DE3683496D1 - PHOSPHITE AND PHOSPHATE BINDERS WITH AMINO FUNCTIONS, PRODUCTS RELATED TO YOU AND PHOSPHORAMIDITE PRE-PRODUCTS. - Google Patents
PHOSPHITE AND PHOSPHATE BINDERS WITH AMINO FUNCTIONS, PRODUCTS RELATED TO YOU AND PHOSPHORAMIDITE PRE-PRODUCTS.Info
- Publication number
- DE3683496D1 DE3683496D1 DE8686307285T DE3683496T DE3683496D1 DE 3683496 D1 DE3683496 D1 DE 3683496D1 DE 8686307285 T DE8686307285 T DE 8686307285T DE 3683496 T DE3683496 T DE 3683496T DE 3683496 D1 DE3683496 D1 DE 3683496D1
- Authority
- DE
- Germany
- Prior art keywords
- products
- phosphoramidite
- phosphite
- amino functions
- phosphate binders
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
Abstract
2-Substd,-3-protected- 1,3,2-oxazaphosphacycloalkanes of formula (I) are new. n= 2-4; R1 = protecting gp.; R2,R3 = H, 1-6C alkyl opt. substd. by electron-withdrawing substituents, lower cycloalkyl, 1-7C acyl, CN, halogen or NO2; R4 = alkyl, alkenyl, aryl, aralkyl or cycloalkyl contg. up to 10C. Bicyclic cpds. of formula (II) are new. m = 1-3; p = 0 or 1.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
PCT/US1986/001970 WO1988002004A1 (en) | 1985-08-26 | 1986-09-20 | Amino-derivatized phosphite and phosphate linking agents, phosphoramidite precursors, and useful conjugates |
EP86307285A EP0261283B2 (en) | 1985-08-26 | 1986-09-22 | Amino-derivatized phosphite and phosphate linking agents, phosphoramidite precursors and useful conjugates thereof |
Publications (1)
Publication Number | Publication Date |
---|---|
DE3683496D1 true DE3683496D1 (en) | 1992-02-27 |
Family
ID=8196151
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DE8686307285T Expired - Lifetime DE3683496D1 (en) | 1986-09-20 | 1986-09-22 | PHOSPHITE AND PHOSPHATE BINDERS WITH AMINO FUNCTIONS, PRODUCTS RELATED TO YOU AND PHOSPHORAMIDITE PRE-PRODUCTS. |
Country Status (1)
Country | Link |
---|---|
DE (1) | DE3683496D1 (en) |
-
1986
- 1986-09-22 DE DE8686307285T patent/DE3683496D1/en not_active Expired - Lifetime
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
8363 | Opposition against the patent | ||
8366 | Restricted maintained after opposition proceedings | ||
8327 | Change in the person/name/address of the patent owner |
Owner name: THE PERKIN-ELMER CORP. (N.D.GES.D.STAATES NEW YORK |
|
8327 | Change in the person/name/address of the patent owner |
Owner name: APPLERA CORP., FOSTER CITY, CALIF., US |
|
8339 | Ceased/non-payment of the annual fee |