DE3772423D1 - METHOD FOR PRODUCING MACROLIDE DERIVATIVES. - Google Patents

METHOD FOR PRODUCING MACROLIDE DERIVATIVES.

Info

Publication number
DE3772423D1
DE3772423D1 DE8787302663T DE3772423T DE3772423D1 DE 3772423 D1 DE3772423 D1 DE 3772423D1 DE 8787302663 T DE8787302663 T DE 8787302663T DE 3772423 T DE3772423 T DE 3772423T DE 3772423 D1 DE3772423 D1 DE 3772423D1
Authority
DE
Germany
Prior art keywords
macrolide derivatives
producing macrolide
producing
derivatives
macrolide
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE8787302663T
Other languages
German (de)
Inventor
Eddie Vi-Ping Tao
Jeffrey Thomas Vicenzi
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Eli Lilly and Co
Original Assignee
Eli Lilly and Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eli Lilly and Co filed Critical Eli Lilly and Co
Application granted granted Critical
Publication of DE3772423D1 publication Critical patent/DE3772423D1/en
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H5/00—Compounds containing saccharide radicals in which the hetero bonds to oxygen have been replaced by the same number of hetero bonds to halogen, nitrogen, sulfur, selenium, or tellurium
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
DE8787302663T 1986-03-31 1987-03-27 METHOD FOR PRODUCING MACROLIDE DERIVATIVES. Expired - Lifetime DE3772423D1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/846,446 US4921947A (en) 1986-03-31 1986-03-31 Process for preparing macrolide derivatives

Publications (1)

Publication Number Publication Date
DE3772423D1 true DE3772423D1 (en) 1991-10-02

Family

ID=25297965

Family Applications (1)

Application Number Title Priority Date Filing Date
DE8787302663T Expired - Lifetime DE3772423D1 (en) 1986-03-31 1987-03-27 METHOD FOR PRODUCING MACROLIDE DERIVATIVES.

Country Status (21)

Country Link
US (1) US4921947A (en)
EP (1) EP0240264B1 (en)
JP (1) JPH0710876B2 (en)
KR (1) KR900001166B1 (en)
CN (1) CN1018647B (en)
AR (1) AR247402A1 (en)
AT (1) ATE66678T1 (en)
AU (1) AU593894B2 (en)
CA (1) CA1292737C (en)
DE (1) DE3772423D1 (en)
DK (1) DK172935B1 (en)
EG (1) EG18550A (en)
ES (1) ES2028865T3 (en)
GR (1) GR3002764T3 (en)
HK (1) HK82492A (en)
HU (1) HU199864B (en)
IE (1) IE61018B1 (en)
IL (1) IL82005A (en)
NZ (1) NZ219784A (en)
PT (1) PT84561B (en)
ZA (1) ZA872201B (en)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2638458A1 (en) * 1988-10-27 1990-05-04 Adir NOVEL TYLOSIN DERIVATIVES, PROCESS FOR PREPARING THEM AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME
US5354708A (en) * 1992-06-04 1994-10-11 Taskar Nikhil R Method of nitrogen doping of II-VI semiconductor compounds during epitaxial growth using an amine
TW226373B (en) * 1992-07-15 1994-07-11 Pfizer
AU6019794A (en) * 1993-03-18 1994-10-11 Pfizer Inc. Antibacterial 16-membered ring macrolides containing olefins at c-20
WO1995002594A1 (en) * 1993-07-15 1995-01-26 Pfizer Inc. Amide derivatives of 16-membered ring antibiotic macrolides
ES2076107B1 (en) * 1993-09-20 1996-04-01 Pfizer DERIVATIVES OF MACROLID ANTIBIOTICS OF RINGS OF 16 MEMBERS.
EP0778283A3 (en) * 1995-12-05 1998-01-28 Pfizer Inc. Antibiotic macrolides
DE102004027417A1 (en) * 2004-06-04 2005-12-22 Basf Ag composite element
DK2455382T3 (en) 2005-12-13 2017-01-02 Incyte Holdings Corp Heteroberl substituted pyrrolo [2,3-b] pyridines and pyrrolo [2,3-b] pyrimidines as Janus kinase inhibitors
US8124744B2 (en) * 2006-05-01 2012-02-28 Taisho Pharmaceutical Co., Ltd. Macrolide derivatives
US8227429B2 (en) 2006-07-28 2012-07-24 Intervet International B.V. Macrolide synthesis process and solid-state forms
EP2019112A1 (en) * 2007-07-26 2009-01-28 Intervet International BV Macrolide solid-state forms
SI2089408T1 (en) * 2006-07-28 2012-02-29 Intervet Int Bv Macrolide synthesis process
US9034884B2 (en) 2010-11-19 2015-05-19 Incyte Corporation Heterocyclic-substituted pyrrolopyridines and pyrrolopyrimidines as JAK inhibitors
UA113156C2 (en) 2010-11-19 2016-12-26 CYCLOBUTYL-SUBSTITUTED PYROLOPYRIDINE AND PYROLOPYRIMIDINE DERIVATIVES AS JAK INHIBITORS
JP5876146B2 (en) 2011-06-20 2016-03-02 インサイト・ホールディングス・コーポレイションＩｎｃｙｔｅ Ｈｏｌｄｉｎｇｓ Ｃｏｒｐｏｒａｔｉｏｎ Azetidinylphenyl, pyridyl, or pyrazinylcarboxamide derivatives as JAK inhibitors
BR112014012585B1 (en) 2011-11-25 2021-05-25 Bayer Intellectual Property Gmbh compound comprising tylosin derivatives, method of preparation thereof and pharmaceutical or veterinary composition
CN102382159B (en) * 2011-12-07 2013-11-13 齐鲁动物保健品有限公司 Preparation method of tilmicosin
UA121532C2 (en) 2013-03-06 2020-06-10 Інсайт Холдінгс Корпорейшн METHODS AND INTERMEDIATES IN THE PREPARATION OF JAK INHIBITOR
TR201809189T4 (en) * 2013-05-23 2018-07-23 Bayer Animal Health Gmbh TYLOSIN DERIVATIVES AND METHOD FOR THEIR PREPARATION.
CN105837648B (en) * 2015-11-02 2018-07-06 湖北龙翔药业科技股份有限公司 A kind of preparation method of tilmicosin phosphate
CN108299531B (en) * 2018-01-23 2021-02-05 郑州大学 Methetavlosin pharmaceutical salt and preparation method thereof
CN111269275A (en) * 2020-03-09 2020-06-12 浙江康牧药业有限公司 Preparation method of tilmicosin
CN117304241B (en) * 2023-11-30 2024-03-01 中国农业科学院饲料研究所 Macrolide compound and preparation method and application thereof

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SI8110592A8 (en) * 1981-03-06 1996-06-30 Pliva Pharm & Chem Works Process for preparing of n-methyl-11-aza-10-deoxo-10-dihydroerythromycine a and derivatives thereof
JPS58146595A (en) * 1982-02-25 1983-09-01 Satoshi Omura Macrolide antibiotic
US4454314A (en) * 1982-08-02 1984-06-12 Pfizer Inc. Antibacterial mycaminosyl tylonolide and related macrolide derivatives
US4443436A (en) * 1982-09-13 1984-04-17 Eli Lilly And Company C-20-Modified macrolide derivatives of the macrolide antibiotics tylosin, desmycosin, macrocin, and lactenocin
IL69666A (en) * 1982-09-13 1987-10-20 Lilly Co Eli 20-amino-20-deoxo-5-o-mycaminosyl-23-o-mycinosyltylonolide derivatives,their preparation and veterinary antibiotic use
US4468511A (en) * 1983-02-28 1984-08-28 Eli Lilly And Company C-20- And C-23-Modified macrolide derivatives

Also Published As

Publication number Publication date
ZA872201B (en) 1988-10-26
GR3002764T3 (en) 1993-01-25
IE61018B1 (en) 1994-09-07
DK172935B1 (en) 1999-10-11
IE870796L (en) 1987-09-30
US4921947A (en) 1990-05-01
DK154087A (en) 1987-10-01
NZ219784A (en) 1989-01-27
EP0240264A3 (en) 1987-11-19
PT84561B (en) 1989-11-10
CN1018647B (en) 1992-10-14
CA1292737C (en) 1991-12-03
AR247402A1 (en) 1994-12-29
ATE66678T1 (en) 1991-09-15
HUT43087A (en) 1987-09-28
JPS62240681A (en) 1987-10-21
PT84561A (en) 1987-04-01
KR900001166B1 (en) 1990-02-27
JPH0710876B2 (en) 1995-02-08
AU593894B2 (en) 1990-02-22
CN87102397A (en) 1987-10-07
EG18550A (en) 1993-10-30
AU7067087A (en) 1987-10-08
HK82492A (en) 1992-10-30
IL82005A (en) 1991-08-16
KR870008906A (en) 1987-10-21
HU199864B (en) 1990-03-28
EP0240264A2 (en) 1987-10-07
ES2028865T3 (en) 1992-07-16
DK154087D0 (en) 1987-03-26
EP0240264B1 (en) 1991-08-28
IL82005A0 (en) 1987-10-20

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Legal Events

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