DK621688A - ETHYLERED AVERMECTINES AND PREPARATIONS CONTAINING THESE FOR THE TREATMENT AND PREVENTION OF HUMAN AND ANIMAL PARASITE INFECTIONS - Google Patents

ETHYLERED AVERMECTINES AND PREPARATIONS CONTAINING THESE FOR THE TREATMENT AND PREVENTION OF HUMAN AND ANIMAL PARASITE INFECTIONS

Info

Publication number
DK621688A
DK621688A DK621688A DK621688A DK621688A DK 621688 A DK621688 A DK 621688A DK 621688 A DK621688 A DK 621688A DK 621688 A DK621688 A DK 621688A DK 621688 A DK621688 A DK 621688A
Authority
DK
Denmark
Prior art keywords
ethylered
avermectines
prevention
human
treatment
Prior art date
Application number
DK621688A
Other languages
Danish (da)
Other versions
DK621688D0 (en
Inventor
Steven Joseph Hawrylik
Shih-Jen Edward Lee
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of DK621688D0 publication Critical patent/DK621688D0/en
Publication of DK621688A publication Critical patent/DK621688A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/10Anthelmintics
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10STECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10S435/00Chemistry: molecular biology and microbiology
    • Y10S435/8215Microorganisms
    • Y10S435/822Microorganisms using bacteria or actinomycetales
    • Y10S435/886Streptomyces

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Molecular Biology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Medicinal Chemistry (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Fodder In General (AREA)

Abstract

Avermectins wherein one or both of the 3 min - and 3 sec - positions of the cleandrose disaccharide moiety is substituted by an ethoxy rather than a methoxy group, process for their preparation; and their use as antiparasitic agents.
DK621688A 1987-11-09 1988-11-08 ETHYLERED AVERMECTINES AND PREPARATIONS CONTAINING THESE FOR THE TREATMENT AND PREVENTION OF HUMAN AND ANIMAL PARASITE INFECTIONS DK621688A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US11868487A 1987-11-09 1987-11-09

Publications (2)

Publication Number Publication Date
DK621688D0 DK621688D0 (en) 1988-11-08
DK621688A true DK621688A (en) 1989-07-06

Family

ID=22380121

Family Applications (1)

Application Number Title Priority Date Filing Date
DK621688A DK621688A (en) 1987-11-09 1988-11-08 ETHYLERED AVERMECTINES AND PREPARATIONS CONTAINING THESE FOR THE TREATMENT AND PREVENTION OF HUMAN AND ANIMAL PARASITE INFECTIONS

Country Status (10)

Country Link
US (1) US5387509A (en)
EP (1) EP0316124B1 (en)
JP (1) JPH0695947B2 (en)
AT (1) ATE87926T1 (en)
CA (1) CA1340771C (en)
DE (1) DE3880088T2 (en)
DK (1) DK621688A (en)
ES (1) ES2045146T3 (en)
IE (1) IE62446B1 (en)
PT (1) PT88952B (en)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8726730D0 (en) * 1987-11-14 1987-12-16 Pfizer Ltd Antiparasitic agents
ES2052173T3 (en) * 1989-04-11 1994-07-01 Pfizer INJECTABLE COMPOSITIONS CONTAINING 25-CYCLOHEXIL-AVERMECTIN B1.
US6426333B1 (en) 1996-09-19 2002-07-30 Merial Spot-on formulations for combating parasites
US6998131B2 (en) * 1996-09-19 2006-02-14 Merial Limited Spot-on formulations for combating parasites

Family Cites Families (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE434277B (en) * 1976-04-19 1984-07-16 Merck & Co Inc SET TO MAKE NEW ANTIHELMINTICALLY EFFECTIVE ASSOCIATIONS BY CULTIVATING STREPTOMYCS AVERMITILIS
US4199569A (en) * 1977-10-03 1980-04-22 Merck & Co., Inc. Selective hydrogenation products of C-076 compounds and derivatives thereof
PH15982A (en) * 1977-10-03 1983-05-18 Merck & Co Inc Selective hydrogenation producta of c-076 compounds and derivatives thereof
IL56149A (en) * 1977-12-19 1989-09-28 Merck & Co Inc 13-halo and 13-deoxy derivatives of c-076 compounds,their preparation and method for the treatment of parasitic infections in animals therewith
US4203976A (en) * 1978-08-02 1980-05-20 Merck & Co., Inc. Sugar derivatives of C-076 compounds
US4200581A (en) * 1978-08-04 1980-04-29 Merck & Co., Inc. Alkyl derivatives of C-076 compounds
US4429042A (en) * 1978-09-08 1984-01-31 Merck & Co., Inc. Strain of Streptomyces for producing antiparasitic compounds
US4328335A (en) * 1979-08-13 1982-05-04 Merck & Co., Inc. Process for the interconversion of C-076 compounds
US4285963A (en) * 1980-08-07 1981-08-25 Merck & Co., Inc. Novel derivatives of C-076 compounds
US4378353A (en) * 1981-02-17 1983-03-29 Merck & Co., Inc. Novel C-076 compounds
US4333925A (en) * 1981-05-11 1982-06-08 Merck & Co., Inc. Derivatives of C-076 compounds
US4423209A (en) * 1982-02-26 1983-12-27 Merck & Co., Inc. Processes for the interconversion of avermectin compounds
NZ213463A (en) * 1984-09-14 1993-04-28 American Cyanamid Co Antibiotic compound and compositions
HUT39739A (en) * 1984-12-04 1986-10-29 Ciba Geigy Ag Process for production of derivatives of 13,3-milbemycin and medical preparatives containing thereof
AU596586B2 (en) * 1985-04-30 1990-05-10 American Cyanamid Company Chemical derivatives of antibiotics S541
ES8800986A1 (en) * 1985-07-27 1987-12-01 Pfizer Antiparasitic avermectin and milbemycin derivatives and process for their preparation.
JPH085893B2 (en) * 1985-09-13 1996-01-24 アメリカン・サイアナミツド・カンパニー Macrolide antibiotic and method for producing the same
GB8606120D0 (en) * 1986-03-12 1986-04-16 Glaxo Group Ltd Process
US4831016A (en) * 1986-10-31 1989-05-16 Merck & Co., Inc. Reduced avermectin derivatives

Also Published As

Publication number Publication date
DE3880088D1 (en) 1993-05-13
DE3880088T2 (en) 1993-07-22
JPH0695947B2 (en) 1994-11-30
JPH01157986A (en) 1989-06-21
EP0316124A3 (en) 1989-10-18
IE62446B1 (en) 1995-02-08
ES2045146T3 (en) 1994-01-16
EP0316124B1 (en) 1993-04-07
ATE87926T1 (en) 1993-04-15
DK621688D0 (en) 1988-11-08
PT88952A (en) 1988-12-01
CA1340771C (en) 1999-09-28
PT88952B (en) 1993-02-26
EP0316124A2 (en) 1989-05-17
US5387509A (en) 1995-02-07
IE883358L (en) 1989-05-09

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Legal Events

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AHS Application shelved for other reasons than non-payment