DE602004026781D1 - USE OF PIPAMPERONE AND A D2 RECEPTOR ANTAGONIST OR A SEROTONINE / DOPAMINE ANTAGONIST - Google Patents
USE OF PIPAMPERONE AND A D2 RECEPTOR ANTAGONIST OR A SEROTONINE / DOPAMINE ANTAGONISTInfo
- Publication number
- DE602004026781D1 DE602004026781D1 DE602004026781T DE602004026781T DE602004026781D1 DE 602004026781 D1 DE602004026781 D1 DE 602004026781D1 DE 602004026781 T DE602004026781 T DE 602004026781T DE 602004026781 T DE602004026781 T DE 602004026781T DE 602004026781 D1 DE602004026781 D1 DE 602004026781D1
- Authority
- DE
- Germany
- Prior art keywords
- antagonist
- pipamperone
- serotonine
- dopamine
- receptor antagonist
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Active
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
- A61K31/343—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide condensed with a carbocyclic ring, e.g. coumaran, bufuralol, befunolol, clobenfurol, amiodarone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
- A61K31/4545—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (11)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP03447279A EP1547650A1 (en) | 2003-12-02 | 2003-12-02 | Use of D4 and 5-HT2A antagonists, inverse agonists or partial agonists |
US10/725,965 US7884096B2 (en) | 2003-12-02 | 2003-12-02 | Method of treating mental disorders using of D4 and 5-HT2A antagonists, inverse agonists or partial agonists |
CA2451798A CA2451798C (en) | 2003-12-02 | 2003-12-02 | Use of d4 and 5-ht2a antagonists, inverse agonists or partial agonists |
EP04447001 | 2004-01-05 | ||
US10/752,423 US7855195B2 (en) | 2003-12-02 | 2004-01-06 | Method of treating mental disorders using D4 and 5-HT2A antagonists, inverse agonists or partial agonists |
EP04447066A EP1576985A1 (en) | 2004-03-18 | 2004-03-18 | Use of D4 and 5-HT2A antagonists, inverse agonists or partial agonists |
US10/803,793 US20050119249A1 (en) | 2003-12-02 | 2004-03-18 | Method of treating neurodegenerative diseases using D4 and 5-HT2A antagonists, inverse agonists or partial agonists |
CA 2461248 CA2461248C (en) | 2003-12-02 | 2004-03-18 | Use of d4 and 5-ht2a antagonists, inverse agonists or partial agonists |
EP04025035A EP1541197B8 (en) | 2003-12-02 | 2004-10-21 | Use of pipamperone and an SNDRI, SNRI or SSRI for the treatment of mood or anxiety disorders |
CA 2487529 CA2487529A1 (en) | 2003-12-02 | 2004-11-15 | Use of d4 and 5-ht2a antagonists, inverse agonists or partial agonists |
PCT/BE2004/000172 WO2005053796A1 (en) | 2003-12-02 | 2004-12-02 | Use of d4 and 5-ht2a antagonists, inverse agonists or partial agonists |
Publications (1)
Publication Number | Publication Date |
---|---|
DE602004026781D1 true DE602004026781D1 (en) | 2010-06-02 |
Family
ID=42134278
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DE602004026781T Active DE602004026781D1 (en) | 2003-12-02 | 2004-12-02 | USE OF PIPAMPERONE AND A D2 RECEPTOR ANTAGONIST OR A SEROTONINE / DOPAMINE ANTAGONIST |
Country Status (8)
Country | Link |
---|---|
AT (1) | ATE464901T1 (en) |
DE (1) | DE602004026781D1 (en) |
DK (1) | DK1708790T3 (en) |
ES (1) | ES2343962T3 (en) |
HR (1) | HRP20100376T1 (en) |
PT (1) | PT1708790E (en) |
RS (1) | RS51331B (en) |
SI (1) | SI1708790T1 (en) |
-
2004
- 2004-12-02 ES ES04801138T patent/ES2343962T3/en active Active
- 2004-12-02 RS RSP-2010/0323A patent/RS51331B/en unknown
- 2004-12-02 DE DE602004026781T patent/DE602004026781D1/en active Active
- 2004-12-02 PT PT04801138T patent/PT1708790E/en unknown
- 2004-12-02 DK DK04801138.1T patent/DK1708790T3/en active
- 2004-12-02 SI SI200431439T patent/SI1708790T1/en unknown
- 2004-12-02 AT AT04801138T patent/ATE464901T1/en active
-
2010
- 2010-07-06 HR HR20100376T patent/HRP20100376T1/en unknown
Also Published As
Publication number | Publication date |
---|---|
RS51331B (en) | 2011-02-28 |
ATE464901T1 (en) | 2010-05-15 |
HRP20100376T1 (en) | 2010-08-31 |
PT1708790E (en) | 2010-07-09 |
ES2343962T3 (en) | 2010-08-13 |
SI1708790T1 (en) | 2010-09-30 |
DK1708790T3 (en) | 2010-06-21 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
NO20051871D0 (en) | Opioid receptor antagonists | |
IS8190A (en) | New P2X7 receptor antagonists and their use | |
DE602006010870D1 (en) | PIPERIDINE DERIVATIVES SUITED AS ANTAGONISTS OF HISTAMINE H3 | |
NO20050429D0 (en) | Substituted quinoline CCR5 receptor antagonists | |
DK3059321T3 (en) | MICROARRAY SYNTHESIS AND COLLECTION OF LENGTH POLYNUCLEOTIDS | |
ATE409182T1 (en) | TETRAHYDROCINOLINONES AND THEIR USE AS ANTAGONISTS OF METABOTROPIC GLUTAMA RECEPTORS | |
NO20053530D0 (en) | Multivalent lymphotoxin-beta receptor antagonists and their use | |
DE60214996D1 (en) | ANTAGONISTS OF THE MCP-1 FUNCTION AND METHOD OF USE THEREOF | |
ATE344798T1 (en) | INDOLE DERIVATIVES SUITABLE AS HISTAMINE H3 ANTAGONISTS | |
DE60312659D1 (en) | LIGHT WEIGHT IDENTIFICATION OF INFORMATION | |
ATE413400T1 (en) | CGRP RECEPTOR ANTAGONISTS | |
ATE409700T1 (en) | CANNABINOID RECEPTOR LIGANDS AND THEIR USE | |
DE60317093D1 (en) | quinoline; ISOCHINOLIN AND CHINAZOLINE OXYALKYLAMIDES AND THEIR USE AS FUNGICIDES | |
DE60234167D1 (en) | BIPIPERIDIN DERIVATIVES AND THEIR USE AS INHIBITORS OF CHEMOKIN RECEPTORS | |
DE60321958D1 (en) | INDAZONE DERIVATIVES AND THEIR USE AS CRF ANTAGONISTS | |
DE602004014372D1 (en) | N-PYRROLIDIN-3-YL-AMIDE DERIVATIVES AS INHIBITORS OF SEROTONIN AND NORADRENALINE RECOVERY | |
DE60106607D1 (en) | SUBSTITUTED 1-AMINOALKYL-LACTAME AND THEIR USE AS MUSCARIN RECEPTOR ANTAGONISTS | |
DE60229673D1 (en) | HETEROCYCLIC SUBSTITUTED CARBONYL DERIVATIVES AND THEIR USE AS DOPAMINE D3 RECEPTOR LIGANDS | |
DE60334292D1 (en) | YELLOW COMPOSITION EMULSION COMPOSITION AND USE THEREOF | |
ATE438395T1 (en) | PYRAZOLE DERIVATIVES AND THEIR USE AS OREXIN RECEPTOR ANTAGONISTS | |
DE60318733D1 (en) | SUBSTITUTED BENZOXAZINONES AND THEIR USE | |
DE502004011575D1 (en) | Use of Dioldimerfettsäureestern | |
DK2336124T3 (en) | Stable hydrate of a muscarinic receptor antagonist | |
DE60206781D1 (en) | 2-SUBSTITUTED 1-ARYLPIPERAZINS AS TACHYKININ ANTAGONISTS AND / OR SEROTONIN RECOVERY INHIBITORS | |
DE602004031527D1 (en) | COMBINATION OF SEROTONIN RECOVERY INHIBITORS AND AGOMELATIN |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
8364 | No opposition during term of opposition |