DK149611C - METHOD OF ANALOGUE FOR THE PREPARATION OF TRH-ANALOGUE TRIPEPTIDAMIDES OR THERAPEUTICALLY ACCEPTABLE COMPLEXES OR SALTS THEREOF - Google Patents

METHOD OF ANALOGUE FOR THE PREPARATION OF TRH-ANALOGUE TRIPEPTIDAMIDES OR THERAPEUTICALLY ACCEPTABLE COMPLEXES OR SALTS THEREOF

Info

Publication number
DK149611C
DK149611C DK274680A DK274680A DK149611C DK 149611 C DK149611 C DK 149611C DK 274680 A DK274680 A DK 274680A DK 274680 A DK274680 A DK 274680A DK 149611 C DK149611 C DK 149611C
Authority
DK
Denmark
Prior art keywords
analogue
tripeptidamides
trh
salts
preparation
Prior art date
Application number
DK274680A
Other languages
Danish (da)
Other versions
DK274680A (en
DK149611B (en
Inventor
Lajos Kisfaludy
Tamas Szirtes
Lajos Balaspiri
Eva Palosi
Laszlo Szporny
Adam Sarkadi
Original Assignee
Richter Gedeon Vegyeszet
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Richter Gedeon Vegyeszet filed Critical Richter Gedeon Vegyeszet
Publication of DK274680A publication Critical patent/DK274680A/en
Publication of DK149611B publication Critical patent/DK149611B/en
Application granted granted Critical
Publication of DK149611C publication Critical patent/DK149611C/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06008—Dipeptides with the first amino acid being neutral
    • C07K5/06017—Dipeptides with the first amino acid being neutral and aliphatic
    • C07K5/06034—Dipeptides with the first amino acid being neutral and aliphatic the side chain containing 2 to 4 carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06008—Dipeptides with the first amino acid being neutral
    • C07K5/06017—Dipeptides with the first amino acid being neutral and aliphatic
    • C07K5/06034—Dipeptides with the first amino acid being neutral and aliphatic the side chain containing 2 to 4 carbon atoms
    • C07K5/06043—Leu-amino acid
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06104—Dipeptides with the first amino acid being acidic
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08—Tripeptides
    • C07K5/0821—Tripeptides with the first amino acid being heterocyclic, e.g. His, Pro, Trp
    • C07K5/0825—Tripeptides with the first amino acid being heterocyclic, e.g. His, Pro, Trp and Glp-amino acid; Derivatives thereof

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Neurology (AREA)
  • Engineering & Computer Science (AREA)
  • Biomedical Technology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurosurgery (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
DK274680A 1979-06-28 1980-06-26 METHOD OF ANALOGUE FOR THE PREPARATION OF TRH-ANALOGUE TRIPEPTIDAMIDES OR THERAPEUTICALLY ACCEPTABLE COMPLEXES OR SALTS THEREOF DK149611C (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
HURI000717 1979-06-28
HU79RI717A HU180925B (en) 1979-06-28 1979-06-28 Process for producing tripeptide-amides trh-analogues,effectives on the central nerve systhem

Publications (3)

Publication Number Publication Date
DK274680A DK274680A (en) 1980-12-29
DK149611B DK149611B (en) 1986-08-11
DK149611C true DK149611C (en) 1987-01-26

Family

ID=11001100

Family Applications (1)

Application Number Title Priority Date Filing Date
DK274680A DK149611C (en) 1979-06-28 1980-06-26 METHOD OF ANALOGUE FOR THE PREPARATION OF TRH-ANALOGUE TRIPEPTIDAMIDES OR THERAPEUTICALLY ACCEPTABLE COMPLEXES OR SALTS THEREOF

Country Status (21)

Country Link
US (1) US4299821A (en)
JP (1) JPS5636442A (en)
AT (1) AT373578B (en)
AU (1) AU538100B2 (en)
BE (1) BE884014A (en)
CA (1) CA1151154A (en)
CH (1) CH650518A5 (en)
CS (1) CS239907B2 (en)
DD (1) DD151746A5 (en)
DE (1) DE3024313A1 (en)
DK (1) DK149611C (en)
FI (1) FI74473C (en)
FR (1) FR2460292A1 (en)
GB (1) GB2058080B (en)
HU (1) HU180925B (en)
IL (1) IL60407A (en)
IT (1) IT1150023B (en)
NL (1) NL8003767A (en)
PL (1) PL127100B1 (en)
SE (1) SE447261B (en)
SU (1) SU963463A3 (en)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2533209B1 (en) * 1982-09-22 1985-11-08 Centre Nat Rech Scient LIPOPEPTIDES, THEIR OBTAINMENT AND THEIR APPLICATION AS EMULSIFIERS
WO1986003746A1 (en) * 1984-12-14 1986-07-03 La Trobe University Amino acid and peptide inhibitors of human leucocytic elastase
IT1186733B (en) * 1985-06-05 1987-12-16 Eniricerche Spa TRIPEPTIDIC COMPOUNDS WITH HYPOTHENSIVE ACTION
FR2597100A1 (en) * 1986-01-21 1987-10-16 Nippon Shinyaku Co Ltd PYROGLUTAMIDE DERIVATIVES
HUT74733A (en) * 1993-11-09 1997-02-28 Merck & Co Inc Piperidines, pyrrolidines and hexahydro-1h-azepines promote release of growth hormone
US5494919A (en) * 1993-11-09 1996-02-27 Merck & Co., Inc. 2-substituted piperidines, pyrrolidines and hexahydro-1H-azepines promote release of growth hormone
FR2733995B1 (en) * 1995-05-09 1997-07-25 Inst Nat Sante Rech Med INHIBITORS OF INACTIVATION OF ENDOGENOUS NEUROPEPTIDES IN PARTICULAR CHOLECYSTOKININ, METHODS OF PREPARING THEIR USE AS MEDICAMENTS AND METHOD OF SCREENING MEDICINAL PRODUCTS
DE19527575A1 (en) * 1995-07-28 1997-01-30 Basf Ag Process for the preparation of peptide active ingredients
US20020151502A1 (en) * 1997-10-09 2002-10-17 Albert Sattin Tri-peptides for neurological and neurobehavior applications
US20050233973A1 (en) * 1997-10-09 2005-10-20 Albert Sattin Tri-peptides for antidepressant applications
US7462595B2 (en) * 2004-09-17 2008-12-09 Prange Jr Arthur Jergen Methods for treating cancer-related fatigue

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3959248A (en) * 1974-04-03 1976-05-25 Merck & Co., Inc. Analogs of thyrotropin-releasing hormone
LU73294A1 (en) * 1975-09-02 1977-05-11

Also Published As

Publication number Publication date
DE3024313C2 (en) 1991-05-29
SU963463A3 (en) 1982-09-30
IT1150023B (en) 1986-12-10
FR2460292B1 (en) 1983-11-18
US4299821A (en) 1981-11-10
DD151746A5 (en) 1981-11-04
ATA334680A (en) 1983-06-15
SE447261B (en) 1986-11-03
AU538100B2 (en) 1984-07-26
FI74473B (en) 1987-10-30
SE8004744L (en) 1980-12-29
FR2460292A1 (en) 1981-01-23
IL60407A (en) 1984-11-30
AU5971980A (en) 1981-01-08
FI74473C (en) 1988-02-08
NL8003767A (en) 1980-12-30
GB2058080B (en) 1983-02-23
DK274680A (en) 1980-12-29
GB2058080A (en) 1981-04-08
AT373578B (en) 1984-02-10
PL225268A1 (en) 1981-10-16
FI802057A (en) 1980-12-29
IL60407A0 (en) 1980-09-16
PL127100B1 (en) 1983-09-30
IT8023096A0 (en) 1980-06-26
DK149611B (en) 1986-08-11
CA1151154A (en) 1983-08-02
HU180925B (en) 1983-05-30
CH650518A5 (en) 1985-07-31
CS239907B2 (en) 1986-01-16
DE3024313A1 (en) 1981-01-29
BE884014A (en) 1980-12-29
JPS5636442A (en) 1981-04-09
CS458480A2 (en) 1985-05-15

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