DK157875C - Vandoploeselige rifampicinderivater, fremgangsmaade til fremstilling deraf og farmaceutisk praeparat indeholdende saadanne forbindelser - Google Patents
Vandoploeselige rifampicinderivater, fremgangsmaade til fremstilling deraf og farmaceutisk praeparat indeholdende saadanne forbindelserInfo
- Publication number
- DK157875C DK157875C DK311484A DK311484A DK157875C DK 157875 C DK157875 C DK 157875C DK 311484 A DK311484 A DK 311484A DK 311484 A DK311484 A DK 311484A DK 157875 C DK157875 C DK 157875C
- Authority
- DK
- Denmark
- Prior art keywords
- derivatives
- preparing
- rifampicine
- procedures
- soluble
- Prior art date
Links
- JQXXHWHPUNPDRT-WLSIYKJHSA-N rifampicin Chemical class O([C@](C1=O)(C)O/C=C/[C@@H]([C@H]([C@@H](OC(C)=O)[C@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@@H](C)\C=C\C=C(C)/C(=O)NC=2C(O)=C3C([O-])=C4C)C)OC)C4=C1C3=C(O)C=2\C=N\N1CC[NH+](C)CC1 JQXXHWHPUNPDRT-WLSIYKJHSA-N 0.000 title abstract 3
- 150000001875 compounds Chemical class 0.000 title 1
- 238000000034 method Methods 0.000 title 1
- 239000000825 pharmaceutical preparation Substances 0.000 title 1
- 125000005041 acyloxyalkyl group Chemical group 0.000 abstract 1
- 230000000844 anti-bacterial effect Effects 0.000 abstract 1
- 239000007864 aqueous solution Substances 0.000 abstract 1
- 230000003115 biocidal effect Effects 0.000 abstract 1
- 125000001589 carboacyl group Chemical group 0.000 abstract 1
- 238000007911 parenteral administration Methods 0.000 abstract 1
- 229960001225 rifampicin Drugs 0.000 abstract 1
- 239000000126 substance Substances 0.000 abstract 1
- XLYOFNOQVPJJNP-UHFFFAOYSA-N water Substances O XLYOFNOQVPJJNP-UHFFFAOYSA-N 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/08—Bridged systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Oncology (AREA)
- Pharmacology & Pharmacy (AREA)
- Communicable Diseases (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Cephalosporin Compounds (AREA)
- Steroid Compounds (AREA)
- Saccharide Compounds (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB838318072A GB8318072D0 (en) | 1983-07-04 | 1983-07-04 | Water-soluble rifampicin derivatives |
| GB8318072 | 1983-07-04 |
Publications (4)
| Publication Number | Publication Date |
|---|---|
| DK311484D0 DK311484D0 (da) | 1984-06-26 |
| DK311484A DK311484A (da) | 1985-01-05 |
| DK157875B DK157875B (da) | 1990-02-26 |
| DK157875C true DK157875C (da) | 1990-08-20 |
Family
ID=10545208
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK311484A DK157875C (da) | 1983-07-04 | 1984-06-26 | Vandoploeselige rifampicinderivater, fremgangsmaade til fremstilling deraf og farmaceutisk praeparat indeholdende saadanne forbindelser |
Country Status (17)
| Country | Link |
|---|---|
| US (1) | US4585589A (OSRAM) |
| EP (1) | EP0133887B1 (OSRAM) |
| JP (1) | JPS6036490A (OSRAM) |
| KR (1) | KR910005847B1 (OSRAM) |
| AT (1) | ATE29136T1 (OSRAM) |
| AU (1) | AU558707B2 (OSRAM) |
| CA (1) | CA1212670A (OSRAM) |
| DE (1) | DE3465597D1 (OSRAM) |
| DK (1) | DK157875C (OSRAM) |
| ES (1) | ES533957A0 (OSRAM) |
| GB (1) | GB8318072D0 (OSRAM) |
| HU (1) | HU190576B (OSRAM) |
| IE (1) | IE57930B1 (OSRAM) |
| IL (1) | IL72234A (OSRAM) |
| NZ (1) | NZ208757A (OSRAM) |
| PH (1) | PH20342A (OSRAM) |
| ZA (1) | ZA844661B (OSRAM) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB8408924D0 (en) * | 1984-04-06 | 1984-05-16 | Dobfar Spa | 3-azinomethyl rifamycins |
| JPH02501301A (ja) * | 1987-09-25 | 1990-05-10 | チバ‐ガイギー アクチェンゲゼルシャフト | ４‐（トリアルキルベンジル）‐ピペラジニル化合物のジアシル誘導体 |
| US5180718A (en) * | 1989-03-02 | 1993-01-19 | Ciba-Geigy Corporation | Acyl derivatives of oxazolorifamycins |
| EP0944311B1 (en) * | 1996-11-19 | 2006-03-01 | Georgetown University | Method for antagonizing HEREGUlin or its receptor and use for the inhibition of cancer cells |
| US7122525B2 (en) * | 2001-11-21 | 2006-10-17 | Activbiotics, Inc. | Targeted therapeutics and uses thereof |
| US7137963B2 (en) * | 2002-08-26 | 2006-11-21 | Flowcardia, Inc. | Ultrasound catheter for disrupting blood vessel obstructions |
| US7820652B2 (en) * | 2003-09-24 | 2010-10-26 | Activbiotics Pharma, Llc | Regimen for the administration of rifamycin-class antibiotics |
| WO2015157512A1 (en) * | 2014-04-11 | 2015-10-15 | Drexel University | Novel methods and kits for detecting a rifamycin, or derivative or analogue thereof |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR208F (OSRAM) * | 1964-07-31 | |||
| GB1159267A (en) * | 1966-11-03 | 1969-07-23 | Lepetit Spa | Rifamycin Derivatives |
| NL145554B (nl) * | 1967-06-07 | 1975-04-15 | Lepetit Spa | Werkwijze voor het bereiden van een 3-formylrifamycine sv-derivaat |
| AR207762A1 (es) * | 1973-07-25 | 1976-10-29 | Archifar Ind Chim Trentino | Procedimiento para la preparacion de 3-((4-metil-1-piperazin-1-il)-imino)-metil-rifamicina sv o rifampicina |
| GB1594134A (en) * | 1977-11-25 | 1981-07-30 | Holco Investment Inc | Rifamycins |
| US4298692A (en) * | 1979-01-25 | 1981-11-03 | Ciba-Geigy Corporation | Fermentation process for producing a rifamycin derivative |
| US4411896A (en) * | 1981-06-03 | 1983-10-25 | Ciba-Geigy Corporation | Rifamycins, their compositions and use as antibiotics |
-
1983
- 1983-07-04 GB GB838318072A patent/GB8318072D0/en active Pending
-
1984
- 1984-06-15 AU AU29411/84A patent/AU558707B2/en not_active Ceased
- 1984-06-17 AT AT84106938T patent/ATE29136T1/de not_active IP Right Cessation
- 1984-06-17 EP EP84106938A patent/EP0133887B1/en not_active Expired
- 1984-06-17 DE DE8484106938T patent/DE3465597D1/de not_active Expired
- 1984-06-20 ZA ZA844661A patent/ZA844661B/xx unknown
- 1984-06-26 DK DK311484A patent/DK157875C/da active
- 1984-06-27 IL IL72234A patent/IL72234A/xx unknown
- 1984-06-27 PH PH30892A patent/PH20342A/en unknown
- 1984-06-29 US US06/626,358 patent/US4585589A/en not_active Expired - Fee Related
- 1984-07-02 JP JP59135371A patent/JPS6036490A/ja active Granted
- 1984-07-03 NZ NZ208757A patent/NZ208757A/en unknown
- 1984-07-03 CA CA000457960A patent/CA1212670A/en not_active Expired
- 1984-07-03 IE IE1693/84A patent/IE57930B1/en not_active IP Right Cessation
- 1984-07-03 ES ES533957A patent/ES533957A0/es active Granted
- 1984-07-03 KR KR1019840003836A patent/KR910005847B1/ko not_active Expired
- 1984-07-03 HU HU842575A patent/HU190576B/hu not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| EP0133887B1 (en) | 1987-08-26 |
| DE3465597D1 (en) | 1987-10-01 |
| KR850001207A (ko) | 1985-03-16 |
| GB8318072D0 (en) | 1983-08-03 |
| CA1212670A (en) | 1986-10-14 |
| DK311484A (da) | 1985-01-05 |
| JPH0544467B2 (OSRAM) | 1993-07-06 |
| ES8601949A1 (es) | 1985-11-01 |
| AU2941184A (en) | 1985-01-10 |
| ES533957A0 (es) | 1985-11-01 |
| IE57930B1 (en) | 1993-05-19 |
| AU558707B2 (en) | 1987-02-05 |
| DK157875B (da) | 1990-02-26 |
| PH20342A (en) | 1986-12-04 |
| ZA844661B (en) | 1985-04-24 |
| HUT36128A (en) | 1985-08-28 |
| NZ208757A (en) | 1987-08-31 |
| JPS6036490A (ja) | 1985-02-25 |
| US4585589A (en) | 1986-04-29 |
| IE841693L (en) | 1985-01-04 |
| IL72234A0 (en) | 1984-10-31 |
| ATE29136T1 (de) | 1987-09-15 |
| DK311484D0 (da) | 1984-06-26 |
| HU190576B (en) | 1986-09-29 |
| IL72234A (en) | 1987-09-16 |
| EP0133887A1 (en) | 1985-03-13 |
| KR910005847B1 (ko) | 1991-08-05 |
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