DK323278A - 1h-pyrimido (4,5-c)-1,2-diazepiner og deres fremstilling omdannelse og anvendelse - Google Patents

1h-pyrimido (4,5-c)-1,2-diazepiner og deres fremstilling omdannelse og anvendelse

Info

Publication number
DK323278A
DK323278A DK323278A DK323278A DK323278A DK 323278 A DK323278 A DK 323278A DK 323278 A DK323278 A DK 323278A DK 323278 A DK323278 A DK 323278A DK 323278 A DK323278 A DK 323278A
Authority
DK
Denmark
Prior art keywords
diazepines
pyrimido
transformation
manufacturing
manufacturing transformation
Prior art date
Application number
DK323278A
Other languages
English (en)
Inventor
R W Morrison
W R Mollory
V L Styles
Original Assignee
Wellcome Found
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wellcome Found filed Critical Wellcome Found
Publication of DK323278A publication Critical patent/DK323278A/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48—Two nitrogen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
DK323278A 1977-07-20 1978-07-19 1h-pyrimido (4,5-c)-1,2-diazepiner og deres fremstilling omdannelse og anvendelse DK323278A (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB3038077 1977-07-20

Publications (1)

Publication Number Publication Date
DK323278A true DK323278A (da) 1979-01-21

Family

ID=10306770

Family Applications (1)

Application Number Title Priority Date Filing Date
DK323278A DK323278A (da) 1977-07-20 1978-07-19 1h-pyrimido (4,5-c)-1,2-diazepiner og deres fremstilling omdannelse og anvendelse

Country Status (5)

Country Link
US (4) US4288365A (da)
EP (1) EP0000541B1 (da)
JP (1) JPS5422393A (da)
DE (1) DE2861598D1 (da)
DK (1) DK323278A (da)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2862102D1 (en) * 1977-07-08 1982-11-18 Wellcome Found Pyrimido (4,5-c) pyridazines, their use in pharmaceutical preparations, and process for their preparation
EP0075267B1 (en) * 1981-09-19 1986-01-15 Sumitomo Chemical Company, Limited 4-(2-fluoro-4-halo-5-substituted phenyl)urazols, and their production and use
WO1993020075A1 (en) * 1992-04-01 1993-10-14 The University Of Sydney 8-substituted-n5-deazapterins as antifolates
WO2008117047A1 (en) * 2007-03-27 2008-10-02 Astrazeneca Ab Pyrazolo[3, 4-d]pyrimidine derivatives as antibacterial compounds

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB447094A (en) 1934-06-22 1936-05-12 Anonima Eternit Pietra Artific Improvements in lead-packed couplings for pipe lines
GB774095A (en) 1953-01-02 1957-05-08 Wellcome Found Improvements in or relating to pyrimidine compounds
GB798646A (en) * 1955-08-10 1958-07-23 Wellcome Found Improvements in and relating to derivatives of pyrimidine and the manufacture thereof
GB1129084A (en) 1965-02-18 1968-10-02 Wellcome Found Novel pyrido[2,3-d]pyrimidines
US3947442A (en) * 1969-11-20 1976-03-30 The Sherwin-Williams Company Method for producing heterocyclic acid anhydrides and pyrimidinediones
DE2038035A1 (de) * 1970-07-31 1972-02-03 Boehringer Mannheim GmbH, 6800 Mannheim-Waldhof 2-Amino-pyrido eckige Klammer auf 2,3-d eckige Klammer zu pyrimidin-4(3H)on-Derivate
BE790014A (fr) 1971-10-12 1973-04-12 Woods Hamish C S Pyrido (2,3-d) pyrimidines a usage therapeutique
US4113859A (en) * 1972-10-12 1978-09-12 Burroughs Wellcome Co. Certain pyrido-pyrimidines for treating mammalian and avian infections
DE2862102D1 (en) * 1977-07-08 1982-11-18 Wellcome Found Pyrimido (4,5-c) pyridazines, their use in pharmaceutical preparations, and process for their preparation

Also Published As

Publication number Publication date
US4237289A (en) 1980-12-02
US4288365A (en) 1981-09-08
EP0000541A2 (en) 1979-02-07
DE2861598D1 (en) 1982-03-11
US4315932A (en) 1982-02-16
JPS5422393A (en) 1979-02-20
US4235905A (en) 1980-11-25
EP0000541A3 (en) 1979-07-11
EP0000541B1 (en) 1982-02-03

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Legal Events

Date Code Title Description
AHS Application shelved for other reasons than non-payment