DE60313657D1 - Antivirale zusammensetzungen - Google Patents
Antivirale zusammensetzungenInfo
- Publication number
- DE60313657D1 DE60313657D1 DE60313657T DE60313657T DE60313657D1 DE 60313657 D1 DE60313657 D1 DE 60313657D1 DE 60313657 T DE60313657 T DE 60313657T DE 60313657 T DE60313657 T DE 60313657T DE 60313657 D1 DE60313657 D1 DE 60313657D1
- Authority
- DE
- Germany
- Prior art keywords
- antiviral compositions
- antiviral
- compositions
- oxathiolan
- deoxythymidine
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
- 230000000840 anti-viral effect Effects 0.000 title 1
- 239000000203 mixture Substances 0.000 title 1
- JTEGQNOMFQHVDC-NKWVEPMBSA-N lamivudine Chemical compound O=C1N=C(N)C=CN1[C@H]1O[C@@H](CO)SC1 JTEGQNOMFQHVDC-NKWVEPMBSA-N 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- HBOMLICNUCNMMY-XLPZGREQSA-N zidovudine Chemical compound O=C1NC(=O)C(C)=CN1[C@@H]1O[C@H](CO)[C@@H](N=[N+]=[N-])C1 HBOMLICNUCNMMY-XLPZGREQSA-N 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
- A61K9/209—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat containing drug in at least two layers or in the core and in at least one outer layer
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
- A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
- A61K31/706—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom
- A61K31/7064—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines
- A61K31/7068—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines having oxo groups directly attached to the pyrimidine ring, e.g. cytidine, cytidylic acid
- A61K31/7072—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines having oxo groups directly attached to the pyrimidine ring, e.g. cytidine, cytidylic acid having two oxo groups directly attached to the pyrimidine ring, e.g. uridine, uridylic acid, thymidine, zidovudine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Epidemiology (AREA)
- Molecular Biology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Virology (AREA)
- Communicable Diseases (AREA)
- Tropical Medicine & Parasitology (AREA)
- AIDS & HIV (AREA)
- Oncology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Plural Heterocyclic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Saccharide Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US42518202P | 2002-11-08 | 2002-11-08 | |
US425182P | 2002-11-08 | ||
PCT/US2003/035830 WO2004043433A2 (en) | 2002-11-08 | 2003-11-07 | Pharmaceutical antiviral compositions |
Publications (2)
Publication Number | Publication Date |
---|---|
DE60313657D1 true DE60313657D1 (de) | 2007-06-14 |
DE60313657T2 DE60313657T2 (de) | 2008-01-03 |
Family
ID=32312939
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DE60313657T Expired - Lifetime DE60313657T2 (de) | 2002-11-08 | 2003-11-07 | Antivirale zusammensetzungen |
Country Status (9)
Country | Link |
---|---|
US (1) | US20050287177A1 (de) |
EP (1) | EP1567133B1 (de) |
JP (1) | JP2006508134A (de) |
AT (1) | ATE361059T1 (de) |
AU (1) | AU2003291457A1 (de) |
CA (1) | CA2505130C (de) |
DE (1) | DE60313657T2 (de) |
ES (1) | ES2286471T3 (de) |
WO (1) | WO2004043433A2 (de) |
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
MY169670A (en) | 2003-09-03 | 2019-05-08 | Tibotec Pharm Ltd | Combinations of a pyrimidine containing nnrti with rt inhibitors |
EP1658068B1 (de) | 2003-08-26 | 2009-02-18 | Smithkline Beecham Corporation | Cycloalkyl[b] kondensierte indole |
TW201414495A (zh) | 2005-04-04 | 2014-04-16 | Tibotec Pharm Ltd | Hiv-感染之預防 |
RU2008128424A (ru) * | 2005-12-14 | 2010-01-20 | Сипла Лимитед (In) | Фармацевтическая комбинация, включающая нуклеотидный и нуклеозидный ингибиторы обратной транскриптазы (такие как тенофовир и ламивудин) в различных частях дозы |
AR065720A1 (es) | 2007-03-14 | 2009-06-24 | Tibotec Pharm Ltd | Polvos para reconstitucion que comprenden rilpivirina dispersos en ciertos polimeros. uso. proceso. |
CA2686964A1 (en) * | 2007-06-06 | 2008-12-11 | Basf Se | Pharmaceutical formulation for the production of rapidly disintegrating tablets |
US20100184785A1 (en) * | 2007-06-06 | 2010-07-22 | Basf Se | Pharmaceutical formulation for the production of chewable tablets and lozenges |
US20100178340A1 (en) * | 2007-06-22 | 2010-07-15 | Bristol-Myers Squibb Company | Tableted compositions containing atazanavir |
WO2010137855A2 (en) * | 2009-05-27 | 2010-12-02 | Dasan Medichem Co., Ltd. | Multi-layer tablet comprising effervescent layer |
Family Cites Families (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4724232A (en) * | 1985-03-16 | 1988-02-09 | Burroughs Wellcome Co. | Treatment of human viral infections |
GB8707421D0 (en) * | 1987-03-27 | 1987-04-29 | Wellcome Found | Pharmaceutical formulations |
US5047407A (en) * | 1989-02-08 | 1991-09-10 | Iaf Biochem International, Inc. | 2-substituted-5-substituted-1,3-oxathiolanes with antiviral properties |
US5009895A (en) * | 1990-02-02 | 1991-04-23 | Merck & Co., Inc. | Sustained release with high and low viscosity HPMC |
GB9009861D0 (en) * | 1990-05-02 | 1990-06-27 | Glaxo Group Ltd | Chemical compounds |
CZ285232B6 (cs) * | 1991-05-16 | 1999-06-16 | Glaxo Group Limited | Protivirové směsi |
GB9111902D0 (en) * | 1991-06-03 | 1991-07-24 | Glaxo Group Ltd | Chemical compounds |
US6177435B1 (en) * | 1992-05-13 | 2001-01-23 | Glaxo Wellcome Inc. | Therapeutic combinations |
US5681581A (en) * | 1992-08-04 | 1997-10-28 | Dunn; James M. | Controlled release pharmaceutical formulations of 3'-azido-3'-deoxythymidine and methods of use |
US6113920A (en) * | 1996-10-31 | 2000-09-05 | Glaxo Wellcome Inc. | Pharmaceutical compositions |
GB9622681D0 (en) * | 1996-10-31 | 1997-01-08 | Glaxo Group Ltd | Pharmaceutical compositions |
US6541014B2 (en) * | 2000-10-13 | 2003-04-01 | Advancis Pharmaceutical Corp. | Antiviral product, use and formulation thereof |
-
2003
- 2003-11-07 WO PCT/US2003/035830 patent/WO2004043433A2/en active IP Right Grant
- 2003-11-07 JP JP2004552010A patent/JP2006508134A/ja active Pending
- 2003-11-07 EP EP03768857A patent/EP1567133B1/de not_active Expired - Lifetime
- 2003-11-07 ES ES03768857T patent/ES2286471T3/es not_active Expired - Lifetime
- 2003-11-07 CA CA002505130A patent/CA2505130C/en not_active Expired - Fee Related
- 2003-11-07 AT AT03768857T patent/ATE361059T1/de not_active IP Right Cessation
- 2003-11-07 US US10/533,325 patent/US20050287177A1/en not_active Abandoned
- 2003-11-07 DE DE60313657T patent/DE60313657T2/de not_active Expired - Lifetime
- 2003-11-07 AU AU2003291457A patent/AU2003291457A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
EP1567133B1 (de) | 2007-05-02 |
EP1567133A2 (de) | 2005-08-31 |
AU2003291457A1 (en) | 2004-06-03 |
WO2004043433A3 (en) | 2004-12-29 |
CA2505130C (en) | 2009-10-06 |
CA2505130A1 (en) | 2004-05-27 |
JP2006508134A (ja) | 2006-03-09 |
US20050287177A1 (en) | 2005-12-29 |
DE60313657T2 (de) | 2008-01-03 |
ES2286471T3 (es) | 2007-12-01 |
WO2004043433A2 (en) | 2004-05-27 |
AU2003291457A8 (en) | 2004-06-03 |
ATE361059T1 (de) | 2007-05-15 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
8364 | No opposition during term of opposition |