5,4-C) RIFAMYCIN SV DERIVATIVES AND MEDICINAL CONTAINING SUCH DERIVATIVES

Info

Publication number
DK630686A
DK630686A DK630686A DK630686A DK630686A DK 630686 A DK630686 A DK 630686A DK 630686 A DK630686 A DK 630686A DK 630686 A DK630686 A DK 630686A DK 630686 A DK630686 A DK 630686A
Authority
DK
Denmark
Prior art keywords
derivatives
rifamycin
substituted
deoxytiazolo
medicinal containing
Prior art date
Application number
DK630686A
Other languages
Danish (da)
Other versions
DK630686D0 (en
DK170100B1 (en
Inventor
Bruno Cavalleri
Marco Turconi
Giovanni Tamborini
Original Assignee
Lepetit Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lepetit Spa filed Critical Lepetit Spa
Publication of DK630686D0 publication Critical patent/DK630686D0/en
Publication of DK630686A publication Critical patent/DK630686A/en
Application granted granted Critical
Publication of DK170100B1 publication Critical patent/DK170100B1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/10—Spiro-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains three hetero rings
    • C07D513/18—Bridged systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Thiazole And Isothizaole Compounds (AREA)

Abstract

The present invention concerns new 2'-substituted-4-deoxy-thiazolo[5,4-c]rifamycin SV derivatives having antibacterial activity.These compounds are obtained by chemical modification of thiazolo[5,4-c]rifamycin SV.
DK630686A 1985-12-30 1986-12-29 2'-Substituted 4-deoxytiazolo (5,4-c) rifamycin SV derivatives, process for their preparation, such a compound for use as a drug, use of the compound for the preparation of an antibacterial drug, and pharmaceutical composition containing the compound DK170100B1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB8531887 1985-12-30
GB858531887A GB8531887D0 (en) 1985-12-30 1985-12-30 Rifamycin sv derivatives

Publications (3)

Publication Number Publication Date
DK630686D0 DK630686D0 (en) 1986-12-29
DK630686A true DK630686A (en) 1987-07-01
DK170100B1 DK170100B1 (en) 1995-05-22

Family

ID=10590333

Family Applications (1)

Application Number Title Priority Date Filing Date
DK630686A DK170100B1 (en) 1985-12-30 1986-12-29 2'-Substituted 4-deoxytiazolo (5,4-c) rifamycin SV derivatives, process for their preparation, such a compound for use as a drug, use of the compound for the preparation of an antibacterial drug, and pharmaceutical composition containing the compound

Country Status (17)

Country Link
US (1) US4880789A (en)
EP (1) EP0228606B1 (en)
JP (1) JPH07108909B2 (en)
KR (1) KR940009795B1 (en)
AT (1) ATE60772T1 (en)
CA (1) CA1271472A (en)
DE (1) DE3677485D1 (en)
DK (1) DK170100B1 (en)
ES (1) ES2031815T3 (en)
GB (1) GB8531887D0 (en)
GR (1) GR3001543T3 (en)
HK (1) HK97391A (en)
HU (1) HU196812B (en)
IE (1) IE59505B1 (en)
IL (1) IL80447A (en)
SG (1) SG67091G (en)
ZA (1) ZA869453B (en)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL100642A (en) * 1991-01-28 1995-11-27 Lepetit Spa Process for preparing 2' - (diethylamino) rifamycin p (p/dea) and a novel intermediate therefor
US6375658B1 (en) 2000-04-28 2002-04-23 Smith & Nephew, Inc. Cartilage grafting
US7265107B2 (en) 2004-03-10 2007-09-04 Cumbre Pharmaceuticals Inc. Rifamycin C-11 oxime cyclo derivatives effective against drug-resistant microbes
US7256187B2 (en) 2004-03-10 2007-08-14 Cumbre Pharmaceuticals Inc. Rifamycin C-11 oxime derivatives effective against drug-resistant microbes
US20100125146A1 (en) * 2008-11-19 2010-05-20 Johnson Matthey Public Limited Company Method for making pharmaceutical compounds

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1470426A (en) * 1974-08-30 1977-04-14 Lepetit Spa Rifamycins
GB1523198A (en) * 1976-05-28 1978-08-31 Lepetit Spa Thiazolo-rifamycin derivatives
GB1523199A (en) * 1976-05-28 1978-08-31 Lepetit Spa Rifamycin sv derivatives
CH629212A5 (en) * 1976-10-18 1982-04-15 Erba Farmitalia PROCEDURE FOR THE PREPARATION OF RIFAMICIN COMPOUNDS.
GB1594134A (en) * 1977-11-25 1981-07-30 Holco Investment Inc Rifamycins
IT1111173B (en) * 1978-04-27 1986-01-13 Lepetit Spa RIFAMICINICI DERIVATIVES
DD204925A5 (en) * 1980-09-25 1983-12-14 Ciba Geigy Ag PROCESS FOR PREPARING A 4-AMINOIMIDAZOLO (4,5-C) RIFAMYCIN SV OR S

Also Published As

Publication number Publication date
DK630686D0 (en) 1986-12-29
EP0228606A2 (en) 1987-07-15
JPH07108909B2 (en) 1995-11-22
EP0228606B1 (en) 1991-02-06
GR3001543T3 (en) 1992-11-23
ES2031815T3 (en) 1993-01-01
EP0228606A3 (en) 1989-01-11
GB8531887D0 (en) 1986-02-05
IL80447A0 (en) 1987-01-30
ZA869453B (en) 1987-09-30
KR870006057A (en) 1987-07-09
HU196812B (en) 1989-01-30
JPS62158292A (en) 1987-07-14
SG67091G (en) 1991-09-13
DE3677485D1 (en) 1991-03-14
US4880789A (en) 1989-11-14
IL80447A (en) 1990-09-17
HK97391A (en) 1991-12-13
DK170100B1 (en) 1995-05-22
IE59505B1 (en) 1994-03-09
CA1271472A (en) 1990-07-10
HUT45072A (en) 1988-05-30
KR940009795B1 (en) 1994-10-17
IE863277L (en) 1987-06-30
ATE60772T1 (en) 1991-02-15

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Legal Events

Date Code Title Description
B1 Patent granted (law 1993)
PBP Patent lapsed