DK138698B - Fremgangsmåde til fremstilling af 13-ethynyl-steroider. - Google Patents

Fremgangsmåde til fremstilling af 13-ethynyl-steroider.

Info

Publication number
DK138698B
DK138698B DK563775AA DK563775A DK138698B DK 138698 B DK138698 B DK 138698B DK 563775A A DK563775A A DK 563775AA DK 563775 A DK563775 A DK 563775A DK 138698 B DK138698 B DK 138698B
Authority
DK
Denmark
Prior art keywords
preparation
ethynyl
steroids
ethynyl steroids
Prior art date
Application number
DK563775AA
Other languages
English (en)
Other versions
DK138698C (da
DK563775A (da
Inventor
Michel Biollaz
Jaroslav Kalvoda
Original Assignee
Ciba Geigy Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy Ag filed Critical Ciba Geigy Ag
Publication of DK563775A publication Critical patent/DK563775A/da
Publication of DK138698B publication Critical patent/DK138698B/da
Application granted granted Critical
Publication of DK138698C publication Critical patent/DK138698C/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J21/00Normal steroids containing carbon, hydrogen, halogen or oxygen having an oxygen-containing hetero ring spiro-condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J21/005Ketals
    • C07J21/008Ketals at position 17
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J1/00Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0003Androstane derivatives
    • C07J1/0011Androstane derivatives substituted in position 17 by a keto group
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J1/00Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0003Androstane derivatives
    • C07J1/0018Androstane derivatives substituted in position 17 beta, not substituted in position 17 alfa
    • C07J1/0022Androstane derivatives substituted in position 17 beta, not substituted in position 17 alfa the substituent being an OH group free esterified or etherified
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J1/00Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0003Androstane derivatives
    • C07J1/0033Androstane derivatives substituted in position 17 alfa and 17 beta
    • C07J1/004Androstane derivatives substituted in position 17 alfa and 17 beta the substituent in position 17 alfa being an unsaturated hydrocarbon group
    • C07J1/0048Alkynyl derivatives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J1/00Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0051Estrane derivatives
    • C07J1/0059Estrane derivatives substituted in position 17 by a keto group
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J1/00Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0051Estrane derivatives
    • C07J1/0066Estrane derivatives substituted in position 17 beta not substituted in position 17 alfa
    • C07J1/007Estrane derivatives substituted in position 17 beta not substituted in position 17 alfa the substituent being an OH group free esterified or etherified
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J1/00Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0051Estrane derivatives
    • C07J1/0081Substituted in position 17 alfa and 17 beta
    • C07J1/0088Substituted in position 17 alfa and 17 beta the substituent in position 17 alfa being an unsaturated hydrocarbon group
    • C07J1/0096Alkynyl derivatives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J51/00Normal steroids with unmodified cyclopenta(a)hydrophenanthrene skeleton not provided for in groups C07J1/00 - C07J43/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
  • Fodder In General (AREA)
DK563775AA 1975-01-30 1975-12-11 Fremgangsmåde til fremstilling af 13-ethynyl-steroider. DK138698B (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH112375A CH606101A5 (da) 1975-01-30 1975-01-30

Publications (3)

Publication Number Publication Date
DK563775A DK563775A (da) 1976-07-31
DK138698B true DK138698B (da) 1978-10-16
DK138698C DK138698C (da) 1979-03-19

Family

ID=4203021

Family Applications (1)

Application Number Title Priority Date Filing Date
DK563775AA DK138698B (da) 1975-01-30 1975-12-11 Fremgangsmåde til fremstilling af 13-ethynyl-steroider.

Country Status (15)

Country Link
US (1) US4052421A (da)
JP (1) JPS51100068A (da)
AU (1) AU503505B2 (da)
BE (1) BE838019A (da)
CA (1) CA1065302A (da)
CH (1) CH606101A5 (da)
DE (1) DE2602891A1 (da)
DK (1) DK138698B (da)
ES (1) ES444689A1 (da)
FR (1) FR2299034A1 (da)
GB (1) GB1514621A (da)
IE (1) IE42468B1 (da)
IL (1) IL48937A (da)
SE (1) SE7514455L (da)
ZA (1) ZA76506B (da)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4297350A (en) * 1978-10-10 1981-10-27 The Upjohn Company Male contraceptive steroids and methods of use
US4289762A (en) * 1980-06-27 1981-09-15 Merrell Dow Pharmaceuticals Inc. 10-(1,2-Propadienyl) steroids as irreversible aromatase inhibitors
US4293548A (en) * 1980-09-02 1981-10-06 Merrell Dow Pharmaceuticals Inc. 18-Substituted pregn-4-ene-3,20-diones
ATE527192T1 (de) 2009-03-02 2011-10-15 Sala Jaime Marti Rotationsförderer für leichte gegenstände

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3959322A (en) * 1960-09-22 1976-05-25 Herchel Smith Synthesis of 13-alkyl-gon-4-ones
US3267005A (en) * 1963-10-23 1966-08-16 American Home Prod Resolution of racemic delta4-3-ketosteroids
US3798215A (en) * 1968-11-25 1974-03-19 Sandoz Ag Propadienyl-substituted carbinols

Also Published As

Publication number Publication date
CA1065302A (en) 1979-10-30
IE42468L (en) 1976-07-30
DK138698C (da) 1979-03-19
SE7514455L (sv) 1976-08-02
IL48937A0 (en) 1976-03-31
US4052421A (en) 1977-10-04
BE838019A (fr) 1976-07-29
CH606101A5 (da) 1978-10-13
IE42468B1 (en) 1980-08-13
AU503505B2 (en) 1979-09-06
GB1514621A (en) 1978-06-14
ZA76506B (en) 1977-01-26
JPS51100068A (da) 1976-09-03
ES444689A1 (es) 1977-05-16
IL48937A (en) 1979-07-25
FR2299034B1 (da) 1979-09-21
DE2602891A1 (de) 1976-08-05
FR2299034A1 (fr) 1976-08-27
DK563775A (da) 1976-07-31
AU1064476A (en) 1977-08-04

Similar Documents

Publication Publication Date Title
DK49676A (da) Fremgangsmade til fremstilling af hypolipidemiske midler
DK136655B (da) Analogifremgangsmåde til fremstilling af piperazinyliminorifamyciner.
DK113476A (da) Fremgangsmade til fremstilling af amoxicillintrihydrat
DK137835B (da) Analogifremgangsmåde til fremstilling af thienothiazinderivater.
DK107876A (da) Fremgangsmade til fremstilling af thiocarbamider
DK139846B (da) Analogifremgangsmåde til fremstilling af 3-alkoxypyrazin-2-carboxamider.
DK139969B (da) Analogifremgangsmåde til fremstilling af 1-alkylcarbamoyl-5-fluoruraciler.
DK150676A (da) Fremgangsmade til fremstilling af krystallinsk natrium-o-formyl-cefamandol
DK136656B (da) Analogifremgangsmåde til fremstilling af substituerede piperazinyliminorifamyciner.
DK139029B (da) Analogifremgangsmåde til fremstilling af 5-m-tolyloxyuracil.
DK137957B (da) Analogifremgangsmåde til fremstilling af 2-substituerede 5-fluorpyrimidin-4-oner.
DK415576A (da) Fremgangsmade til fremstilling af krystallinsk dipilocarpiniumpamoat
DK399976A (da) Fremgangsmade til fremstilling af aralkylamider
DK140728B (da) Fremgangsmåde til fremstilling af pregnanderivater.
DK139682B (da) Analogifremgangsmåde til fremstilling af eburnameninderivater.
DK138698B (da) Fremgangsmåde til fremstilling af 13-ethynyl-steroider.
DK29276A (da) Fremgangsmade til fremstilling af 8-bromothieno-triazolo-1,4-diazepiner
DK137646B (da) Fremgangsmåde til fremstilling af 6-chlor-2-chlormethyl-4-phenylquinazolin-3-oxid.
DK138694B (da) Fremgangsmåde til fremstilling af phenylphosphonothiodichlorid.
DK140502B (da) Analogifremgangsmåde til fremstilling af triazolobenzocycloalkylthiadiaziner.
DK140670B (da) Analogifremgangsmåde til fremstilling af ergopeptinderivater.
DK136652B (da) Fremgangsmåde til fremstilling af thieno-pyridinderivater.
DK141584C (da) Fremgangsmaade til fremstilling af slagseje vinylaromat-podecopolymere
DK424676A (da) Fremgangsmade til fremstilling af 2-alkylindan
DK480676A (da) Fremgangsmade til fremstilling af s-alkylphosphordihalogeniddithioater