DK139870B - Analogous process for the preparation of pharmacologically active heterocyclic compounds. - Google Patents
Analogous process for the preparation of pharmacologically active heterocyclic compounds.Info
- Publication number
- DK139870B DK139870B DK90972AA DK90972A DK139870B DK 139870 B DK139870 B DK 139870B DK 90972A A DK90972A A DK 90972AA DK 90972 A DK90972 A DK 90972A DK 139870 B DK139870 B DK 139870B
- Authority
- DK
- Denmark
- Prior art keywords
- preparation
- pharmacologically active
- heterocyclic compounds
- analogous process
- active heterocyclic
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/62—Oxygen or sulfur atoms
- C07D213/70—Sulfur atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D213/28—Radicals substituted by singly-bound oxygen or sulphur atoms
- C07D213/32—Sulfur atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/62—Oxygen or sulfur atoms
- C07D213/63—One oxygen atom
- C07D213/65—One oxygen atom attached in position 3 or 5
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/72—Nitrogen atoms
- C07D213/74—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/84—Sulfur atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/06—Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
- C07D249/10—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D249/12—Oxygen or sulfur atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/30—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D263/34—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D263/46—Sulfur atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/36—Sulfur atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
- C07D285/01—Five-membered rings
- C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
- C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
- C07D285/12—1,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles
- C07D285/125—1,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles with oxygen, sulfur or nitrogen atoms, directly attached to ring carbon atoms, the nitrogen atoms not forming part of a nitro radical
- C07D285/135—Nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Handcart (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Priority Applications (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DK349776A DK137645B (en) | 1971-03-09 | 1976-08-03 | Heterocyclically substituted aminoalkylthioethers for use as intermediates in the preparation of the corresponding pharmacologically active thioethers. |
DK580278A DK144308C (en) | 1971-03-09 | 1978-12-22 | METHOD OF ANALOGUE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE HETEROCYCLIC SUBSTITUTED GUANIDINES |
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB635271A GB1338169A (en) | 1971-03-09 | 1971-03-09 | Ureas thioureas and guanidines |
GB3433471 | 1971-07-22 |
Publications (2)
Publication Number | Publication Date |
---|---|
DK139870B true DK139870B (en) | 1979-05-07 |
DK139870C DK139870C (en) | 1979-10-08 |
Family
ID=26240626
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK90972AA DK139870B (en) | 1971-03-09 | 1972-02-28 | Analogous process for the preparation of pharmacologically active heterocyclic compounds. |
Country Status (21)
Country | Link |
---|---|
JP (5) | JPS5324422B1 (en) |
AR (2) | AR197080A1 (en) |
BE (1) | BE779775A (en) |
CY (1) | CY856A (en) |
DK (1) | DK139870B (en) |
EG (1) | EG10876A (en) |
ES (1) | ES400587A1 (en) |
FI (1) | FI60393C (en) |
HK (1) | HK55176A (en) |
HU (1) | HU164509B (en) |
IE (1) | IE36050B1 (en) |
IL (1) | IL38821A (en) |
IT (1) | IT1041101B (en) |
KE (1) | KE2625A (en) |
MY (1) | MY7600228A (en) |
NO (1) | NO133196C (en) |
PH (2) | PH12207A (en) |
SE (3) | SE402288B (en) |
SG (1) | SG28576G (en) |
SU (1) | SU460628A3 (en) |
ZM (1) | ZM3672A1 (en) |
Families Citing this family (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1397436A (en) * | 1972-09-05 | 1975-06-11 | Smith Kline French Lab | Heterocyclic n-cyanoguinidines |
US4083988A (en) * | 1972-09-05 | 1978-04-11 | Smith Kline & French Laboratories Limited | Pharmacologically active compounds |
GB1398426A (en) * | 1972-09-05 | 1975-06-18 | Smith Kline French Lab | Heterocyclic substituted guanidines |
US4000296A (en) * | 1972-09-05 | 1976-12-28 | Smith Kline & French Laboratories Limited | Imidazole alkylguanidine compounds |
US4129657A (en) | 1975-03-21 | 1978-12-12 | Smith, Kline & French Laboratories Limited | Imidazole guanidines and use as inhibitors of histamine activity |
IL56265A (en) * | 1977-12-28 | 1982-08-31 | Om Lab Sa | Process for preparing imidazolyl methylthio guanidine derivatives and a novel intermediate therefor |
JPH07107054B2 (en) * | 1987-05-20 | 1995-11-15 | 株式会社日本触媒 | Process for producing 4-methyl-5-[(2-aminoethyl) thiomethyl] imidazole dihydrochloride |
JP2933739B2 (en) * | 1990-04-09 | 1999-08-16 | 明治製菓株式会社 | Thiazole or imidazole derivatives and anti-ulcer agents |
-
1972
- 1972-02-03 IE IE136/72A patent/IE36050B1/en unknown
- 1972-02-08 EG EG48/72A patent/EG10876A/en active
- 1972-02-18 PH PH13276A patent/PH12207A/en unknown
- 1972-02-22 ZM ZM36/72A patent/ZM3672A1/en unknown
- 1972-02-23 IL IL38821A patent/IL38821A/en unknown
- 1972-02-24 BE BE779775A patent/BE779775A/en not_active IP Right Cessation
- 1972-02-25 SU SU1751534A patent/SU460628A3/en active
- 1972-02-28 DK DK90972AA patent/DK139870B/en not_active IP Right Cessation
- 1972-03-03 FI FI580/72A patent/FI60393C/en active
- 1972-03-07 HU HUSI1249A patent/HU164509B/hu unknown
- 1972-03-07 AR AR240830A patent/AR197080A1/en active
- 1972-03-08 NO NO747/72A patent/NO133196C/no unknown
- 1972-03-08 IT IT21604/72A patent/IT1041101B/en active
- 1972-03-08 SE SE7202933A patent/SE402288B/en unknown
- 1972-03-09 CY CY856A patent/CY856A/en unknown
- 1972-03-09 ES ES400587A patent/ES400587A1/en not_active Expired
- 1972-03-09 JP JP2437172A patent/JPS5324422B1/ja active Pending
- 1972-09-29 AR AR244346A patent/AR197093A1/en active
-
1974
- 1974-10-09 SE SE7412680A patent/SE410103B/en not_active IP Right Cessation
-
1976
- 1976-05-18 KE KE2625*UA patent/KE2625A/en unknown
- 1976-09-08 HK HK551/76*UA patent/HK55176A/en unknown
- 1976-09-30 SE SE7610842A patent/SE430689B/en not_active IP Right Cessation
- 1976-12-31 MY MY1976228A patent/MY7600228A/en unknown
- 1976-12-31 SG SG285/76A patent/SG28576G/en unknown
-
1977
- 1977-10-14 PH PH20334A patent/PH12247A/en unknown
- 1977-12-22 JP JP52160989A patent/JPS5811948B2/en not_active Expired
- 1977-12-22 JP JP16098877A patent/JPS53119868A/en active Granted
- 1977-12-22 JP JP16098777A patent/JPS53119867A/en active Granted
-
1978
- 1978-09-19 JP JP11573678A patent/JPS5459275A/en active Pending
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
DK137329B (en) | Analogous process for the preparation of 2-carbalkoxyaminobenzimidazole derivatives. | |
DK133672B (en) | Analogous process for the preparation of imidazole derivatives. | |
DK134316B (en) | Process for the preparation of methyl substituted cuinones. | |
DK136981B (en) | Analogous process for the preparation of basic substituted benzylphthalazone derivatives. | |
DK133811B (en) | Analogous process for the preparation of heterocyclic esters of benzopyranopyridines. | |
DK127119B (en) | Analogous process for the preparation of 6-amino-9-benzylpurine compounds. | |
DK139870B (en) | Analogous process for the preparation of pharmacologically active heterocyclic compounds. | |
DK130212B (en) | Analogous process for the preparation of 7-aminoindazole derivatives. | |
DK131465B (en) | Analogous process for the preparation of pyrimidinone compounds. | |
DK138796B (en) | Analogous process for the preparation of 2-carboxypyrazine-4-oxide derivatives. | |
DK135122B (en) | Analogous process for the preparation of 4-aryl-5-aminoalkyl-4-oxazolin-2-one derivatives. | |
DK133464B (en) | Analogous process for the preparation of nitrosourine derivatives. | |
DK127297B (en) | Analogous process for the preparation of heterocyclically substituted nebularin derivatives. | |
DK126998B (en) | Analogous process for the preparation of amino-s-triazolylbenzenesulfonamide compounds. | |
DK133809B (en) | Analogous process for the preparation of heterocyclic compounds. | |
DK133902B (en) | Process for the preparation of Cephalosporin C. | |
DK129794B (en) | Analogous process for the preparation of N-acyl-3- (piperazinoethyl) -pyrazoles. | |
DK139871B (en) | Analogous process for the preparation of 3-isonicotinoyl-benzofuran derivatives. | |
DK134012B (en) | Process for the preparation of thioformamide. | |
DK138950B (en) | Analogous process for the preparation of alpha-aminopenicillin or cephalosporin derivatives. | |
DK139583B (en) | Analogous process for the preparation of penicillins. | |
DK129658B (en) | Process for the preparation of 3-substituted thienyl compounds. | |
DK128928B (en) | Analogous process for the preparation of rifamycin derivatives. | |
DK138323B (en) | Process for the preparation of bis-chromonyl compounds. | |
DK130980B (en) | Process for the preparation of penicillin compounds. |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
PUP | Patent expired |