DE60102137T2 - BETA-AMINIC ACID DERIVATIVES FOR USE AS MATRIX METALLOPROTEASES AND TNA ALPHA INHIBITORS - Google Patents
BETA-AMINIC ACID DERIVATIVES FOR USE AS MATRIX METALLOPROTEASES AND TNA ALPHA INHIBITORS Download PDFInfo
- Publication number
- DE60102137T2 DE60102137T2 DE60102137T DE60102137T DE60102137T2 DE 60102137 T2 DE60102137 T2 DE 60102137T2 DE 60102137 T DE60102137 T DE 60102137T DE 60102137 T DE60102137 T DE 60102137T DE 60102137 T2 DE60102137 T2 DE 60102137T2
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- Prior art keywords
- beta
- acid derivatives
- matrix metalloproteases
- alpha inhibitors
- aminic acid
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- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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- C07D—HETEROCYCLIC COMPOUNDS
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- C07D211/56—Nitrogen atoms
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Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US19018300P | 2000-03-17 | 2000-03-17 | |
US23546700P | 2000-09-26 | 2000-09-26 | |
US25206200P | 2000-11-20 | 2000-11-20 | |
PCT/US2001/008336 WO2001070734A2 (en) | 2000-03-17 | 2001-03-15 | Beta-amino acid derivatives as inhibitors of matrix metalloproteases and tnf-alpha |
Publications (2)
Publication Number | Publication Date |
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DE60102137D1 DE60102137D1 (en) | 2004-04-01 |
DE60102137T2 true DE60102137T2 (en) | 2004-10-21 |
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DE60102137T Expired - Lifetime DE60102137T2 (en) | 2000-03-17 | 2001-03-15 | BETA-AMINIC ACID DERIVATIVES FOR USE AS MATRIX METALLOPROTEASES AND TNA ALPHA INHIBITORS |
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US (1) | US6495565B2 (en) |
EP (1) | EP1263756B1 (en) |
JP (1) | JP2003528097A (en) |
CN (1) | CN1420881A (en) |
AR (1) | AR035174A1 (en) |
AT (1) | ATE260272T1 (en) |
AU (1) | AU2001250850A1 (en) |
BR (1) | BR0109469A (en) |
CA (1) | CA2400168A1 (en) |
DE (1) | DE60102137T2 (en) |
ES (1) | ES2215893T3 (en) |
HK (1) | HK1049334B (en) |
IL (1) | IL151018A0 (en) |
NZ (1) | NZ521245A (en) |
WO (1) | WO2001070734A2 (en) |
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AUPP982399A0 (en) | 1999-04-19 | 1999-05-13 | Fujisawa Pharmaceutical Co., Ltd. | Mmp inhibitor |
-
2001
- 2001-03-15 ES ES01924171T patent/ES2215893T3/en not_active Expired - Lifetime
- 2001-03-15 CA CA002400168A patent/CA2400168A1/en not_active Abandoned
- 2001-03-15 AU AU2001250850A patent/AU2001250850A1/en not_active Abandoned
- 2001-03-15 EP EP01924171A patent/EP1263756B1/en not_active Expired - Lifetime
- 2001-03-15 CN CN01806737A patent/CN1420881A/en active Pending
- 2001-03-15 DE DE60102137T patent/DE60102137T2/en not_active Expired - Lifetime
- 2001-03-15 JP JP2001568935A patent/JP2003528097A/en active Pending
- 2001-03-15 AT AT01924171T patent/ATE260272T1/en not_active IP Right Cessation
- 2001-03-15 NZ NZ521245A patent/NZ521245A/en unknown
- 2001-03-15 WO PCT/US2001/008336 patent/WO2001070734A2/en active IP Right Grant
- 2001-03-15 IL IL15101801A patent/IL151018A0/en unknown
- 2001-03-15 BR BR0109469-6A patent/BR0109469A/en active Pending
- 2001-03-16 AR ARP010101253A patent/AR035174A1/en unknown
- 2001-03-16 US US09/811,116 patent/US6495565B2/en not_active Expired - Lifetime
-
2003
- 2003-02-26 HK HK03101437.6A patent/HK1049334B/en not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
WO2001070734A3 (en) | 2002-03-14 |
ES2215893T3 (en) | 2004-10-16 |
EP1263756B1 (en) | 2004-02-25 |
AR035174A1 (en) | 2004-05-05 |
ATE260272T1 (en) | 2004-03-15 |
DE60102137D1 (en) | 2004-04-01 |
BR0109469A (en) | 2003-04-29 |
IL151018A0 (en) | 2003-02-12 |
HK1049334B (en) | 2004-07-16 |
AU2001250850A1 (en) | 2001-10-03 |
CA2400168A1 (en) | 2001-09-27 |
EP1263756A2 (en) | 2002-12-11 |
JP2003528097A (en) | 2003-09-24 |
US6495565B2 (en) | 2002-12-17 |
CN1420881A (en) | 2003-05-28 |
NZ521245A (en) | 2004-04-30 |
HK1049334A1 (en) | 2003-05-09 |
US20020013341A1 (en) | 2002-01-31 |
WO2001070734A2 (en) | 2001-09-27 |
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