DK146822C - ANALOGY PROCEDURE FOR PREPARING DERIVATIVES OF 4-DESACETYL-VINBLASTIN OR SALTS THEREOF - Google Patents

ANALOGY PROCEDURE FOR PREPARING DERIVATIVES OF 4-DESACETYL-VINBLASTIN OR SALTS THEREOF

Info

Publication number
DK146822C
DK146822C DK398577A DK398577A DK146822C DK 146822 C DK146822 C DK 146822C DK 398577 A DK398577 A DK 398577A DK 398577 A DK398577 A DK 398577A DK 146822 C DK146822 C DK 146822C
Authority
DK
Denmark
Prior art keywords
desacetyl
vinblastin
salts
preparing derivatives
analogy procedure
Prior art date
Application number
DK398577A
Other languages
Danish (da)
Other versions
DK146822B (en
DK398577A (en
Inventor
George Joseph Cullinan
Koert Gerzon
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of DK398577A publication Critical patent/DK398577A/en
Publication of DK146822B publication Critical patent/DK146822B/en
Application granted granted Critical
Publication of DK146822C publication Critical patent/DK146822C/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D519/00Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
    • C07D519/04Dimeric indole alkaloids, e.g. vincaleucoblastine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
DK398577A 1976-09-08 1977-09-07 ANALOGY PROCEDURE FOR PREPARING DERIVATIVES OF 4-DESACETYL-VINBLASTIN OR SALTS THEREOF DK146822C (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US72165076A 1976-09-08 1976-09-08
US72165076 1976-09-08

Publications (3)

Publication Number Publication Date
DK398577A DK398577A (en) 1978-03-09
DK146822B DK146822B (en) 1984-01-16
DK146822C true DK146822C (en) 1984-06-25

Family

ID=24898757

Family Applications (1)

Application Number Title Priority Date Filing Date
DK398577A DK146822C (en) 1976-09-08 1977-09-07 ANALOGY PROCEDURE FOR PREPARING DERIVATIVES OF 4-DESACETYL-VINBLASTIN OR SALTS THEREOF

Country Status (27)

Country Link
JP (1) JPS5340799A (en)
AR (3) AR226411A1 (en)
AT (1) AT360513B (en)
AU (1) AU511055B2 (en)
BE (1) BE858451A (en)
CA (1) CA1082179A (en)
CH (1) CH631990A5 (en)
DD (1) DD133055A5 (en)
DE (1) DE2739443A1 (en)
DK (1) DK146822C (en)
ES (1) ES462229A1 (en)
FR (1) FR2364220A1 (en)
GB (1) GB1586709A (en)
GR (1) GR69783B (en)
HU (1) HU180722B (en)
IE (1) IE45558B1 (en)
IL (1) IL52731A0 (en)
MX (1) MX4740E (en)
NL (1) NL7709806A (en)
NZ (1) NZ184932A (en)
PH (1) PH14771A (en)
PL (1) PL104309B1 (en)
PT (1) PT66984B (en)
RO (3) RO77921A (en)
SE (1) SE434953B (en)
YU (1) YU209777A (en)
ZA (1) ZA774988B (en)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
USRE30561E (en) * 1976-12-06 1981-03-31 Eli Lilly And Company Vinca alkaloid intermediates
US4199504A (en) * 1978-05-15 1980-04-22 Eli Lilly And Company Bridged cathranthus alkaloid dimers
AR225153A1 (en) * 1978-10-10 1982-02-26 Lilly Co Eli A PROCEDURE FOR THE PREPARATION OF VINDESINE SULPHATE
US4357334A (en) 1980-03-20 1982-11-02 Eli Lilly And Company Use of VLB 3-(2-chloroethyl) carboxamide in treating neoplasms
OA06421A (en) * 1980-06-10 1981-09-30 Omnium Chimique Sa Process for the preparation of N- (vinblastinoyl-23) derivatives of amino acids and peptides.
US4362664A (en) * 1980-12-29 1982-12-07 Eli Lilly And Company Vinblastine oxazolidinedione disulfides and related compounds
JPH075608B2 (en) * 1986-01-13 1995-01-25 イ−ル−セルタ−ク ソシエテ アノニム Vinblastine derivative

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR204004A1 (en) * 1973-04-02 1975-11-12 Lilly Co Eli PROCEDURES FOR PREPARING VINBLASTIN LEUROSIDINE AND LEUROCRISTINE DERIVATIVES
IL48685A (en) * 1975-01-09 1980-03-31 Lilly Co Eli Amides of vincadioline and vinblastine

Also Published As

Publication number Publication date
ZA774988B (en) 1979-03-28
CA1082179A (en) 1980-07-22
AR231643A1 (en) 1985-01-31
AR226411A1 (en) 1982-07-15
FR2364220B1 (en) 1980-04-25
DD133055A5 (en) 1978-11-29
IE45558B1 (en) 1982-09-22
AU511055B2 (en) 1980-07-24
PT66984A (en) 1977-10-01
ATA644277A (en) 1980-06-15
JPS5340799A (en) 1978-04-13
YU209777A (en) 1982-08-31
DE2739443C2 (en) 1991-08-14
CH631990A5 (en) 1982-09-15
RO77922A (en) 1981-12-25
JPS624398B2 (en) 1987-01-30
AU2803977A (en) 1979-02-22
PT66984B (en) 1979-02-13
DK146822B (en) 1984-01-16
DK398577A (en) 1978-03-09
DE2739443A1 (en) 1978-03-09
GB1586709A (en) 1981-03-25
NZ184932A (en) 1979-11-01
AR230642A1 (en) 1984-05-31
NL7709806A (en) 1978-03-10
MX4740E (en) 1982-08-25
RO77921A (en) 1981-12-25
PL200607A1 (en) 1978-05-22
IE771700L (en) 1978-03-08
BE858451A (en) 1978-03-07
SE434953B (en) 1984-08-27
ES462229A1 (en) 1978-07-16
RO72474A (en) 1982-05-10
SE7710059L (en) 1978-03-09
IL52731A0 (en) 1977-10-31
PH14771A (en) 1981-12-09
HU180722B (en) 1983-04-29
AT360513B (en) 1981-01-12
GR69783B (en) 1982-07-07
FR2364220A1 (en) 1978-04-07
PL104309B1 (en) 1979-08-31

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