DK138988B - Analogifremgangsmåde til fremstilling af racemiske eller optisk aktive morphinanderivater. - Google Patents

Analogifremgangsmåde til fremstilling af racemiske eller optisk aktive morphinanderivater.

Info

Publication number
DK138988B
DK138988B DK106673AA DK106673A DK138988B DK 138988 B DK138988 B DK 138988B DK 106673A A DK106673A A DK 106673AA DK 106673 A DK106673 A DK 106673A DK 138988 B DK138988 B DK 138988B
Authority
DK
Denmark
Prior art keywords
racemic
preparation
optically active
analogous process
morphinan derivatives
Prior art date
Application number
DK106673AA
Other languages
Danish (da)
English (en)
Other versions
DK138988C (zh
Inventor
Ernest Mohacsi
Willy Leimgruber
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of DK138988B publication Critical patent/DK138988B/da
Application granted granted Critical
Publication of DK138988C publication Critical patent/DK138988C/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D221/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/22—Bridged ring systems
    • C07D221/26—Benzomorphans
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
    • C07D217/12—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with radicals, substituted by hetero atoms, attached to carbon atoms of the nitrogen-containing ring
    • C07D217/18—Aralkyl radicals
    • C07D217/20—Aralkyl radicals with oxygen atoms directly attached to the aromatic ring of said aralkyl radical, e.g. papaverine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D221/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/22—Bridged ring systems
    • C07D221/28—Morphinans

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK106673AA 1972-03-10 1973-02-27 Analogifremgangsmåde til fremstilling af racemiske eller optisk aktive morphinanderivater. DK138988B (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US23371572A 1972-03-10 1972-03-10
US00299478A US3810899A (en) 1972-03-10 1972-10-20 2-hydroxy-n-substituted-morphinan derivatives

Publications (2)

Publication Number Publication Date
DK138988B true DK138988B (da) 1978-11-27
DK138988C DK138988C (zh) 1979-05-07

Family

ID=26927165

Family Applications (1)

Application Number Title Priority Date Filing Date
DK106673AA DK138988B (da) 1972-03-10 1973-02-27 Analogifremgangsmåde til fremstilling af racemiske eller optisk aktive morphinanderivater.

Country Status (11)

Country Link
US (1) US3810899A (zh)
AU (1) AU475007B2 (zh)
CA (1) CA1014954A (zh)
CH (2) CH586205A5 (zh)
DK (1) DK138988B (zh)
FR (1) FR2181800B1 (zh)
GB (1) GB1402502A (zh)
IL (1) IL41562A (zh)
NL (1) NL7303050A (zh)
PH (1) PH11649A (zh)
SE (1) SE403908B (zh)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4556712A (en) * 1981-05-20 1985-12-03 The United States Of America As Represented By The Secretary Of The Department Of Health And Human Services Preparation and racemization of chiral 1-benzyl-1,2,3,4-tetrahydroisoquinolines
US4410700A (en) * 1980-07-03 1983-10-18 The United States Of America As Represented By The Department Of Health And Human Services Preparation of chiral 1-benzyl-1,2,3,4-tetrahydroisoquinolines by optical resolution
US4496762A (en) * 1983-03-29 1985-01-29 Eastman Kodak Company Process for the preparation of N-(2-(cyclo-hexen-1-yl)ethyl)-4-methoxybenzeneacetamide
US5905153A (en) * 1996-10-02 1999-05-18 Roche Vitamins Inc. Process for preparing (9α,13α,14α)-1-(3-methoxy-morphinan-17-yl)alkanones
US5849917A (en) * 1996-10-02 1998-12-15 Roche Vitamins Inc. Process for the preparation of isoquinoline compounds
ATE438649T1 (de) * 2006-04-21 2009-08-15 Zach System Spa Verfahren zur herstellung von dorzolamid

Also Published As

Publication number Publication date
AU475007B2 (en) 1976-08-12
IL41562A (en) 1977-04-29
FR2181800A1 (zh) 1973-12-07
AU5222773A (en) 1974-08-15
DK138988C (zh) 1979-05-07
PH11649A (en) 1978-05-08
CA1014954A (en) 1977-08-02
FR2181800B1 (zh) 1976-05-14
CH586205A5 (zh) 1977-03-31
IL41562A0 (en) 1973-04-30
GB1402502A (en) 1975-08-13
US3810899A (en) 1974-05-14
CH591449A5 (zh) 1977-09-15
SE403908B (sv) 1978-09-11
NL7303050A (zh) 1973-09-12

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